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Found 43 with Last Name = 'bellotti' and Initial = 'm'
TargetLanC-like protein 2(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50041087(CHEMBL3355910)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of ABA binding to LANCL2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123364(CHEMBL3622696)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123399(CHEMBL3623254)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123399(CHEMBL3623254)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123364(CHEMBL3622696)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123357(CHEMBL3622695)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123400(CHEMBL3623256)
Affinity DataIC50:  7.70E+4nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123404(CHEMBL3623250)
Affinity DataIC50:  8.20E+4nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123364(CHEMBL3622696)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibition of human SIRT2 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123400(CHEMBL3623256)
Affinity DataIC50:  1.02E+5nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50017341(CHEMBL3288034)
Affinity DataIC50:  1.06E+5nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50017341(CHEMBL3288034)
Affinity DataIC50:  1.14E+5nMAssay Description:Inhibition of human SIRT2 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123451(CHEMBL3623255)
Affinity DataIC50:  1.27E+5nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50017341(CHEMBL3288034)
Affinity DataIC50:  1.36E+5nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123372(CHEMBL3623251)
Affinity DataIC50:  1.37E+5nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123372(CHEMBL3623251)
Affinity DataIC50:  1.37E+5nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123357(CHEMBL3622695)
Affinity DataIC50:  1.59E+5nMAssay Description:Inhibition of human SIRT2 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123357(CHEMBL3622695)
Affinity DataIC50:  2.38E+5nMAssay Description:Inhibition of human SIRT1 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123403(CHEMBL3623259)
Affinity DataIC50:  2.42E+5nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123399(CHEMBL3623254)
Affinity DataIC50:  2.42E+5nMAssay Description:Inhibition of human SIRT2 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123401(CHEMBL3623257)
Affinity DataIC50:  2.70E+5nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123401(CHEMBL3623257)
Affinity DataIC50:  2.75E+5nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123403(CHEMBL3623259)
Affinity DataIC50:  2.97E+5nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123452(CHEMBL3623260)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50017341(CHEMBL3288034)
Affinity DataIC50:  3.14E+5nMAssay Description:Inhibition of human SIRT1 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123364(CHEMBL3622696)
Affinity DataIC50:  4.24E+5nMAssay Description:Inhibition of human SIRT1 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123402(CHEMBL3623258)
Affinity DataIC50:  4.41E+5nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123448(CHEMBL3623253)
Affinity DataIC50:  5.17E+5nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123405(CHEMBL3623252)
Affinity DataIC50:  2.87E+6nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123399(CHEMBL3623254)
Affinity DataIC50:  6.52E+6nMAssay Description:Inhibition of human SIRT1 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108523(CHEMBL3597889)
Affinity DataEC50:  5.70E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as iodide influx after 24 hrs by HS-YFP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50105909(CHEMBL3597937)
Affinity DataEC50:  1.50E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108483(CHEMBL3597841)
Affinity DataEC50:  3.40E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108350(CHEMBL3597884)
Affinity DataEC50:  9.50E+3nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108513(CHEMBL3597853)
Affinity DataEC50:  5.30E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108496(CHEMBL3597875)
Affinity DataEC50:  7.10E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50105911(CHEMBL3597886)
Affinity DataEC50:  5.80E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108492(CHEMBL3597874)
Affinity DataEC50:  6.40E+3nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50105910(CHEMBL3597907)
Affinity DataEC50:  3.20E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108517(CHEMBL3597843)
Affinity DataEC50:  2.70E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108302(CHEMBL3597927)
Affinity DataEC50:  1.40E+4nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as iodide influx after 24 hrs by HS-YFP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108513(CHEMBL3597853)
Affinity DataEC50:  5.30E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as iodide influx after 24 hrs by HS-YFP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108301(CHEMBL3597882)
Affinity DataEC50:  8.50E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as iodide influx after 24 hrs by HS-YFP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed