Compile Data Set for Download or QSAR
maximum 50k data
Found 6 with Last Name = 'blethrow' and Initial = 'j'
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Princeton University

LigandPNGBDBM25116(1-tert-butyl-3-(4-methylphenyl)-1H-pyrazolo[3,4-d]...)
Affinity DataIC50:  5nMAssay Description:Inhibition of protein tyrosine kinasesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Princeton University

LigandPNGBDBM25116(1-tert-butyl-3-(4-methylphenyl)-1H-pyrazolo[3,4-d]...)
Affinity DataIC50:  6nMAssay Description:Inhibition of protein tyrosine kinasesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50253632(6-Azido-7-nitro-1,4-dihydroquinoxaline-2,3-dione |...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of GluR2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50253650(CHEMBL462490 | [1,2,5]oxadiazolo[3,4-g]quinoxaline...)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of GluR2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Princeton University

LigandPNGBDBM25116(1-tert-butyl-3-(4-methylphenyl)-1H-pyrazolo[3,4-d]...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of protein tyrosine kinasesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Princeton University

LigandPNGBDBM25116(1-tert-butyl-3-(4-methylphenyl)-1H-pyrazolo[3,4-d]...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of protein tyrosine kinasesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed