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Found 93 with Last Name = 'belle' and Initial = 'c'
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50205807(CHEMBL3978212)
Affinity DataKi:  350nMAssay Description:Inhibition of recombinant human tyrosinase expressed in baculovirus infected Sf9 cells assessed as diphenolase activity using L-DOPA as substrate by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50205815(CHEMBL3907670)
Affinity DataKi:  1.02E+3nMAssay Description:Inhibition of recombinant human tyrosinase expressed in baculovirus infected Sf9 cells assessed as diphenolase activity using L-DOPA as substrate by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50205806(CHEMBL3969839)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of recombinant human tyrosinase expressed in baculovirus infected Sf9 cells assessed as diphenolase activity using L-DOPA as substrate by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50205814(CHEMBL3898657)
Affinity DataKi:  1.28E+5nMAssay Description:Inhibition of recombinant human tyrosinase expressed in baculovirus infected Sf9 cells assessed as diphenolase activity using L-DOPA as substrate by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Univ. Grenoble-Alpes/Cnrs

Curated by ChEMBL
LigandPNGBDBM50031467(5-HYDROXY-2-(HYDROXYMETHYL)-4H-PYRAN-4-ONE | 5-Hyd...)
Affinity DataKi:  3.50E+5nMAssay Description:Inhibition of recombinant human tyrosinase expressed in baculovirus infected Sf9 cells assessed as diphenolase activity using L-DOPA as substrate by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369335(CHEMBL1201841)
Affinity DataIC50:  2.20nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate compared with finasteride in experiment 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50057290((5aS,7aS,10aS,10bS)-7a-Methyl-1,5a,6,7,7a,9,10,10a...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50057297((5aS,7aS,8S,10aS,10bS)-8-Hydroxy-7a-methyl-3,4,6,7...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50057289((5aS,7aS,10aS,10bS,12aS)-7a-Methyl-tetradecahydro-...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369338(CHEMBL1237294)
Affinity DataIC50:  3nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50334788((17beta-(N-tert-butylcarbamoyl)-4-aza-5alpha-andro...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50057292((5aS,7aS,10aS,10bS)-7a-Methyl-3,4,5a,6,7,7a,9,10,1...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369336(CHEMBL1237306)
Affinity DataIC50:  4.10nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369335(CHEMBL1201841)
Affinity DataIC50:  4.30nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate compared with finasteride in experiment 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50057295((5aS,7aS,8S,10aS,10bS)-7a-Methyl-2-oxo-2,3,4,5a,6,...)
Affinity DataIC50:  5.5nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369335(CHEMBL1201841)
Affinity DataIC50:  5.70nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate compared with finasteride in experiment 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369334(CHEMBL1237307)
Affinity DataIC50:  6.10nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369337(CHEMBL1794821)
Affinity DataIC50:  6.10nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369335(CHEMBL1201841)
Affinity DataIC50:  7.30nMAssay Description:Tested against 5 alpha R-2 on human prostate homogenate from surgically derived benign hyperplastic tissue in experiment 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369335(CHEMBL1201841)
Affinity DataIC50:  10nMAssay Description:Tested against 5 alpha R-2 on human prostate homogenate from surgically derived benign hyperplastic tissue in experiment 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369335(CHEMBL1201841)
Affinity DataIC50:  37nMAssay Description:Inhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissue in experiment 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50334788((17beta-(N-tert-butylcarbamoyl)-4-aza-5alpha-andro...)
Affinity DataIC50:  42nMAssay Description:Inhibitory activity against human 5-alpha Reductase-1 expressed in DU-145 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369335(CHEMBL1201841)
Affinity DataIC50:  122nMAssay Description:TInhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissue in experiment 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369335(CHEMBL1201841)
Affinity DataIC50:  127nMAssay Description:Inhibitory activity against human 5-alpha Reductase-1 expressed in DU-145 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369335(CHEMBL1201841)
Affinity DataIC50:  150nMAssay Description:Tested against 5 alpha R-2 on human prostate homogenate from surgically derived benign hyperplastic tissue in experiment 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369336(CHEMBL1237306)
Affinity DataIC50:  263nMAssay Description:Inhibitory activity against human 5-alpha Reductase-1 expressed in DU-145 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50057292((5aS,7aS,10aS,10bS)-7a-Methyl-3,4,5a,6,7,7a,9,10,1...)
Affinity DataIC50:  299nMAssay Description:Inhibitory activity against human 5-alpha Reductase-1 expressed in DU-145 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50057297((5aS,7aS,8S,10aS,10bS)-8-Hydroxy-7a-methyl-3,4,6,7...)
Affinity DataIC50:  409nMAssay Description:Inhibitory activity against human 5-alpha Reductase-1 expressed in DU-145 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50057295((5aS,7aS,8S,10aS,10bS)-7a-Methyl-2-oxo-2,3,4,5a,6,...)
Affinity DataIC50:  460nMAssay Description:Inhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50057295((5aS,7aS,8S,10aS,10bS)-7a-Methyl-2-oxo-2,3,4,5a,6,...)
Affinity DataIC50:  1.13E+3nMAssay Description:Inhibitory activity against human 5-alpha Reductase-1 expressed in DU-145 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase III PolC-type(Staphylococcus aureus)
Targanta Therapeutics

Curated by ChEMBL
LigandPNGBDBM50177653(5-allyl-6-chloro-2-(2,3-dihydro-1H-inden-5-ylamino...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase III PolC-type(Staphylococcus aureus)
Targanta Therapeutics

Curated by ChEMBL
LigandPNGBDBM50177648(2-(2,3-dihydro-1H-inden-5-ylamino)-6-hydroxy-5-(3-...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369338(CHEMBL1237294)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase III PolC-type(Staphylococcus aureus)
Targanta Therapeutics

Curated by ChEMBL
LigandPNGBDBM50177654(4-(3-(2-(2,3-dihydro-1H-inden-5-ylamino)-4-hydroxy...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase III PolC-type(Staphylococcus aureus)
Targanta Therapeutics

Curated by ChEMBL
LigandPNGBDBM50177644(2-(2,3-dihydro-1H-inden-5-ylamino)-6-hydroxy-5-(3-...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase III PolC-type(Staphylococcus aureus)
Targanta Therapeutics

Curated by ChEMBL
LigandPNGBDBM50177645(2-(2,3-dihydro-1H-inden-5-ylamino)-6-hydroxy-5-(3-...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase III PolC-type(Staphylococcus aureus)
Targanta Therapeutics

Curated by ChEMBL
LigandPNGBDBM50177651(5-benzyl-2-(3-ethyl-4-methylphenylamino)-6-hydroxy...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50057297((5aS,7aS,8S,10aS,10bS)-8-Hydroxy-7a-methyl-3,4,6,7...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50057292((5aS,7aS,10aS,10bS)-7a-Methyl-3,4,5a,6,7,7a,9,10,1...)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369336(CHEMBL1237306)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50369336(CHEMBL1237306)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase III PolC-type(Staphylococcus aureus)
Targanta Therapeutics

Curated by ChEMBL
LigandPNGBDBM50177657(2-(2,3-dihydro-1H-inden-5-ylamino)-6-hydroxy-5-(3-...)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase III PolC-type(Staphylococcus aureus)
Targanta Therapeutics

Curated by ChEMBL
LigandPNGBDBM50177647(4-(3-(2-(2,3-dihydro-1H-inden-5-ylamino)-4-hydroxy...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
National University Of La Plata (Unlp)

Curated by ChEMBL
LigandPNGBDBM50378783(CLOFAZIMINE)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine in absence of 0.01% TritonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Universit£

Curated by ChEMBL
LigandPNGBDBM50350995(CHEMBL1818876)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of diphenolase activity of mushroom tyrosinase using L-DOPA as substrate preincubated for 5 mins by spectroscopic methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Universit£

Curated by ChEMBL
LigandPNGBDBM50351005(CHEMBL1818886)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of diphenolase activity of mushroom tyrosinase using L-DOPA as substrate preincubated for 5 mins by spectroscopic methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase III PolC-type(Staphylococcus aureus)
Targanta Therapeutics

Curated by ChEMBL
LigandPNGBDBM50177665(5-allyl-2-(3-ethyl-4-methylphenylamino)-6-hydroxyp...)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Universit£

Curated by ChEMBL
LigandPNGBDBM50350996(CHEMBL1818877)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of diphenolase activity of mushroom tyrosinase using L-DOPA as substrate preincubated for 5 mins by spectroscopic methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Universit£

Curated by ChEMBL
LigandPNGBDBM50350993(CHEMBL1818874)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of diphenolase activity of mushroom tyrosinase using L-DOPA as substrate preincubated for 5 mins by spectroscopic methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase III PolC-type(Staphylococcus aureus)
Targanta Therapeutics

Curated by ChEMBL
LigandPNGBDBM50177656(5-(3-(4-aminophenoxy)propyl)-2-(2,3-dihydro-1H-ind...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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