Affinity DataKi: 6.70nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 144nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
Affinity DataKi: 224nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 398nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
Affinity DataKi: 806nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.16E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.36E+3nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.48E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.73E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.87E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.15E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.38E+3nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.83E+3nMAssay Description:Inhibition of dopamine D2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.04E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.47E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.58E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.90E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.18E+3nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.42E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.45E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.74E+3nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.10E+3nMAssay Description:Inhibition of dopamine D2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.57E+3nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.68E+3nMAssay Description:Inhibition of dopamine D2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.27E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.52E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.91E+3nMAssay Description:Inhibition of dopamine D2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of dopamine D2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of dopamine D2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of dopamine D2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of [3H]-Ro- 15-1788 binding to human GABA-A receptor alpha-5-beta-3-gamma-2 subunitsMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-1-beta-3-gamma-2More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-3-beta-3-gamma-2More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-2-beta-3-gamma-2More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Antagonist activity at P2X7 receptor in LPS-stimulated human THP1 cells assessed as inhibition of LPS/BzATP-induced IL-1beta release preincubated for...More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of [3H]-Ro- 15-1788 binding to human GABA-A receptor alpha-5-beta-3-gamma-2 subunitsMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-1-beta-3-gamma-2More data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-5-beta-3-gamma-2More data for this Ligand-Target Pair