TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
Affinity DataIC50: 407nMAssay Description:Antagonist activity at human muscarinic acetylcholine M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobi...More data for this Ligand-Target Pair
Affinity DataIC50: 518nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 729nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 972nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.42E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.99E+3nMAssay Description:Antagonist activity at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.99E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 2.59E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 2.95E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 3.14E+3nMAssay Description:Antagonist activity at human muscarinic acetylcholine M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobi...More data for this Ligand-Target Pair
Affinity DataIC50: 9.54E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair