Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of amyloid beta42 aggregation assessed as reduction in fluorescence after 4 days by thioflavin T-based fluorometryMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of amyloid beta42 aggregation assessed as reduction in fluorescence after 4 days by thioflavin T-based fluorometryMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of amyloid beta42 aggregation assessed as reduction in fluorescence measured immediately post-compound addition by thioflavin T-based fluo...More data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of amyloid beta42 aggregation assessed as reduction in fluorescence measured immediately post-compound addition by thioflavin T-based fluo...More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: 4.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein(RPV).More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataEC50: 3.50E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein(RPV).More data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+5nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+5nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataEC50: 0.5nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 60nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair