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Found 20 with Last Name = 'bloch' and Initial = 's'
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50390490(CHEMBL2071603)
Affinity DataKi:  0.0430nMAssay Description:Displacement of [125I]-c(RGDyK) from human integrin alphavbeta3 after 16 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50390491(CHEMBL2071604)
Affinity DataKi:  0.663nMAssay Description:Displacement of [125I]-c(RGDyK) from human integrin alphavbeta3 after 16 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50390492(CHEMBL2071605)
Affinity DataKi:  2.27nMAssay Description:Displacement of [125I]-c(RGDyK) from human integrin alphavbeta3 after 16 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50390490(CHEMBL2071603)
Affinity DataIC50:  0.281nMAssay Description:Displacement of [125I]-c(RGDyK) from human integrin alphavbeta3 after 16 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50390492(CHEMBL2071605)
Affinity DataIC50:  3.52nMAssay Description:Displacement of [125I]-c(RGDyK) from human integrin alphavbeta3 after 16 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50390491(CHEMBL2071604)
Affinity DataIC50:  4.31nMAssay Description:Displacement of [125I]-c(RGDyK) from human integrin alphavbeta3 after 16 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184908(CHEMBL402661 | cypate-[(RGD)4-NH2]1)
Affinity DataIC50:  25.9nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184904(CHEMBL206344 | cyclo(RGDfV) (control))
Affinity DataIC50:  28.7nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184902(CHEMBL407126 | cyclo[RGDfK(cypate)])
Affinity DataIC50:  63.9nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184906(CHEMBL429568 | cypate-[(RGD)4-NH2]2)
Affinity DataIC50:  79.6nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184903(CHEMBL415188 | cypate-[(RGD)2-NH2]2)
Affinity DataIC50:  104nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184905(CHEMBL413898 | cypate-[(RGD)3-NH2]2)
Affinity DataIC50:  132nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50237601(CHEMBL411941 | CycloRGDfV | [(2S,5R,8S,11S)-5-Benz...)
Affinity DataIC50:  325nMAssay Description:Displacement of [125I]echistatin from human integrin alpha5beta3 expressed in human A549 cells by binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184907(CHEMBL412767 | cypate-[(RGD)3-NH2]1)
Affinity DataIC50:  481nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50340881(CHEMBL1761774 | cyclo[Arg-Gly-Asp-D-Phe-Lys(epselo...)
Affinity DataIC50:  720nMAssay Description:Displacement of [125I]echistatin from human integrin alpha5beta3 expressed in human A549 cells by binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184909(CHEMBL438186 | cypate-[(RGD)2-NH2]1)
Affinity DataIC50:  730nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50340877(CHEMBL1761773 | Cypate-cyclo(Cys-Arg-Gly-Asp-Cys)-...)
Affinity DataIC50:  4.60E+3nMAssay Description:Displacement of [125I]echistatin from human integrin alpha5beta3 expressed in human A549 cells by binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50340878(2-(7-(3-(3-((4R,7S,10S,13S,16R)-4-carbamoyl-7-(car...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]echistatin from human integrin alpha5beta3 expressed in human A549 cells by binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50340879(2-(7-(3-(3-((4R,7S,10S,13S,16R)-4-carbamoyl-7-(car...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]echistatin from human integrin alpha5beta3 expressed in human A549 cells by binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50340880(2-(7-(3-(3-((3S,6R,11R,14S,19aS)-6-carbamoyl-3-(ca...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]echistatin from human integrin alpha5beta3 expressed in human A549 cells by binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed