Compile Data Set for Download or QSAR
maximum 50k data
Found 16 with Last Name = 'blanco' and Initial = 'f'
TargetAndrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50420542(CHEMBL2086965)
Affinity DataIC50:  1.33E+4nMAssay Description:Antagonist activity at wild type AR LBD assessed as inhibition of DHT-induced fluorescent labeled D11-FxxLF recruitment after 2 to 4 hrs by TR-FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50420539(CHEMBL2086966)
Affinity DataIC50:  1.59E+4nMAssay Description:Antagonist activity at wild type AR LBD assessed as inhibition of DHT-induced fluorescent labeled D11-FxxLF recruitment after 2 to 4 hrs by TR-FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50420541(CHEMBL2086967)
Affinity DataIC50:  1.79E+4nMAssay Description:Antagonist activity at wild type AR LBD assessed as inhibition of DHT-induced fluorescent labeled D11-FxxLF recruitment after 2 to 4 hrs by TR-FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50420542(CHEMBL2086965)
Affinity DataIC50:  2.25E+4nMAssay Description:Antagonist activity at PR assessed as inhibition of progesterone-induced fluorescent labelled SRC1-4 recruitment after 2 to 4 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50420540(CHEMBL2086964)
Affinity DataIC50:  2.63E+4nMAssay Description:Antagonist activity at wild type AR LBD assessed as inhibition of DHT-induced fluorescent labeled D11-FxxLF recruitment after 2 to 4 hrs by TR-FRET a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-L(Mus musculus)
Ikerchem

Curated by ChEMBL
LigandPNGBDBM50426077(CHEMBL2315999)
Affinity DataIC50:  2.76E+4nMAssay Description:Inhibition of LFA-1/ICAM-1 interaction in mouse Lim51b cells assessed as PMA-induced adhesion to ICAM-1 expressing HSE cells measured per 10'5 cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50420540(CHEMBL2086964)
Affinity DataIC50:  2.77E+4nMAssay Description:Antagonist activity at PR assessed as inhibition of progesterone-induced fluorescent labelled SRC1-4 recruitment after 2 to 4 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50420542(CHEMBL2086965)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescent labelled SRC1-4 from dexamethasone-GR complex after 2 to 4 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50420540(CHEMBL2086964)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescent labelled PGC-1alpha from estradiol-ERbeta complex after 2 to 4 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50420542(CHEMBL2086965)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescent labelled PGC-1alpha from estradiol-ERbeta complex after 2 to 4 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50420540(CHEMBL2086964)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescent labelled SRC1-4 from dexamethasone-GR complex after 2 to 4 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50420542(CHEMBL2086965)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescent labelled PGC-1alpha from estradiol-ERalpha complex after 2 to 4 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50420540(CHEMBL2086964)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescent labelled PGC-1alpha from estradiol-ERalpha complex after 2 to 4 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-L(Homo sapiens (Human))
Ikerchem

Curated by ChEMBL
LigandPNGBDBM50426077(CHEMBL2315999)
Affinity DataKd:  1.01E+4nMAssay Description:Binding affinity to I-domain of human integrin alphaL (amino acid residues 128 to 307) plus initial methionine expressed in Escherichia coli by NMR s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-L(Homo sapiens (Human))
Ikerchem

Curated by ChEMBL
LigandPNGBDBM34168(LOVASTATIN | MLS000069585 | SMR000058779 | US91151...)
Affinity DataKd:  1.29E+4nMAssay Description:Binding affinity to I-domain of human integrin alphaL (amino acid residues 128 to 307) plus initial methionine expressed in Escherichia coli by NMR s...More data for this Ligand-Target Pair
TargetIntegrin alpha-L(Homo sapiens (Human))
Ikerchem

Curated by ChEMBL
LigandPNGBDBM50426078(CHEMBL2316248)
Affinity DataKd:  7.40E+3nMAssay Description:Binding affinity to I-domain of human integrin alphaL (amino acid residues 128 to 307) plus initial methionine expressed in Escherichia coli by NMR s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed