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Found 16 with Last Name = 'blaszczak' and Initial = 'lc'
TargetEstrogen receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataIC50:  3nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor in MCF-7 cellsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Eli Lilly

LigandPNGBDBM15471(4-[(1-{[2-oxo-2-(thiophen-3-yl)ethyl]amino}cyclope...)
Affinity DataIC50:  5nMpH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Eli Lilly

LigandPNGBDBM15465(4-[(3R)-3-{[2-(3,4-difluorophenyl)-2-oxoethyl]amin...)
Affinity DataIC50:  39nMpH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50230556(CHEMBL176509)
Affinity DataIC50:  73nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor in MCF-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Eli Lilly

LigandPNGBDBM15464(4-[(3R)-3-{[2-(4-fluorophenyl)-2-oxoethyl]amino}bu...)
Affinity DataIC50:  84nMpH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Eli Lilly

LigandPNGBDBM15469(4-[(3R)-3-{[2-oxo-2-(thiophen-3-yl)ethyl]amino}but...)
Affinity DataIC50:  110nMpH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50230557(CHEBI:90187 | LY-117018)
Affinity DataIC50:  120nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor in MCF-7 cellsMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50230560(CHEMBL2112950)
Affinity DataIC50:  125nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor in MCF-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM19441(2-(4-hydroxyphenyl)-3-({4-[2-(piperidin-1-yl)ethox...)
Affinity DataIC50:  170nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor in MCF-7 cellsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Eli Lilly

LigandPNGBDBM15463(4-[(3R)-3-[(2-oxo-2- phenylethyl)amino]butyl]benza...)
Affinity DataIC50:  280nMpH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Eli Lilly

LigandPNGBDBM15470(4-[(2R)-2-{[2-oxo-2-(thiophen-3-yl)ethyl]amino}pro...)
Affinity DataIC50:  340nMpH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50230558(CHEMBL2112949)
Affinity DataIC50:  740nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor in MCF-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Eli Lilly

LigandPNGBDBM15467(4-[(3R)-3-{[2-(4-chlorophenyl)-2-oxoethyl]amino}bu...)
Affinity DataIC50:  820nMpH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50230559(CHEMBL367432)
Affinity DataIC50:  1.65E+3nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor in MCF-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Eli Lilly

LigandPNGBDBM15466(4-[(3R)-3-{[2-(2-fluorophenyl)-2-oxoethyl]amino}bu...)
Affinity DataIC50:  3.80E+3nMpH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Eli Lilly

LigandPNGBDBM15468(4-(3-{[2-(4-methylphenyl)-2-oxoethyl]amino}butyl)b...)
Affinity DataIC50:  2.10E+4nMpH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed