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Found 618 with Last Name = 'bilotta' and Initial = 'ja'
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100437(US8501732, I-1)
Affinity DataIC50:  1nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018759(CHEMBL3291350)
Affinity DataIC50:  4nMAssay Description:Inhibition of rat 11betaHSD1 assessed as reduction of cortisone to cortisol by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018760(CHEMBL3291357)
Affinity DataIC50:  4nMAssay Description:Inhibition of full-length human 11betaHSD1 expressed in HEK293 cells assessed as cortisol level by competitive ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100609(US8501732, I-169)
Affinity DataIC50:  4nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100549(US8501732, I-109)
Affinity DataIC50:  4nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100550(US8501732, I-110)
Affinity DataIC50:  4nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100445(US8501732, I-9)
Affinity DataIC50:  4nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018761(CHEMBL3291348)
Affinity DataIC50:  5nMAssay Description:Inhibition of rat 11betaHSD1 assessed as reduction of cortisone to cortisol by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100551(US8501732, I-111)
Affinity DataIC50:  5nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100573(US8501732, I-133)
Affinity DataIC50:  6nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100552(US8501732, I-112)
Affinity DataIC50:  6nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018793(CHEMBL3291344)
Affinity DataIC50:  7nMAssay Description:Inhibition of full-length human 11betaHSD1 expressed in HEK293 cells assessed as cortisol level by competitive ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018761(CHEMBL3291348)
Affinity DataIC50:  7nMAssay Description:Inhibition of full-length human 11betaHSD1 expressed in HEK293 cells assessed as cortisol level by competitive ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100574(US8501732, I-134)
Affinity DataIC50:  7nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100553(US8501732, I-113)
Affinity DataIC50:  7nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100554(US8501732, I-114)
Affinity DataIC50:  7nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100438(US8501732, I-2)
Affinity DataIC50:  7nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100448(US8501732, I-12)
Affinity DataIC50:  7nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018759(CHEMBL3291350)
Affinity DataIC50:  8nMAssay Description:Inhibition of full-length human 11betaHSD1 expressed in HEK293 cells assessed as cortisol level by competitive ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100575(US8501732, I-135)
Affinity DataIC50:  8nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100555(US8501732, I-115)
Affinity DataIC50:  8nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100556(US8501732, I-116)
Affinity DataIC50:  8nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018795(CHEMBL3291339)
Affinity DataIC50:  9nMAssay Description:Inhibition of full-length human 11betaHSD1 expressed in HEK293 cells assessed as cortisol level by competitive ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018769(CHEMBL3291346)
Affinity DataIC50:  9nMAssay Description:Inhibition of full-length human 11betaHSD1 expressed in HEK293 cells assessed as cortisol level by competitive ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100439(US8501732, I-3)
Affinity DataIC50:  9nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018797(CHEMBL3291345)
Affinity DataIC50:  10nMAssay Description:Inhibition of rat 11betaHSD1 assessed as reduction of cortisone to cortisol by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018760(CHEMBL3291357)
Affinity DataIC50:  10nMAssay Description:Inhibition of rat 11betaHSD1 assessed as reduction of cortisone to cortisol by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018794(CHEMBL3291340)
Affinity DataIC50:  10nMAssay Description:Inhibition of full-length human 11betaHSD1 expressed in HEK293 cells assessed as cortisol level by competitive ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100610(US8501732, I-170)
Affinity DataIC50:  10nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100557(US8501732, I-117)
Affinity DataIC50:  10nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100558(US8501732, I-118)
Affinity DataIC50:  11nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100502(US8501732, I-62)
Affinity DataIC50:  11nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018793(CHEMBL3291344)
Affinity DataIC50:  12nMAssay Description:Inhibition of rat 11betaHSD1 assessed as reduction of cortisone to cortisol by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100576(US8501732, I-136)
Affinity DataIC50:  12nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100577(US8501732, I-137)
Affinity DataIC50:  12nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100590(US8501732, I-150)
Affinity DataIC50:  12nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018769(CHEMBL3291346)
Affinity DataIC50:  13nMAssay Description:Inhibition of rat 11betaHSD1 assessed as reduction of cortisone to cortisol by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018798(CHEMBL3291342)
Affinity DataIC50:  13nMAssay Description:Inhibition of full-length human 11betaHSD1 expressed in HEK293 cells assessed as cortisol level by competitive ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018797(CHEMBL3291345)
Affinity DataIC50:  13nMAssay Description:Inhibition of full-length human 11betaHSD1 expressed in HEK293 cells assessed as cortisol level by competitive ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100578(US8501732, I-138)
Affinity DataIC50:  13nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100579(US8501732, I-139)
Affinity DataIC50:  13nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100559(US8501732, I-119)
Affinity DataIC50:  13nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100469(US8501732, I-29)
Affinity DataIC50:  13nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018799(CHEMBL3291347)
Affinity DataIC50:  14nMAssay Description:Inhibition of full-length human 11betaHSD1 expressed in HEK293 cells assessed as cortisol level by competitive ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018802(CHEMBL3291354)
Affinity DataIC50:  14nMAssay Description:Inhibition of full-length human 11betaHSD1 expressed in HEK293 cells assessed as cortisol level by competitive ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100580(US8501732, I-140)
Affinity DataIC50:  14nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100440(US8501732, I-4)
Affinity DataIC50:  14nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100443(US8501732, I-7)
Affinity DataIC50:  14nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018803(CHEMBL3291358)
Affinity DataIC50:  15nMAssay Description:Inhibition of full-length human 11betaHSD1 expressed in HEK293 cells assessed as cortisol level by competitive ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM100572(US8501732, I-132)
Affinity DataIC50:  15nMAssay Description:In vitro JNK1 assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
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