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Found 50 with Last Name = 'basbaum' and Initial = 'ai'
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585913(CHEMBL5093295)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585914(CHEMBL5079273)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 1 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585912(CHEMBL5075486)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585909(CHEMBL5089996)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585911(CHEMBL5093969)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585910(CHEMBL5094012)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585918(CHEMBL5078567)
Affinity DataKi:  107nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585915(CHEMBL5082151)
Affinity DataKi:  208nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 1 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585919(CHEMBL5090584)
Affinity DataKi:  229nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585920(CHEMBL5092524)
Affinity DataKi:  271nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585916(CHEMBL5085238)
Affinity DataKi:  570nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 1 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585917(CHEMBL5091270)
Affinity DataKi:  705nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 1 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585908(CHEMBL1181770 | SB-699551)
Affinity DataKi: <2.00E+3nMAssay Description:Binding affinity to 5-HT3 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585908(CHEMBL1181770 | SB-699551)
Affinity DataKi: <2.00E+3nMAssay Description:Binding affinity to human 5-HT5ARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585908(CHEMBL1181770 | SB-699551)
Affinity DataKi: <2.00E+3nMAssay Description:Binding affinity to 5-HT2CR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585908(CHEMBL1181770 | SB-699551)
Affinity DataKi: <2.00E+3nMAssay Description:Binding affinity to 5-HT2BR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585908(CHEMBL1181770 | SB-699551)
Affinity DataKi: <2.00E+3nMAssay Description:Binding affinity to 5-HT2AR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585908(CHEMBL1181770 | SB-699551)
Affinity DataKi: <2.00E+3nMAssay Description:Binding affinity to 5-HT1DR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585908(CHEMBL1181770 | SB-699551)
Affinity DataKi: <2.00E+3nMAssay Description:Binding affinity to 5-HT1BR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585908(CHEMBL1181770 | SB-699551)
Affinity DataKi: <2.00E+3nMAssay Description:Binding affinity to 5-HT1AR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585922(CHEMBL5079940)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585901(CHEMBL3459329)
Affinity DataKi:  1.14E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585901(CHEMBL3459329)
Affinity DataKi:  1.15E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585905(CHEMBL5087322)
Affinity DataKi:  1.28E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585905(CHEMBL5087322)
Affinity DataKi:  1.29E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585903(CHEMBL5074821)
Affinity DataKi:  2.08E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585903(CHEMBL5074821)
Affinity DataKi:  2.09E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585902(CHEMBL5092728)
Affinity DataKi:  2.13E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585902(CHEMBL5092728)
Affinity DataKi:  2.14E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585904(CHEMBL5093652)
Affinity DataKi:  2.88E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585904(CHEMBL5093652)
Affinity DataKi:  2.88E+4nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 100 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585913(CHEMBL5093295)
Affinity DataIC50:  4.57E+8nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585909(CHEMBL5089996)
Affinity DataIC50:  4.57E+8nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585911(CHEMBL5093969)
Affinity DataIC50:  4.68E+8nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585917(CHEMBL5091270)
Affinity DataIC50:  4.68E+8nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 1 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585914(CHEMBL5079273)
Affinity DataIC50:  4.79E+8nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 1 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585916(CHEMBL5085238)
Affinity DataIC50:  4.79E+8nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 1 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585906(CHEMBL5077128)
Affinity DataIC50:  4.79E+8nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585919(CHEMBL5090584)
Affinity DataIC50:  4.79E+8nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585915(CHEMBL5082151)
Affinity DataIC50:  4.79E+8nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 1 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585910(CHEMBL5094012)
Affinity DataIC50:  4.90E+8nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585918(CHEMBL5078567)
Affinity DataIC50:  5.01E+8nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585920(CHEMBL5092524)
Affinity DataIC50:  5.13E+8nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585921(CHEMBL5087602)
Affinity DataIC50:  5.13E+8nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585912(CHEMBL5075486)
Affinity DataIC50:  5.13E+8nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor at 32 uM incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585907(CHEMBL5082447)
Affinity DataIC50:  5.25E+8nMAssay Description:Displacement of [3H]-5-CT from human 5-HT5A receptor incubated for 2 hr by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585907(CHEMBL5082447)
Affinity DataEC50:  3.63E+3nMAssay Description:Agonist activity at human 5-HT5A receptor transfected in HTLA cells assessed as increase in beta-arrestin 2 recruitment at 10 uM incubated for 18 to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50585906(CHEMBL5077128)
Affinity DataEC50:  355nMAssay Description:Agonist activity at human 5-HT5A receptor transfected in HTLA cells assessed as increase in beta-arrestin 2 recruitment at 10 uM incubated for 18 to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
Florence University

Curated by ChEMBL
LigandPNGBDBM50242402(4-Hydroxynonenal | 4-hydroxy-2-nonenal | CHEMBL454...)
Affinity DataEC50:  2.70E+4nMAssay Description:Agonist activity at rat TRPA1 channel expressed in tetracycline induced HEK293 cells assessed as increase in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
Florence University

Curated by ChEMBL
LigandPNGBDBM50242402(4-Hydroxynonenal | 4-hydroxy-2-nonenal | CHEMBL454...)
Affinity DataEC50:  7.70E+4nMAssay Description:Activation of TRPA1 channel in rat dorsal root ganglion neurons assessed as increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed