Affinity DataKi: 2.60nMAssay Description:Displacement of [125I]NT from rat NTR1 transfected in mouse LTK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 238nMAssay Description:Binding affinity to NTR3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 7.70E+3nMAssay Description:Antagonist activity at P2X7 in Sprague-Dawley rat synaptosome assessed as inhibition of BzATP-induced [3H]D-aspartate efflux compound preincubated fo...More data for this Ligand-Target Pair