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Found 31 with Last Name = 'baudy-floc''h' and Initial = 'm'
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50347818(CHEMBL1802413 | P518)
Affinity DataIC50:  1.30nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50069792((2S)-2-[(2S)-2-acetamido-4-methylpentanamido]-N-[(...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against Calpain I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396422(CHEMBL2170403)
Affinity DataIC50:  1.99E+3nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396420(CHEMBL2170390)
Affinity DataIC50:  2.99E+3nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50347830(CHEMBL1802425)
Affinity DataIC50:  8.73E+3nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396417(CHEMBL2170395)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as inhibition of human 26RFa-induced increase in intracell...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396419(CHEMBL2170393)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as inhibition of human 26RFa-induced increase in intracell...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396418(CHEMBL2170394)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as inhibition of human 26RFa-induced increase in intracell...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396416(CHEMBL2170398)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as inhibition of human 26RFa-induced increase in intracell...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50159149(CHEMBL179042 | Peptidyl boronic acid derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50159158(CHEMBL433563 | Peptidyl boronic acid derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50159149(CHEMBL179042 | Peptidyl boronic acid derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against Calpain I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50159158(CHEMBL433563 | Peptidyl boronic acid derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against Calpain I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50347830(CHEMBL1802425)
Affinity DataEC50:  739nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50347818(CHEMBL1802413 | P518)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396425(CHEMBL2170400)
Affinity DataEC50:  1.37E+3nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396426(CHEMBL2170399)
Affinity DataEC50:  2.98E+4nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396431(CHEMBL2170389)
Affinity DataEC50:  429nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396430(CHEMBL2170391)
Affinity DataEC50:  2.34E+3nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396429(CHEMBL2170392)
Affinity DataEC50:  1.09E+3nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396419(CHEMBL2170393)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396418(CHEMBL2170394)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396417(CHEMBL2170395)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396428(CHEMBL2170396)
Affinity DataEC50:  341nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396424(CHEMBL2170401)
Affinity DataEC50:  382nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396423(CHEMBL2170402)
Affinity DataEC50:  164nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396421(CHEMBL2170249)
Affinity DataEC50:  138nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396416(CHEMBL2170398)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396427(CHEMBL2170397)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396422(CHEMBL2170403)
Affinity DataEC50:  94nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396420(CHEMBL2170390)
Affinity DataEC50:  136nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed