TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Inhibition of [3H]R-PIA binding to Adenosine A1 receptor from rat brain membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Rattus norvegicus)
Experimental Sugar Cane Station&Quot;Villa Clara-Cienfuegos&Quot
Curated by ChEMBL
Experimental Sugar Cane Station&Quot;Villa Clara-Cienfuegos&Quot
Curated by ChEMBL
Affinity DataKi: 54.1nMAssay Description:Displacement of radioligand [125I]AB-MECA binding at rat A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Rattus norvegicus)
Experimental Sugar Cane Station&Quot;Villa Clara-Cienfuegos&Quot
Curated by ChEMBL
Experimental Sugar Cane Station&Quot;Villa Clara-Cienfuegos&Quot
Curated by ChEMBL
Affinity DataKi: 107nMAssay Description:Displacement of radioligand [125I]AB-MECA binding at rat A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Rattus norvegicus)
Experimental Sugar Cane Station&Quot;Villa Clara-Cienfuegos&Quot
Curated by ChEMBL
Experimental Sugar Cane Station&Quot;Villa Clara-Cienfuegos&Quot
Curated by ChEMBL
Affinity DataKi: 155nMAssay Description:Displacement of radioligand [125I]AB-MECA binding at rat A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 247nMAssay Description:Inhibition of [3H]R-PIA binding to Adenosine A1 receptor from rat brain membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 292nMAssay Description:Inhibition of [3H]R-PIA binding to Adenosine A1 receptor from rat brain membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Rattus norvegicus)
Experimental Sugar Cane Station&Quot;Villa Clara-Cienfuegos&Quot
Curated by ChEMBL
Experimental Sugar Cane Station&Quot;Villa Clara-Cienfuegos&Quot
Curated by ChEMBL
Affinity DataKi: 405nMAssay Description:Displacement of radioligand [125I]AB-MECA binding at rat A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 725nMAssay Description:Inhibition of [3H]R-PIA binding to Adenosine A1 receptor from rat brain membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 901nMAssay Description:Inhibition of [3H]R-PIA binding to Adenosine A1 receptor from rat brain membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Displacement of [3H]R-N6-phenylisopropyladenosine from adenosine A1 receptor in rat cerebral cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 8.12E+3nMAssay Description:Displacement of [3H]R-N6-phenylisopropyladenosine from adenosine A1 receptor in rat cerebral cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 1.44E+4nMAssay Description:Inhibition of [3H]R-PIA binding to Adenosine A1 receptor from rat brain membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 2.55E+4nMAssay Description:Displacement of [3H]R-N6-phenylisopropyladenosine from adenosine A1 receptor in rat cerebral cortical membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Experimental Sugar Cane Station
Curated by ChEMBL
Experimental Sugar Cane Station
Curated by ChEMBL
Affinity DataKi: 3.23E+4nMAssay Description:Displacement of [3H]R-N6-phenylisopropyladenosine from adenosine A1 receptor in rat cerebral cortical membraneMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 2.16E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 2.64E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 3.05E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 5.35E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 6.56E+3nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 7.54E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 1.29E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 1.76E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 1.92E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 2.27E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 3.01E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade De Vigo
Curated by ChEMBL
Universidade De Vigo
Curated by ChEMBL
Affinity DataIC50: 6.87E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...More data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 5.50E+3nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 13nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 80nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 560nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 4.50E+4nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 6.50E+4nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 3.50E+3nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 8.80E+4nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 230nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 1.80E+4nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 1.72E+3nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 800nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 2.30E+3nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 1.10E+3nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as PLC-mediated [3H]IP productionMore data for this Ligand-Target Pair