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Found 72 with Last Name = 'belei' and Initial = 'd'
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50092365((R)-1-((1H-imidazol-5-yl)methyl)-3-benzyl-4-(thiop...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of human FTaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50067584((S)-2-{[5-((R)-2-Amino-3-mercapto-propylamino)-bip...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50189292(CHEMBL3828157)
Affinity DataIC50:  9nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50189293(CHEMBL3827279)
Affinity DataIC50:  23nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50189295(CHEMBL3828384)
Affinity DataIC50:  155nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50059863((Z)-2-Methyl-3-tetradecyl-but-2-enedioic acid | CH...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50059863((Z)-2-Methyl-3-tetradecyl-but-2-enedioic acid | CH...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50189304(CHEMBL3827991)
Affinity DataIC50:  602nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489184(CHEMBL2312764)
Affinity DataIC50:  630nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489185(CHEMBL2312763)
Affinity DataIC50:  650nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50189297(CHEMBL3828545)
Affinity DataIC50:  711nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50189301(CHEMBL3827237)
Affinity DataIC50:  726nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50189302(CHEMBL3827637)
Affinity DataIC50:  931nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489194(CHEMBL2312766)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489198(CHEMBL2312765)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50485345(CHEMBL2046656)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of partially purified human recombinant FTase measured for 15 mins by automated fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50036274(CHEMBL3361086)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50189300(CHEMBL3826996)
Affinity DataIC50:  1.32E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50485343(CHEMBL2046655)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of partially purified human recombinant FTase measured for 15 mins by automated fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50036270(CHEMBL3361094)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50189303(CHEMBL3828130)
Affinity DataIC50:  2.33E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50035931(CHEMBL3361085)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489199(CHEMBL2312491)
Affinity DataIC50:  3.18E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50485735(CHEMBL2159815)
Affinity DataIC50:  3.35E+3nMAssay Description:Inhibition of recombinant human FTase using dansyl-GCVLS as substrate after 15 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50485736(CHEMBL2159814)
Affinity DataIC50:  3.73E+3nMAssay Description:Inhibition of recombinant human FTase using dansyl-GCVLS as substrate after 15 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50036277(CHEMBL3361077)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489183(CHEMBL2312770)
Affinity DataIC50:  4.67E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50498791(CHEMBL3623716)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of recombinant human FTase using FPP/dansyl-GCVLS as substrate measured for 15 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489197(CHEMBL2312492)
Affinity DataIC50:  4.92E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50485344(CHEMBL2046654)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of partially purified human recombinant FTase measured for 15 mins by automated fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489200(CHEMBL2312771)
Affinity DataIC50:  5.33E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50036276(CHEMBL3361076)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489186(CHEMBL2312499)
Affinity DataIC50:  6.36E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489191(CHEMBL2312496)
Affinity DataIC50:  7.01E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489192(CHEMBL2312500)
Affinity DataIC50:  7.27E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50036272(CHEMBL3361092)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50485342(CHEMBL2046652)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of partially purified human recombinant FTase measured for 15 mins by automated fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50485346(CHEMBL2046653)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of partially purified human recombinant FTase measured for 15 mins by automated fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50189299(CHEMBL3828274)
Affinity DataIC50:  8.74E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489187(CHEMBL2312497)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489188(CHEMBL2312495)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50035927(CHEMBL3361080)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50189294(CHEMBL3827132)
Affinity DataIC50:  1.16E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50498787(CHEMBL3623718)
Affinity DataIC50:  1.17E+4nMAssay Description:Inhibition of recombinant human FTase using FPP/dansyl-GCVLS as substrate measured for 15 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50498792(CHEMBL3623720)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of recombinant human FTase using FPP/dansyl-GCVLS as substrate measured for 15 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489196(CHEMBL2312493)
Affinity DataIC50:  1.31E+4nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489195(CHEMBL2312498)
Affinity DataIC50:  1.37E+4nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50035929(CHEMBL3361082)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50035921(CHEMBL3361071)
Affinity DataIC50:  1.48E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
'Al. I. Cuza' University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50035926(CHEMBL3361079)
Affinity DataIC50:  1.49E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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