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Found 80 with Last Name = 'barron' and Initial = 'ml'
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50327238(2-[2-(4'-Methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a...)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50327238(2-[2-(4'-Methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a...)
Affinity DataKi:  8.20nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131400(CHEMBL3634876)
Affinity DataKi:  28nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131380(CHEMBL3634878)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131380(CHEMBL3634878)
Affinity DataKi:  144nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131399(CHEMBL3634877)
Affinity DataKi:  224nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131399(CHEMBL3634877)
Affinity DataKi:  398nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131400(CHEMBL3634876)
Affinity DataKi:  806nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440989(CHEMBL2429890)
Affinity DataKi:  1.16E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440992(CHEMBL2432046)
Affinity DataKi:  1.36E+3nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440992(CHEMBL2432046)
Affinity DataKi:  1.48E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440990(CHEMBL2432051)
Affinity DataKi:  1.73E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440996(CHEMBL2432056)
Affinity DataKi:  1.87E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50334457(CHEMBL1643899 | N-(3-Fluorobenzyl)-8-aminopentacyc...)
Affinity DataKi:  2.15E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50334455(CHEMBL1643900 | N-(2-(3'-Fluorophenyl)ethyl)-8-ami...)
Affinity DataKi:  2.38E+3nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50401366(CHEMBL2205831)
Affinity DataKi:  2.83E+3nMAssay Description:Inhibition of dopamine D2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440995(CHEMBL2432058)
Affinity DataKi:  3.04E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440993(CHEMBL2432045)
Affinity DataKi:  3.47E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50401363(CHEMBL2205827)
Affinity DataKi:  3.58E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440991(CHEMBL2432048)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440989(CHEMBL2429890)
Affinity DataKi:  4.18E+3nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50334455(CHEMBL1643900 | N-(2-(3'-Fluorophenyl)ethyl)-8-ami...)
Affinity DataKi:  4.42E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50334456(CHEMBL1643902 | N-(2-(3'-Fluorophenyl)ethyl)-N-met...)
Affinity DataKi:  4.45E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440988(CHEMBL2432039)
Affinity DataKi:  4.74E+3nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440995(CHEMBL2432058)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibition of dopamine D2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440990(CHEMBL2432051)
Affinity DataKi:  5.57E+3nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440988(CHEMBL2432039)
Affinity DataKi:  5.68E+3nMAssay Description:Inhibition of dopamine D2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440988(CHEMBL2432039)
Affinity DataKi:  6.27E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440994(CHEMBL2432062)
Affinity DataKi:  8.52E+3nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50441001(CHEMBL2432049)
Affinity DataKi:  9.91E+3nMAssay Description:Inhibition of dopamine D2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50334456(CHEMBL1643902 | N-(2-(3'-Fluorophenyl)ethyl)-N-met...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50334458(CHEMBL1643901 | N-(3-Fluorobenzyl)-N-methyl-8-amin...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440999(CHEMBL2432052)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50441000(CHEMBL2432050)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of dopamine D2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440993(CHEMBL2432045)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440998(CHEMBL2432044)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440997(CHEMBL2432055)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131379(CHEMBL3634879)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131379(CHEMBL3634879)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50288954(11-benzyl-11-azahexacyclo[5.4.1.02,6.03,10.04,8.09...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50441002(CHEMBL2432047)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of dopamine D2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50440991(CHEMBL2432048)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of dopamine D2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50237730(CHEMBL4074449)
Affinity DataIC50:  2nMAssay Description:Inhibition of [3H]-Ro- 15-1788 binding to human GABA-A receptor alpha-5-beta-3-gamma-2 subunitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50237707(A-804598 | CHEMBL1628690)
Affinity DataIC50:  9nMAssay Description:Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-1-beta-3-gamma-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Mus musculus)
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50237707(A-804598 | CHEMBL1628690)
Affinity DataIC50:  9nMAssay Description:Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-3-beta-3-gamma-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50237707(A-804598 | CHEMBL1628690)
Affinity DataIC50:  9nMAssay Description:Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-2-beta-3-gamma-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50237707(A-804598 | CHEMBL1628690)
Affinity DataIC50:  9nMAssay Description:Antagonist activity at P2X7 receptor in LPS-stimulated human THP1 cells assessed as inhibition of LPS/BzATP-induced IL-1beta release preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50237730(CHEMBL4074449)
Affinity DataIC50:  18nMAssay Description:Inhibition of [3H]-Ro- 15-1788 binding to human GABA-A receptor alpha-5-beta-3-gamma-2 subunitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50237729(CHEMBL4088143)
Affinity DataIC50:  40nMAssay Description:Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-1-beta-3-gamma-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50237723(CHEMBL4089802)
Affinity DataIC50:  51nMAssay Description:Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-5-beta-3-gamma-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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