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Found 84 with Last Name = 'bazzicalupi' and Initial = 'c'
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50091345(CHEMBL2092861)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530219(CHEMBL4454983)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530219(CHEMBL4454983)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50091347(CHEMBL71429)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530216(CHEMBL4582201)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530216(CHEMBL4582201)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50091336(CHEMBL3582266)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50221885((S)-1,1-Dimethyl-2-quinolin-6-yl-pyrrolidinium; io...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50091338(CHEMBL3582264)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50221885((S)-1,1-Dimethyl-2-quinolin-6-yl-pyrrolidinium; io...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50221887(1,1-dimethyl-2-quinolin-6-yl-pyrrolidinium iodide ...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530217(CHEMBL4550498)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530217(CHEMBL4550498)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50091341(CHEMBL3582261)
Affinity DataKi:  63nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50221882((R)-1,1-Dimethyl-2-quinolin-6-yl-pyrrolidinium; io...)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]alpha-bungarotoxin from alpha7 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50221883((S)-6-(1-methylpyrrolidin-2-yl)-quinoline | CHEMBL...)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50091342(CHEMBL3582260)
Affinity DataKi:  98nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530222(CHEMBL4440670)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530222(CHEMBL4440670)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50221883((S)-6-(1-methylpyrrolidin-2-yl)-quinoline | CHEMBL...)
Affinity DataKi:  124nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50412250(CHEMBL128168)
Affinity DataKi:  126nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50221884(CHEMBL243666 | rac-6-(1-methylpyrrolidin-2-yl)quin...)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50221888(CHEMBL390227 | trimethyl-(4-quinolin-6-yl-but-3-yn...)
Affinity DataKi:  142nMAssay Description:Displacement of [3H]alpha-bungarotoxin from alpha7 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50091344(CHEMBL3582258)
Affinity DataKi:  155nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50091335(CHEMBL3582267)
Affinity DataKi:  195nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50221882((R)-1,1-Dimethyl-2-quinolin-6-yl-pyrrolidinium; io...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530224(CHEMBL4552618)
Affinity DataKi:  227nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530224(CHEMBL4552618)
Affinity DataKi:  227nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50412260(CHEMBL273485)
Affinity DataKi:  309nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530215(CHEMBL4475133)
Affinity DataKi:  352nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530215(CHEMBL4475133)
Affinity DataKi:  352nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  450nMAssay Description:Displacement of [3H]alpha-bungarotoxin from alpha7 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50091340(CHEMBL3582262)
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50091339(CHEMBL3582263)
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530220(CHEMBL4438099)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530221(CHEMBL4522629)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530223(CHEMBL4547457)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530218(CHEMBL4515416)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530223(CHEMBL4547457)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530225(CHEMBL4574804)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530226(CHEMBL4448467)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530220(CHEMBL4438099)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530218(CHEMBL4515416)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530226(CHEMBL4448467)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530221(CHEMBL4522629)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50530225(CHEMBL4574804)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50091337(CHEMBL3582265)
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50221882((R)-1,1-Dimethyl-2-quinolin-6-yl-pyrrolidinium; io...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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