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Found 60 with Last Name = 'bastos' and Initial = 'mm'
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM50137117(CHEMBL3754535)
Affinity DataIC50:  1nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM50137118(CHEMBL3753575)
Affinity DataIC50:  1nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM50137116(CHEMBL378856)
Affinity DataIC50:  2nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM50137113(CHEMBL3753096)
Affinity DataIC50:  6nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM50137112(CHEMBL309896)
Affinity DataIC50:  12nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM2899((4S)-6-chloro-4-[(E)-2-cyclopropylethenyl]-4-(trif...)
Affinity DataIC50:  23nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM27577(5-[(3-ethyl-5-fluoro-1H-indazol-4-yl)oxy]benzene-1...)
Affinity DataIC50:  25nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM2898((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataIC50:  32nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataIC50:  38nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataIC50:  40nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 recombinant reverse transcriptase expressed in Escherichia coli...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM2955(GW420867X | HBY1293 | propan-2-yl (2S)-2-ethyl-7-f...)
Affinity DataIC50:  45nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM2912((3S,5S)-7-chloro-5-[(E)-2-cyclopropylethenyl]-3-me...)
Affinity DataIC50:  46nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM27576(5-[(5-fluoro-3-methyl-1H-indazol-4-yl)oxy]benzene-...)
Affinity DataIC50:  50nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM50137114(CHEMBL3753238)
Affinity DataIC50:  56nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM50137119(CHEMBL3753009)
Affinity DataIC50:  59nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM2906((3S,5S)-7-chloro-5-(2-cyclopropylethynyl)-3-methyl...)
Affinity DataIC50:  82nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataIC50:  500nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 recombinant reverse transcriptase expressed in Escherichia coli...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM50137120(CHEMBL3753006)
Affinity DataIC50:  800nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM50137115(CHEMBL3754170)
Affinity DataIC50:  950nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM93122(3-Hydroxy-2-oxo-3-trifluoromethylindole, 25)
Affinity DataIC50:  3.41E+3nMAssay Description:Biological assay using HIV-1 reverse transcriptase.More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM93122(3-Hydroxy-2-oxo-3-trifluoromethylindole, 25)
Affinity DataIC50:  3.41E+3nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM93121(3-Hydroxy-2-oxo-3-trifluoromethylindole, 21)
Affinity DataIC50:  3.61E+3nMAssay Description:Biological assay using HIV-1 reverse transcriptase.More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM93121(3-Hydroxy-2-oxo-3-trifluoromethylindole, 21)
Affinity DataIC50:  3.61E+3nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM93119(3-Hydroxy-2-oxo-3-trifluoromethylindole, 16)
Affinity DataIC50:  6.07E+3nMAssay Description:Biological assay using HIV-1 reverse transcriptase.More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM93119(3-Hydroxy-2-oxo-3-trifluoromethylindole, 16)
Affinity DataIC50:  6.07E+3nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM93120(3-Hydroxy-2-oxo-3-trifluoromethylindole, 18)
Affinity DataIC50:  7.10E+3nMAssay Description:Biological assay using HIV-1 reverse transcriptase.More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM93120(3-Hydroxy-2-oxo-3-trifluoromethylindole, 18)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM93123(3-Hydroxy-2-oxo-3-trifluoromethylindole, 26)
Affinity DataIC50:  8.37E+3nMAssay Description:Biological assay using HIV-1 reverse transcriptase.More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase(Human immunodeficiency virus 1)
Instituto De Tecnologia Em F£Rmacos

Curated by ChEMBL
LigandPNGBDBM93123(3-Hydroxy-2-oxo-3-trifluoromethylindole, 26)
Affinity DataIC50:  8.37E+3nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301952((3S,6S,9S,12S,15S,21S)-21-(2-((S)-2-amino-3-(1H-im...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonist activity at PTHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301952((3S,6S,9S,12S,15S,21S)-21-(2-((S)-2-amino-3-(1H-im...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonist activity at GIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301952((3S,6S,9S,12S,15S,21S)-21-(2-((S)-2-amino-3-(1H-im...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonist activity at PTHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301952((3S,6S,9S,12S,15S,21S)-21-(2-((S)-2-amino-3-(1H-im...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonist activity at glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301952((3S,6S,9S,12S,15S,21S)-21-(2-((S)-2-amino-3-(1H-im...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonist activity at GIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301935((3S,6S,9S,12S,15S,21S)-21-((S)-2-((S)-2-amino-3-(1...)
Affinity DataEC50:  480nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of intracellular [3H]cAMP accumulation after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301931((4S)-4-[(2S)-2-[(2S)-2-amino-3-(1H-imidazol-5-yl)p...)
Affinity DataEC50:  545nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of intracellular [3H]cAMP accumulation after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301937((3S,6S,9S,12S,15S,21S)-21-((S)-2-((S)-2-amino-3-(1...)
Affinity DataEC50:  390nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of intracellular [3H]cAMP accumulation after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301938((3S,6S,9S,12S,15S,21S)-21-((S)-2-((S)-2-amino-3-(1...)
Affinity DataEC50:  270nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of intracellular [3H]cAMP accumulation after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301939((3S,6S,9S,12S,15S,21S)-21-((S)-2-((S)-2-amino-3-(1...)
Affinity DataEC50:  430nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of intracellular [3H]cAMP accumulation after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301940((3S,6S,9S,12S,15S,21S)-21-((S)-2-((S)-2-amino-3-(1...)
Affinity DataEC50:  148nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of intracellular [3H]cAMP accumulation after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301941((3S,6S,9S,12S,15S,21S)-21-((S)-2-((S)-2-amino-3-(1...)
Affinity DataEC50:  87nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of intracellular [3H]cAMP accumulation after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301942((3S,6S,9S,12S,15S,21S)-21-((S)-2-((S)-2-amino-3-(1...)
Affinity DataEC50:  95nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of intracellular [3H]cAMP accumulation after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301943((3S,6S,9S,12S,15S,21S)-21-((S)-2-((S)-2-amino-3-(1...)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of intracellular [3H]cAMP accumulation after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301944((3S,6S,9S,12S,15S,21S)-21-((S)-2-((S)-2-amino-3-(1...)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of intracellular [3H]cAMP accumulation after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301945((3S,6S,9S,12S,15S,21S)-21-((S)-2-((S)-2-amino-3-(1...)
Affinity DataEC50:  93nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of intracellular [3H]cAMP accumulation after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301946((3S,6S,9S,12S,15S,21S)-21-((S)-2-((S)-2-amino-3-(1...)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of intracellular [3H]cAMP accumulation after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301947((3S,6S,9S,12S,15S,21S)-21-((S)-2-((S)-2-amino-3-(1...)
Affinity DataEC50:  965nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of intracellular [3H]cAMP accumulation after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301948((3S,6S,9S,12S,15S,21S)-21-((S)-2-((S)-2-amino-3-(1...)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of intracellular [3H]cAMP accumulation after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301949(CHEMBL583264)
Affinity DataEC50:  0.0340nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of intracellular [3H]cAMP accumulation after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301950((3S,6S,9S,12S,15S,21S)-21-((S)-2-((S)-2-amino-3-(1...)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at human GLP1R expressed in CHO cells assessed as stimulation of intracellular [3H]cAMP accumulation after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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