Compile Data Set for Download or QSAR
maximum 50k data
Found 17 with Last Name = 'barbini' and Initial = 's'
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto Di Scienze E Tecnologie Molecolari (Istm)

Curated by ChEMBL
LigandPNGBDBM50240586(CHEMBL4098982)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto Di Scienze E Tecnologie Molecolari (Istm)

Curated by ChEMBL
LigandPNGBDBM32609(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 36b)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto Di Scienze E Tecnologie Molecolari (Istm)

Curated by ChEMBL
LigandPNGBDBM50240587(CHEMBL4070316)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto Di Scienze E Tecnologie Molecolari (Istm)

Curated by ChEMBL
LigandPNGBDBM50240589(CHEMBL4091245)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto Di Scienze E Tecnologie Molecolari (Istm)

Curated by ChEMBL
LigandPNGBDBM50240592(CHEMBL4097534)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto Di Scienze E Tecnologie Molecolari (Istm)

Curated by ChEMBL
LigandPNGBDBM50240588(CHEMBL4079500)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))TBA
LigandPNGBDBM50408492(CHEMBL5269133)
Affinity DataIC50:  407nMAssay Description:Antagonist activity at human muscarinic acetylcholine M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobi...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))TBA
LigandPNGBDBM50408498(CHEMBL5270983)
Affinity DataIC50:  518nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))TBA
LigandPNGBDBM50408502(CHEMBL5289168)
Affinity DataIC50:  729nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))TBA
LigandPNGBDBM50408500(CHEMBL5278611)
Affinity DataIC50:  972nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))TBA
LigandPNGBDBM50408497(CHEMBL5287933)
Affinity DataIC50:  1.42E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))TBA
LigandPNGBDBM50408493(CHEMBL5285672)
Affinity DataIC50:  1.99E+3nMAssay Description:Antagonist activity at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobi...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))TBA
LigandPNGBDBM50408496(CHEMBL5291421)
Affinity DataIC50:  1.99E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))TBA
LigandPNGBDBM50408495(CHEMBL5267130)
Affinity DataIC50:  2.59E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))TBA
LigandPNGBDBM50408499(CHEMBL5276647)
Affinity DataIC50:  2.95E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))TBA
LigandPNGBDBM50408494(CHEMBL5267106)
Affinity DataIC50:  3.14E+3nMAssay Description:Antagonist activity at human muscarinic acetylcholine M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobi...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))TBA
LigandPNGBDBM50408501(CHEMBL5283083)
Affinity DataIC50:  9.54E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed