TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against Calpain I activityMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 1.99E+3nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 2.99E+3nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 8.73E+3nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as inhibition of human 26RFa-induced increase in intracell...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as inhibition of human 26RFa-induced increase in intracell...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as inhibition of human 26RFa-induced increase in intracell...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as inhibition of human 26RFa-induced increase in intracell...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against Factor XaMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against Factor XaMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against Calpain I activityMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against Calpain I activityMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 739nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 1.37E+3nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 2.98E+4nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 429nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 2.34E+3nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 1.09E+3nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 341nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 382nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 164nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 138nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 1.10E+3nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 94nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataEC50: 136nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair