TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Hyderabad Campus
Curated by ChEMBL
University Of Hyderabad Campus
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of full length recombinant human SIRT1 expressed in Escherichia coli BL21 (DE3) PLysS using Fluor-de-Lys as substrate by fluorimetric assa...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Hyderabad Campus
Curated by ChEMBL
University Of Hyderabad Campus
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of full length recombinant human SIRT1 expressed in Escherichia coli BL21 (DE3) PLysS using Fluor-de-Lys as substrate by fluorimetric assa...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
University Of Hyderabad Campus
Curated by ChEMBL
University Of Hyderabad Campus
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human SIRT2More data for this Ligand-Target Pair
TargetSecreted chorismate mutase(Mycobacterium tuberculosis H37Rv)
University Of Hyderabad Campus
Curated by ChEMBL
University Of Hyderabad Campus
Curated by ChEMBL
Affinity DataIC50: 1.97E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis chorismate mutase expressed in Escherichia coli BL21 assessed as conversion of chorismate to prephenate afte...More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
University Of Hyderabad Campus
Curated by ChEMBL
University Of Hyderabad Campus
Curated by ChEMBL
Affinity DataEC50: 890nMAssay Description:Inhibition of PDE4B expressed in HEK293 cells assessed as fold reduction in forskolin-stimulated cAMP production pretreated for 30 mins measured 4 hr...More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
University Of Hyderabad Campus
Curated by ChEMBL
University Of Hyderabad Campus
Curated by ChEMBL
Affinity DataEC50: 220nMAssay Description:Inhibition of PDE4B expressed in HEK293 cells assessed as fold reduction in forskolin-stimulated cAMP production pretreated for 30 mins measured 4 hr...More data for this Ligand-Target Pair