Affinity DataKi: 5.20nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10.4nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11.2nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11.2nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 21.3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 23.6nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 26.6nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 35.1nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 37.8nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 38.5nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 40.2nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 42.5nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 64.5nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 66.3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 75.3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 78.3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 175nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 780nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.42E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.45E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of N-type calcium channel (VSCC) in IMR-32 at 10 uMMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of L-type [Ca2+] channel (VSCC) in rat A7r5 vascular smooth muscle cellsMore data for this Ligand-Target Pair
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of N-type calcium channel (VSCC) in IMR-32 at 10 uMMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of L-type [Ca2+] channel (VSCC) in rat A7r5 vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 302nMAssay Description:Agonist activity at human 5HT1A receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 302nMAssay Description:Agonist activity at human 5HT1A receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 169nMAssay Description:Agonist activity at human 5HT1A receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 216nMAssay Description:Agonist activity at human 5HT1A receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 290nMAssay Description:Agonist activity at human 5HT1A receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 51.4nMAssay Description:Agonist activity at human 5HT1A receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 65nMAssay Description:Agonist activity at human 5HT1A receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 40.7nMAssay Description:Agonist activity at human 5HT1A receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataKd: 35.3nMAssay Description:Binding affinity to wild type EGFR (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 140nMAssay Description:Agonist activity at human 5HT1A receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 147nMAssay Description:Agonist activity at human 5HT1A receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 138nMAssay Description:Agonist activity at human 5HT1A receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 41nMAssay Description:Agonist activity at human 5HT1A receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair