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Found 91 with Last Name = 'bermejo' and Initial = 'a'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50298707(1-Benzyl-6-chloro-7-hydroxy-1,2,3,4-tetrahydroisoq...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50298706(1-Butyl-6-chloro-7-hydroxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50022051(1-Phenyl-6-chloro-7-hydroxy-N-methyl-1,2,3,4-tetra...)
Affinity DataKi:  504nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50291655((R)-3-{(2R,11R)-2,11-Dihydroxy-11-[(2S,5R,2'S,5'R)...)
Affinity DataIC50:  0.330nMAssay Description:Concentration required for the inhibition of NADH oxidase in submitochondrial particles from beef heartMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291654((R)-3-{(2R,13R)-2,13-Dihydroxy-13-[(2S,5R,2'S,5'R)...)
Affinity DataIC50:  0.580nMAssay Description:Concentration required for the inhibition of NADH oxidase in submitochondrial particles from beef heartMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291656((R)-3-{(R)-13-Hydroxy-13-[(2S,5R,2'S,5'R)-5'-((S)-...)
Affinity DataIC50:  0.580nMAssay Description:Concentration required for the inhibition of NADH oxidase in submitochondrial particles from beef heartMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50135518((R)-5-{(S)-11-Hydroxy-11-[(2S,5S)-5-((S)-1-hydroxy...)
Affinity DataIC50:  0.700nMAssay Description:Inhibitory activity against NADH oxidase in beef heart mitochondrial complex I.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135523((S)-3-{(2R,13S)-2,13-Dihydroxy-13-[(2S,5S)-5-((S)-...)
Affinity DataIC50:  0.800nMAssay Description:Inhibitory activity against NADH oxidase in beef heart mitochondrial complex I.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135528((R)-5-{(6S,11S)-6,11-Dihydroxy-11-[(2S,5S)-5-((S)-...)
Affinity DataIC50:  1.90nMAssay Description:Inhibitory activity against NADH oxidase in beef heart mitochondrial complex I.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135520((S)-5-Methyl-3-{(2R,8S,13S)-2,8,13-trihydroxy-13-[...)
Affinity DataIC50:  2.30nMAssay Description:Inhibitory activity against NADH oxidase in beef heart mitochondrial complex I.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135522((S)-3-{(2R,13S)-2,13-Dihydroxy-8-[(Z)-hydroxyimino...)
Affinity DataIC50:  2.70nMAssay Description:Inhibitory activity against NADH oxidase in beef heart mitochondrial complex I.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135519((R)-5-{(6S,11S)-6,11-Dihydroxy-11-[(2S,5S)-5-((S)-...)
Affinity DataIC50:  3.30nMAssay Description:Inhibitory activity against NADH oxidase in beef heart mitochondrial complex I.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135526((S)-5-Methyl-3-{(2R,8S,13S)-2,8,13-trihydroxy-13-[...)
Affinity DataIC50:  3.60nMAssay Description:Inhibitory activity against NADH oxidase in beef heart mitochondrial complex I.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135527((-)-cis-rotenone | (-)-rotenone | (2R,6aS,12aS)-8,...)
Affinity DataIC50:  5.10nMAssay Description:Inhibitory activity against NADH oxidase in beef heart mitochondrial complex I.More data for this Ligand-Target Pair
LigandPNGBDBM50135521((R)-5-{(6S,11S)-6,11-Dihydroxy-11-[(2S,5S)-5-((S)-...)
Affinity DataIC50:  5.80nMAssay Description:Inhibitory activity against NADH oxidase in beef heart mitochondrial complex I.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135524((S)-3,4-Dihydroxy-5-methyl-3-{(2R,8S,13S)-2,8,13-t...)
Affinity DataIC50:  22nMAssay Description:Inhibitory activity against NADH oxidase in beef heart mitochondrial complex I.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135525((S)-3-{(2R,13S)-8-[2-(3-Benzyloxy-4-methoxy-phenyl...)
Affinity DataIC50: >150nMAssay Description:Inhibitory activity against NADH oxidase in beef heart mitochondrial complex I.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataIC50:  200nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50005548((+)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinol...)
Affinity DataIC50:  200nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50202322((-)-anonaine | (R)-6,7,7a,8-tetrahydro-5H-benzo[g]...)
Affinity DataIC50:  800nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292474(7-(10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-ylam...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292466(CHEMBL450147 | CHEMBL507970 | Dimethylgrisabine)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50202300((R)-4-methoxy-6,7,7a,8-tetrahydro-5H-benzo[g][1,3]...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50089611((1-Benzyl-6-benzyloxy-7-methoxy-3,4-dihydro-1H-iso...)
Affinity DataIC50:  1.69E+3nMAssay Description:Inhibitory concentration against NADH oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292445(CHEMBL508011 | Isopiline)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50089614(1-Benzyl-6-benzyloxy-7-methoxy-2-methyl-1,2,3,4-te...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibitory concentration against NADH oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50089613(1-Benzyl-6-benzyloxy-7-methoxy-3,4-dihydro-isoquin...)
Affinity DataIC50:  2.91E+3nMAssay Description:Inhibitory concentration against NADH oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292467(Antioquine | Antioquine (S,R) | CHEMBL446564 | CHE...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50099789(5-Benzyl-5,6,7,8-tetrahydro-[1,3]dioxolo[4,5-g]iso...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of [3H]-dopamine uptake in rat striatal synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50089612(1-Benzyl-6-benzyloxy-7-methoxy-1,2,3,4-tetrahydro-...)
Affinity DataIC50:  3.88E+3nMAssay Description:Inhibitory concentration against NADH oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50068644(Acetic acid (2R,3R,4R,5R,6R)-3-acetoxy-5,6-diethox...)
Affinity DataIC50:  3.90E+3nMAssay Description:Compound was tested for NADH oxidase activity in bovine heart submitochondrial particlesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50241642((+)-Obaberine | CHEMBL451211 | CHEMBL464525 | Obab...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50099789(5-Benzyl-5,6,7,8-tetrahydro-[1,3]dioxolo[4,5-g]iso...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of [3H]-Raclopride binding to the rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292468(CHEMBL504757 | Isotetrandrine)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50068645((4R,5S,6S,7S,8R)-4,5-Diethoxy-6,7-dihydroxy-8-phen...)
Affinity DataIC50:  4.40E+3nMAssay Description:Compound was tested for NADH oxidase activity in bovine heart submitochondrial particlesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50022723((+)-(S)-amphetamine | (+)-alpha-methylphenethylami...)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292469(CHEMBL443081 | CHEMBL501861 | O-methyldauricine)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50099787(5-Benzyl-5,6,7,8-tetrahydro-[1,3]dioxolo[4,5-g]iso...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of [3H]-dopamine uptake in rat striatal synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50202287((R)-6,7,7a,8-tetrahydro-5H-benzo[g][1,3]dioxolo[4'...)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50241641((+)-Homoaromoline | CHEMBL509855 | Homoaromoline |...)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292454(CHEMBL508081 | secocularidine)
Affinity DataIC50:  1.34E+4nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292463((1S)-1-(4-hydroxybenzyl)-6-methoxy-1,2,3,4-tetrahy...)
Affinity DataIC50:  1.41E+4nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50099786(1-Benzyl-2-propyl-1,2,3,4-tetrahydro-isoquinoline-...)
Affinity DataIC50:  1.47E+4nMAssay Description:Inhibition of [3H]-Raclopride binding to the rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292446((S)-1,10-Dimethoxy-5,6,6a,7-tetrahydro-4H-dibenzo[...)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50099786(1-Benzyl-2-propyl-1,2,3,4-tetrahydro-isoquinoline-...)
Affinity DataIC50:  1.66E+4nMAssay Description:Inhibition of [3H]-SCH- 23390 binding to the rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50292470(CHEMBL447018 | Dimethylpseudoxandrine)
Affinity DataIC50:  2.01E+4nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50099788(5-Benzyl-6-propyl-5,6,7,8-tetrahydro-[1,3]dioxolo[...)
Affinity DataIC50:  2.03E+4nMAssay Description:Inhibition of [3H]-dopamine uptake in rat striatal synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50099788(5-Benzyl-6-propyl-5,6,7,8-tetrahydro-[1,3]dioxolo[...)
Affinity DataIC50:  2.19E+4nMAssay Description:Inhibition of [3H]-Raclopride binding to the rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50202290(2,3-dimethoxy-7,7-dimethyl-7H-dibenzo[de,g]quinoli...)
Affinity DataIC50:  2.36E+4nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50099789(5-Benzyl-5,6,7,8-tetrahydro-[1,3]dioxolo[4,5-g]iso...)
Affinity DataIC50:  2.39E+4nMAssay Description:Inhibition of [3H]-SCH- 23390 binding to the rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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