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Found 131 with Last Name = 'berger' and Initial = 'v'
TargetNeutral alpha-glucosidase AB(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi:  14nMpH: 6.0Assay Description:Competitive Inhibition constant of the compound was determined on rice alpha Glucosidase at pH 8.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutral alpha-glucosidase AB(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280031((6S,7R,8R)-Octahydro-indolizine-1,6,7,8-tetraol | ...)
Affinity DataKi:  15nMpH: 5.0Assay Description:Competitive Inhibition constant of the compound was determined on yeast alpha Glucosidase at pH 7.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutral alpha-glucosidase AB(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi:  160nMpH: 5.0Assay Description:Competitive Inhibition constant of the compound was determined on yeast alpha Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280031((6S,7R,8R)-Octahydro-indolizine-1,6,7,8-tetraol | ...)
Affinity DataKi:  900nMpH: 5.0Assay Description:Competitive Inhibition constant of the compound was determined on Asp. Wentii beta Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280031((6S,7R,8R)-Octahydro-indolizine-1,6,7,8-tetraol | ...)
Affinity DataKi:  1.50E+3nMpH: 5.0Assay Description:Competitive Inhibition constant of the compound was determined on almonds beta Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutral alpha-glucosidase AB(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280029((2R,3R,4R,5S)-2-(1-Hydroxy-propyl)-piperidine-3,4,...)
Affinity DataKi:  3.00E+3nMpH: 7.0Assay Description:Competitive Inhibition constant of the compound was determined on yeast alpha Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutral alpha-glucosidase AB(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280030((2S,3R,4R,5S)-2-Fluoromethyl-piperidine-3,4,5-trio...)
Affinity DataKi:  8.00E+3nMpH: 8.0Assay Description:Competitive Inhibition constant of the compound was determined on yeast alpha Glucosidase at pH 7.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutral alpha-glucosidase AB(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280030((2S,3R,4R,5S)-2-Fluoromethyl-piperidine-3,4,5-trio...)
Affinity DataKi:  1.50E+4nMpH: 5.0Assay Description:Competitive Inhibition constant of the compound was determined on yeast alpha Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutral alpha-glucosidase AB(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi:  2.10E+4nMpH: 7.0Assay Description:Competitive Inhibition constant of the compound was determined on yeast alpha Glucosidase at pH 7.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutral alpha-glucosidase AB(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi:  2.30E+4nMpH: 6.0Assay Description:Competitive Inhibition constant of the compound was determined on yeast alpha Glucosidase at pH 6.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutral alpha-glucosidase AB(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280030((2S,3R,4R,5S)-2-Fluoromethyl-piperidine-3,4,5-trio...)
Affinity DataKi:  2.90E+4nMpH: 6.0Assay Description:Competitive Inhibition constant of the compound was determined on rice alpha Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280029((2R,3R,4R,5S)-2-(1-Hydroxy-propyl)-piperidine-3,4,...)
Affinity DataKi:  4.20E+4nMpH: 5.0Assay Description:Competitive Inhibition constant of the compound was determined on Asp. Wentii beta Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutral alpha-glucosidase AB(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280030((2S,3R,4R,5S)-2-Fluoromethyl-piperidine-3,4,5-trio...)
Affinity DataKi:  4.70E+4nMpH: 7.0Assay Description:Competitive Inhibition constant of the compound was determined on yeast alpha Glucosidase at pH 7.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutral alpha-glucosidase AB(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280030((2S,3R,4R,5S)-2-Fluoromethyl-piperidine-3,4,5-trio...)
Affinity DataKi:  4.70E+4nMpH: 7.0Assay Description:Competitive Inhibition constant of the compound was determined on Asp. Wentii beta Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutral alpha-glucosidase AB(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280029((2R,3R,4R,5S)-2-(1-Hydroxy-propyl)-piperidine-3,4,...)
Affinity DataKi:  6.00E+4nMpH: 6.0Assay Description:Competitive Inhibition constant of the compound was determined on almonds beta Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi:  3.00E+5nMpH: 5.0Assay Description:Competitive Inhibition constant of the compound was determined on yeast alpha Glucosidase at pH 7.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi:  3.00E+5nMpH: 5.0Assay Description:Competitive Inhibition constant of the compound was determined on almonds beta Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280030((2S,3R,4R,5S)-2-Fluoromethyl-piperidine-3,4,5-trio...)
Affinity DataKi:  3.80E+5nMpH: 5.0Assay Description:Competitive Inhibition constant of the compound was determined on Asp. Wentii beta Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutral alpha-glucosidase AB(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi:  4.60E+5nMpH: 5.0Assay Description:Competitive Inhibition constant of the compound was determined on rice alpha Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280030((2S,3R,4R,5S)-2-Fluoromethyl-piperidine-3,4,5-trio...)
Affinity DataKi:  6.00E+5nMpH: 5.0Assay Description:Competitive Inhibition constant of the compound was determined on yeast alpha Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280029((2R,3R,4R,5S)-2-(1-Hydroxy-propyl)-piperidine-3,4,...)
Affinity DataKi:  6.30E+5nMpH: 5.0Assay Description:Competitive Inhibition constant of the compound was determined on almonds beta Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280032((2R,3R,4R,5S)-2-Methyl-piperidine-3,4,5-triol | 1,...)
Affinity DataKi:  7.80E+5nMpH: 5.0Assay Description:Competitive Inhibition constant of the compound was determined on almonds beta Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutral alpha-glucosidase AB(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280031((6S,7R,8R)-Octahydro-indolizine-1,6,7,8-tetraol | ...)
Affinity DataKi: >1.50E+6nMpH: 5.0Assay Description:Competitive Inhibition constant of the compound was determined on rice alpha Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutral alpha-glucosidase AB(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280032((2R,3R,4R,5S)-2-Methyl-piperidine-3,4,5-triol | 1,...)
Affinity DataKi:  1.56E+6nMpH: 7.0Assay Description:Competitive Inhibition constant of the compound was determined on yeast alpha Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutral alpha-glucosidase AB(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280029((2R,3R,4R,5S)-2-(1-Hydroxy-propyl)-piperidine-3,4,...)
Affinity DataKi:  2.00E+6nMpH: 7.0Assay Description:Competitive Inhibition constant of the compound was determined on yeast alpha Glucosidase at pH 5.0More data for this Ligand-Target Pair
In DepthDetails Article
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078118(CHEMBL3417524)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078123(CHEMBL3417526)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078080(CHEMBL3417520)
Affinity DataIC50:  1.30nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078053(CHEMBL3417414)
Affinity DataIC50:  1.40nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078078(CHEMBL3417518)
Affinity DataIC50:  1.60nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078119(CHEMBL3417525)
Affinity DataIC50:  1.70nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078035(CHEMBL3417429)
Affinity DataIC50:  1.90nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078077(CHEMBL3417517)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078146(CHEMBL3417531)
Affinity DataIC50:  2.10nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078052(CHEMBL3417415)
Affinity DataIC50:  2.20nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078036(CHEMBL3417428)
Affinity DataIC50:  2.30nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078040(CHEMBL3417425)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078033(CHEMBL3417431)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078038(CHEMBL3417427)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078043(CHEMBL3417422)
Affinity DataIC50:  2.5nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078031(CHEMBL3417508)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078115(CHEMBL3417522)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078045(CHEMBL3417421)
Affinity DataIC50:  2.90nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078141(CHEMBL3417527)
Affinity DataIC50:  2.90nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078145(CHEMBL3417530)
Affinity DataIC50:  3.10nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078060(CHEMBL3417511)
Affinity DataIC50:  3.5nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078059(CHEMBL3417510)
Affinity DataIC50:  3.60nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078058(CHEMBL3417509)
Affinity DataIC50:  3.60nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078042(CHEMBL3417423)
Affinity DataIC50:  4.70nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50078050(CHEMBL3417417)
Affinity DataIC50:  5.70nMAssay Description:Displacement of [125I]-L-691831 from human FLAP expressed in insect SF9 cell membranes after 2 hrs by Topcount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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