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Found 37 with Last Name = 'becquart' and Initial = 'j'
LigandPNGBDBM50058202((S)-2-[(2-{(S)-2-[((R)-2-Amino-3-mercapto-propiony...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of Human farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50284949((S)-2-{[(S)-2-((S)-2-{[(S)-2-((R)-2,6-Diamino-hexa...)
Affinity DataIC50:  5nMAssay Description:Inhibition of farnesyl transferase (FTase) of rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50403479(CHEMBL2115457)
Affinity DataIC50:  20nMAssay Description:Inhibition of farnesyl transferase (FTase) of rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50059852((S)-2-((S)-2-((S)-2-((R)-2-amino-3-mercaptopropyla...)
Affinity DataIC50:  21nMAssay Description:In vitro inhibiion of bovine farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50284165((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propyl...)
Affinity DataIC50:  23nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay under reducing (+DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50284951((S)-2-[((S)-2-{(S)-2-[(S)-2-((R)-2,6-Diamino-hexan...)
Affinity DataIC50:  40nMAssay Description:Inhibition of farnesyl transferase (FTase) of rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285838(CHEMBL89836 | Pseudopeptide derivative)
Affinity DataIC50:  50nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  57nMAssay Description:In vitro inhibiion of bovine farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticleMMDB

LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  60nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay in non-reducing (-DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails ArticleMMDB

LigandPNGBDBM50285846((S)-2-({(S)-2-[2-(2-Mercapto-ethylamino)-acetyl]-1...)
Affinity DataIC50:  100nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285842(CHEMBL420801 | Pseudopeptide derivative)
Affinity DataIC50:  145nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285837((S)-2-({(S)-2-[2-(2-Mercapto-ethylamino)-acetyl]-1...)
Affinity DataIC50:  290nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50284952((S)-2-((S)-2-{(S)-2-[(S)-2-((R)-2,6-Diamino-hexano...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of farnesyl transferase (FTase) of rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50284950((S)-2-((S)-2-{(S)-2-[(S)-2-((R)-2,6-Diamino-hexano...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of farnesyl transferase (FTase) of rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50284948((S)-2-[(S)-2-((S)-2-{[(S)-2-((R)-2,6-Diamino-hexan...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of farnesyl transferase (FTase) of rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50284953((S)-2-[(S)-2-((S)-2-{[(S)-2-((R)-2,6-Diamino-hexan...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of farnesyl transferase (FTase) of rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibition of Human farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticleMMDB

LigandPNGBDBM50285845(2-({2-[(2-Mercapto-ethylcarbamoyl)-methyl]-1,2,3,4...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50403478(CHEMBL2115458)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of farnesyl transferase (FTase) of rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50403477(CHEMBL2115025)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of farnesyl transferase (FTase) of rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50403477(CHEMBL2115025)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of farnesyl transferase (FTase) of rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of farnesyl transferase (FTase) of rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50213274(CHEMBL3350314)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of farnesyl transferase (FTase) of rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50213274(CHEMBL3350314)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of farnesyl transferase (FTase) of rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285840(CHEMBL412576 | Pseudopeptide derivative)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285842(CHEMBL420801 | Pseudopeptide derivative)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay under reducing (+DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285843((S)-2-[((S)-2-{2-[tert-Butoxycarbonyl-(2-mercapto-...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50213273(CHEMBL3350692)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of farnesyl transferase (FTase) of rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285841(CHEMBL262383 | Pseudopeptide derivative)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285842(CHEMBL420801 | Pseudopeptide derivative)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay in non-reducing (-DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285839((S)-2-[((S)-2-{2-[tert-Butoxycarbonyl-(2-mercapto-...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285838(CHEMBL89836 | Pseudopeptide derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay under reducing (+DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285841(CHEMBL262383 | Pseudopeptide derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay in non-reducing (-DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285838(CHEMBL89836 | Pseudopeptide derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibiion of bovine farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285840(CHEMBL412576 | Pseudopeptide derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay under reducing (+DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285841(CHEMBL262383 | Pseudopeptide derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibiion of bovine farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285840(CHEMBL412576 | Pseudopeptide derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay in non-reducing (-DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails Article