Affinity DataKi: 1.10nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 6.80nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Displacement of [3H]alpha-bungarotoxin from alpha7 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 98nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 116nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 116nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 124nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 132nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 142nMAssay Description:Displacement of [3H]alpha-bungarotoxin from alpha7 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 195nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 227nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 227nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 309nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 352nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 352nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:Displacement of [3H]alpha-bungarotoxin from alpha7 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 1.05E+3nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Florence
Curated by ChEMBL
University Of Florence
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cerebral cortexMore data for this Ligand-Target Pair