Affinity DataKi: 350nMAssay Description:Inhibition of recombinant human tyrosinase expressed in baculovirus infected Sf9 cells assessed as diphenolase activity using L-DOPA as substrate by ...More data for this Ligand-Target Pair
Affinity DataKi: 1.02E+3nMAssay Description:Inhibition of recombinant human tyrosinase expressed in baculovirus infected Sf9 cells assessed as diphenolase activity using L-DOPA as substrate by ...More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of recombinant human tyrosinase expressed in baculovirus infected Sf9 cells assessed as diphenolase activity using L-DOPA as substrate by ...More data for this Ligand-Target Pair
Affinity DataKi: 1.28E+5nMAssay Description:Inhibition of recombinant human tyrosinase expressed in baculovirus infected Sf9 cells assessed as diphenolase activity using L-DOPA as substrate by ...More data for this Ligand-Target Pair
Affinity DataKi: 3.50E+5nMAssay Description:Inhibition of recombinant human tyrosinase expressed in baculovirus infected Sf9 cells assessed as diphenolase activity using L-DOPA as substrate by ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate compared with finasteride in experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate compared with finasteride in experiment 3More data for this Ligand-Target Pair
Affinity DataIC50: 5.5nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
Affinity DataIC50: 5.70nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate compared with finasteride in experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMAssay Description:Inhibition against 5 alpha R-2 in human prostate homogenate relative to finasterideMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30nMAssay Description:Tested against 5 alpha R-2 on human prostate homogenate from surgically derived benign hyperplastic tissue in experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Tested against 5 alpha R-2 on human prostate homogenate from surgically derived benign hyperplastic tissue in experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissue in experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibitory activity against human 5-alpha Reductase-1 expressed in DU-145 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 122nMAssay Description:TInhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissue in experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 127nMAssay Description:Inhibitory activity against human 5-alpha Reductase-1 expressed in DU-145 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Tested against 5 alpha R-2 on human prostate homogenate from surgically derived benign hyperplastic tissue in experiment 3More data for this Ligand-Target Pair
Affinity DataIC50: 263nMAssay Description:Inhibitory activity against human 5-alpha Reductase-1 expressed in DU-145 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 299nMAssay Description:Inhibitory activity against human 5-alpha Reductase-1 expressed in DU-145 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 409nMAssay Description:Inhibitory activity against human 5-alpha Reductase-1 expressed in DU-145 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 460nMAssay Description:Inhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibitory activity against human 5-alpha Reductase-1 expressed in DU-145 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibitory activity against 5-alpha Reductase-2 on human prostate homogenates from surgically derived benign hyperplastic tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine in absence of 0.01% TritonMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of diphenolase activity of mushroom tyrosinase using L-DOPA as substrate preincubated for 5 mins by spectroscopic methodMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of diphenolase activity of mushroom tyrosinase using L-DOPA as substrate preincubated for 5 mins by spectroscopic methodMore data for this Ligand-Target Pair
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of diphenolase activity of mushroom tyrosinase using L-DOPA as substrate preincubated for 5 mins by spectroscopic methodMore data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of diphenolase activity of mushroom tyrosinase using L-DOPA as substrate preincubated for 5 mins by spectroscopic methodMore data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of DNA polymerase3C from Staphylococcus aureusMore data for this Ligand-Target Pair