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Found 59 with Last Name = 'bezverkov' and Initial = 'r'
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143361((S)-N*4*-Acridin-9-yl-N*1*,N*1*-diethyl-heptane-1,...)
Affinity DataIC50:  9nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145324((2-m-Tolyl-ethyl)-[6-(3-trifluoromethyl-[1,2,4]tri...)
Affinity DataIC50:  15nMAssay Description:Binding affinity against alpha2 delta-1 subunit of voltage-gated calcium channel in human.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143364(CHEMBL57657 | N*4*-Acridin-9-yl-N*1*,N*1*-diethyl-...)
Affinity DataIC50:  18nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50080153((1-Aminomethyl-cyclohexyl)-acetic acid | 2-(1-(ami...)
Affinity DataIC50:  27nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145330(CHEMBL310121 | [2-(3-Bromo-phenyl)-ethyl]-{(S)-1-[...)
Affinity DataIC50:  28nMAssay Description:Binding affinity against alpha2 delta-1 subunit of voltage-gated calcium channel in human.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145307((2-m-Tolyl-ethyl)-{1-[6-(3-trifluoromethyl-[1,2,4]...)
Affinity DataIC50:  29nMAssay Description:Binding affinity against alpha2 delta-1 subunit of voltage-gated calcium channel in human.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145305(CHEMBL446627 | Phenethyl-{(S)-1-[6-(3-trifluoromet...)
Affinity DataIC50:  30nMAssay Description:Binding affinity against alpha2 delta-1 subunit of voltage-gated calcium channel in human.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366906(CHEMBL1169381)
Affinity DataIC50:  30nMAssay Description:Binding affinity against alpha2 delta-1 subunit of voltage-gated calcium channel in human.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145329(CHEMBL79184 | Phenethyl-{1-[6-(3-trifluoromethyl-[...)
Affinity DataIC50:  36nMAssay Description:Binding affinity against alpha2 delta-1 subunit of voltage-gated calcium channel in human.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143345(CHEMBL57487 | N*4*-Acridin-9-yl-N*1*,N*1*-diethyl-...)
Affinity DataIC50:  38nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143358((S)-N*1*,N*1*-Diethyl-N*4*-(1,2,3,4,5,6,7,8-octahy...)
Affinity DataIC50:  43nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143348(CHEMBL299461 | N*1*-Acridin-9-yl-1-cyclopropyl-N*4...)
Affinity DataIC50:  52nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145306(CHEMBL84067 | Phenethyl-[6-(3-trifluoromethyl-[1,2...)
Affinity DataIC50:  72nMAssay Description:Binding affinity against alpha-2 delta-1 subunit of voltage gated subunit of Ca+2 channel in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143357((S)-N*4*-Acridin-9-yl-N*1*,N*1*-diethyl-pentane-1,...)
Affinity DataIC50:  110nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145326(CHEMBL311873 | [2-(3-Methoxy-phenyl)-ethyl]-[6-(3-...)
Affinity DataIC50:  116nMAssay Description:Binding affinity against alpha-2 delta-1 subunit of voltage gated subunit of Ca+2 channel in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145313(CHEMBL81850 | [6-(3-Methoxymethyl-[1,2,4]triazolo[...)
Affinity DataIC50:  131nMAssay Description:Binding affinity against alpha-2 delta-1 subunit of voltage gated subunit of Ca+2 channel in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145314(CHEMBL81225 | [6-(3-Methyl-[1,2,4]triazolo[3,4-a]p...)
Affinity DataIC50:  145nMAssay Description:Binding affinity against alpha-2 delta-1 subunit of voltage gated subunit of Ca+2 channel in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145316(CHEMBL79968 | [6-(3-Cyclohexyl-[1,2,4]triazolo[3,4...)
Affinity DataIC50:  145nMAssay Description:Binding affinity against alpha-2 delta-1 subunit of voltage gated subunit of Ca+2 channel in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143347(CHEMBL58047 | N*1*,N*1*-Diethyl-N*4*-(1,2,3,4,5,6,...)
Affinity DataIC50:  160nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145311(CHEMBL79762 | [2-(3-Fluoro-phenyl)-ethyl]-[6-(3-tr...)
Affinity DataIC50:  161nMAssay Description:Binding affinity against alpha2 delta-1 subunit of voltage-gated calcium channel in human.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145331(CHEMBL309198 | {2-Methyl-1-[6-(3-trifluoromethyl-[...)
Affinity DataIC50:  174nMAssay Description:Binding affinity against alpha2 delta-1 subunit of voltage-gated calcium channel in human.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145328(CHEMBL81495 | Phenethyl-{1-[6-(3-trifluoromethyl-[...)
Affinity DataIC50:  183nMAssay Description:Binding affinity against alpha2 delta-1 subunit of voltage-gated calcium channel in human.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145322(CHEMBL79400 | [6-(3-Methylsulfanyl-[1,2,4]triazolo...)
Affinity DataIC50:  194nMAssay Description:Binding affinity against alpha-2 delta-1 subunit of voltage gated subunit of Ca+2 channel in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145301(CHEMBL310209 | Phenethyl-[6-(3-phenyl-[1,2,4]triaz...)
Affinity DataIC50:  195nMAssay Description:Binding affinity against alpha-2 delta-1 subunit of voltage gated subunit of Ca+2 channel in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145302((2-Phenyl-propyl)-[6-(3-trifluoromethyl-[1,2,4]tri...)
Affinity DataIC50:  198nMAssay Description:Binding affinity against alpha2 delta-1 subunit of voltage-gated calcium channel in human.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143363(CHEMBL59367 | N*4*-Acridin-9-yl-N*1*,N*1*-diethyl-...)
Affinity DataIC50:  220nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145327(CHEMBL81141 | {6-[3-(5-Methyl-isoxazol-3-yl)-[1,2,...)
Affinity DataIC50:  220nMAssay Description:Binding affinity against alpha-2 delta-1 subunit of voltage gated subunit of Ca+2 channel in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145319((R)-((S)-2-Phenyl-cyclopropyl)-[6-(3-trifluorometh...)
Affinity DataIC50:  229nMAssay Description:Binding affinity against alpha2 delta-1 subunit of voltage-gated calcium channel in human.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145299(CHEMBL79423 | Phenethyl-[6-([1,2,4]triazolo[3,4-a]...)
Affinity DataIC50:  230nMAssay Description:Binding affinity against alpha-2 delta-1 subunit of voltage gated subunit of Ca+2 channel in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145318(CHEMBL418920 | [6-(3-Ethyl-[1,2,4]triazolo[3,4-a]p...)
Affinity DataIC50:  241nMAssay Description:Binding affinity against alpha-2 delta-1 subunit of voltage gated subunit of Ca+2 channel in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145303((2-p-Tolyl-ethyl)-[6-(3-trifluoromethyl-[1,2,4]tri...)
Affinity DataIC50:  260nMAssay Description:Binding affinity against alpha2 delta-1 subunit of voltage-gated calcium channel in human.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143355(CHEMBL59368 | N*4*-Acridin-9-yl-N*1*,N*1*-diethyl-...)
Affinity DataIC50:  270nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145304(CHEMBL82891 | [6-(3-Cyclopropyl-[1,2,4]triazolo[3,...)
Affinity DataIC50:  272nMAssay Description:Binding affinity against alpha-2 delta-1 subunit of voltage gated subunit of Ca+2 channel in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145321(CHEMBL79618 | [2-(2-Fluoro-phenyl)-ethyl]-[6-(3-tr...)
Affinity DataIC50:  291nMAssay Description:Binding affinity against alpha-2 delta-1 subunit of voltage gated subunit of Ca+2 channel in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145317(CHEMBL81851 | [6-(3-Isopropyl-[1,2,4]triazolo[3,4-...)
Affinity DataIC50:  342nMAssay Description:Binding affinity against alpha-2 delta-1 subunit of voltage gated subunit of Ca+2 channel in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143351(CHEMBL292915 | N*1*,N*1*-Diethyl-N*4*-(1,2,3,4-tet...)
Affinity DataIC50:  420nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145308((2-o-Tolyl-ethyl)-[6-(3-trifluoromethyl-[1,2,4]tri...)
Affinity DataIC50:  448nMAssay Description:Binding affinity against alpha2 delta-1 subunit of voltage-gated calcium channel in human.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145300(CHEMBL420593 | [2-(4-Fluoro-phenyl)-ethyl]-[6-(3-t...)
Affinity DataIC50:  630nMAssay Description:Binding affinity against alpha2 delta-1 subunit of voltage-gated calcium channel in human.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145325(((S)-1-Methyl-2-phenyl-ethyl)-[6-(3-trifluoromethy...)
Affinity DataIC50:  700nMAssay Description:Binding affinity against alpha2 delta-1 subunit of voltage-gated calcium channel in human.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143359((R)-N*1*,N*1*-Diethyl-N*4*-(1,2,3,4,5,6,7,8-octahy...)
Affinity DataIC50:  760nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145309(CHEMBL315485 | [2-(4-Methoxy-phenyl)-ethyl]-[6-(3-...)
Affinity DataIC50:  829nMAssay Description:Binding affinity against alpha-2 delta-1 subunit of voltage gated subunit of Ca+2 channel in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143353(CHEMBL59208 | N*1*,N*1*-Diethyl-N*4*-(2-phenyl-qui...)
Affinity DataIC50:  960nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143360(CHEMBL56880 | N*1*-Acridin-9-yl-N*4*,N*4*-diethyl-...)
Affinity DataIC50:  1.10E+3nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145312((1-Methyl-2-phenyl-ethyl)-[6-(3-trifluoromethyl-[1...)
Affinity DataIC50:  1.37E+3nMAssay Description:Binding affinity against alpha2 delta-1 subunit of voltage-gated calcium channel in human.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50145310(CHEMBL309390 | [2-(2-Methoxy-phenyl)-ethyl]-[6-(3-...)
Affinity DataIC50:  3.16E+3nMAssay Description:Binding affinity against alpha-2 delta-1 subunit of voltage gated subunit of Ca+2 channel in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143366(CHEMBL56754 | N*4*-Acridin-9-yl-N*1*-isopropyl-pen...)
Affinity DataIC50:  5.10E+3nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143352(Acridin-9-yl-[1-methyl-4-((R)-2-methyl-6-(S)-methy...)
Affinity DataIC50:  5.90E+3nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143365(CHEMBL59089 | N*5*-Acridin-9-yl-N*1*,N*1*-diethyl-...)
Affinity DataIC50:  6.00E+3nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143362(Acridin-9-yl-(1-methyl-4-pyrrolidin-1-yl-butyl)-am...)
Affinity DataIC50:  9.90E+3nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50143346(CHEMBL58470 | N*3*-Acridin-9-yl-N*1*,N*1*-diethyl-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards alpha2-delta subunit of a voltage gated calcium channel using [3H]-gabapentin in human brain membrane (A710 membrane)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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