Affinity DataKi: 4.50E+3nMAssay Description:Competitive inhibition of human recombinant DPP4 using AP-pNA as substrate preincubated for 30 mins followed by substrate addition measured after 30 ...More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Competitive inhibition of human recombinant DPP4 using AP-pNA as substrate preincubated for 30 mins followed by substrate addition measured after 30 ...More data for this Ligand-Target Pair
Affinity DataKi: 6.30E+3nMAssay Description:Competitive inhibition of human recombinant DPP4 using AP-pNA as substrate preincubated for 30 mins followed by substrate addition measured after 30 ...More data for this Ligand-Target Pair
Affinity DataKi: 6.10E+4nMAssay Description:Competitive inhibition of human recombinant DPP4 using AP-pNA as substrate preincubated for 30 mins followed by substrate addition measured after 30 ...More data for this Ligand-Target Pair
Affinity DataKi: 1.42E+5nMAssay Description:Competitive inhibition of human recombinant DPP4 using AP-pNA as substrate preincubated for 30 mins followed by substrate addition measured after 30 ...More data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Displacement of [125I]-exendin (9 to 39) from human GLP-1R expressed in African green monkey COS7 cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 5.10nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 6.60nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 6.60nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 7.60nMAssay Description:Displacement of [125I]-exendin (9 to 39) from human GLP-1R expressed in African green monkey COS7 cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Displacement of [125I]-exendin (9 to 39) from human GLP-1R expressed in African green monkey COS7 cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 113nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 229nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 9.20E+3nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataIC50: 9.20E+3nMAssay Description:Displacement of [125I]exendin(9-39) from human GLP1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataEC50: 0.170nMAssay Description:Agonist activity at human GLP-1R expressed in African green monkey COS7 cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataEC50: 0.0120nMAssay Description:Activation of human GLP1R expressed in HEK293 cells assessed as effect on cAMP responsive element promoter driven luciferase expressionMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataEC50: 8.30nMAssay Description:Activation of human GLP1R expressed in HEK293 cells assessed as effect on cAMP responsive element promoter driven luciferase expressionMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataEC50: 0.00360nMAssay Description:Activation of human GLP1R expressed in HEK293 cells assessed as effect on cAMP responsive element promoter driven luciferase expressionMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Activation of human GLP1R expressed in HEK293 cells assessed as effect on cAMP responsive element promoter driven luciferase expressionMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University Of Texas At Dallas
Curated by ChEMBL
University Of Texas At Dallas
Curated by ChEMBL
Affinity DataEC50: 0.380nMAssay Description:Activation of human GLP1R expressed in HEK293 cells assessed as effect on cAMP responsive element promoter driven luciferase expressionMore data for this Ligand-Target Pair