Compile Data Set for Download or QSAR
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Found 9 with Last Name = 'blakemore' and Initial = 'w'
TargetProthrombin(Homo sapiens (Human))
Astex

LigandPNGBDBM12588((2R,3S)-3-({[5-chloro-2-(1H-1,2,3,4-tetrazol-1-yl)...)
Affinity DataIC50:  1.40nMpH: 8.0 T: 2°CAssay Description:The cleavage of the substrate was followed by monitoring the change in fluorescence at 460 nm (excitation at 365 nm) for 25 min at room temperature o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Astex

LigandPNGBDBM12589((2R,3S)-3-({[5-chloro-2-(1H-1,2,3,4-tetrazol-1-yl)...)
Affinity DataIC50:  3.70nMpH: 8.0 T: 2°CAssay Description:The cleavage of the substrate was followed by monitoring the change in fluorescence at 460 nm (excitation at 365 nm) for 25 min at room temperature o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Astex

LigandPNGBDBM12587((2R,3S)-3-{[(3-chlorophenyl)methyl]amino}-2-hydrox...)
Affinity DataIC50:  220nMpH: 8.0 T: 2°CAssay Description:The cleavage of the substrate was followed by monitoring the change in fluorescence at 460 nm (excitation at 365 nm) for 25 min at room temperature o...More data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
Astex

LigandPNGBDBM12586((2R,3S)-3-amino-2-hydroxy-N-(4-methoxy-2,3,6-trime...)
Affinity DataIC50:  1.20E+4nMpH: 8.0 T: 2°CAssay Description:The cleavage of the substrate was followed by monitoring the change in fluorescence at 460 nm (excitation at 365 nm) for 25 min at room temperature o...More data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
Astex

LigandPNGBDBM12590((6-aminoacridin-3-yl)amine | MLS003876812 | Profla...)
Affinity DataIC50:  1.20E+4nMpH: 8.0 T: 2°CAssay Description:The cleavage of the substrate was followed by monitoring the change in fluorescence at 460 nm (excitation at 365 nm) for 25 min at room temperature o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Astex

LigandPNGBDBM12585((2R,3S)-3-amino-2-hydroxy-N-(naphthalen-2-yl)-4-ph...)
Affinity DataIC50:  1.00E+5nMpH: 8.0 T: 2°CAssay Description:The cleavage of the substrate was followed by monitoring the change in fluorescence at 460 nm (excitation at 365 nm) for 25 min at room temperature o...More data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
Astex

LigandPNGBDBM12584((3-chlorophenyl)methanamine | 1-(3-CHLOROPHENYL)ME...)
Affinity DataIC50:  3.00E+5nMpH: 8.0 T: 2°CAssay Description:The cleavage of the substrate was followed by monitoring the change in fluorescence at 460 nm (excitation at 365 nm) for 25 min at room temperature o...More data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
Astex

LigandPNGBDBM12582(1-(4-chlorophenyl)-1H-1,2,3,4-tetrazole | 1-(4-chl...)
Affinity DataIC50:  3.30E+5nMpH: 8.0 T: 2°CAssay Description:The cleavage of the substrate was followed by monitoring the change in fluorescence at 460 nm (excitation at 365 nm) for 25 min at room temperature o...More data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
Astex

LigandPNGBDBM772(Benzamidine | CHEMBL79897 | [amino(phenyl)methylid...)
Affinity DataIC50:  4.40E+5nMpH: 8.0 T: 2°CAssay Description:The cleavage of the substrate was followed by monitoring the change in fluorescence at 460 nm (excitation at 365 nm) for 25 min at room temperature o...More data for this Ligand-Target Pair