TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Binding affinity in rat forebrain against Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition constant from beta adrenergic receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Evaluated for beta-receptor affinity determined in rat brain membrane fraction with [3H]- dihydroalprenololMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: 92nMAssay Description:binding affinity in rat hippocampi against alpha7 nicotinic receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: 92nMAssay Description:binding affinity in rat hippocampi against alpha7 nicotinic receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Binding affinity in rat forebrain against Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:binding affinity in rat hippocampi against alpha7 nicotinic receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:binding affinity in rat hippocampi against alpha7 nicotinic receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:binding affinity in rat forebrain against alpha4-beta2 nicotinic receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:binding affinity in rat forebrain against alpha4-beta2 nicotinic receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: 480nMAssay Description:Binding affinity in rat hippocampi against Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: 560nMAssay Description:Binding affinity in rat hippocampi against Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: 690nMAssay Description:Binding affinity in rat hippocampi against Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Binding affinity against muscarinic acetylcholine receptor from rat brain crude membrane, using [3H]-NMS (N-Methylscopolamine) as the radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.47E+3nMAssay Description:Binding affinity against muscarinic acetylcholine receptor from rat brain crude membrane, using [3H]-NMS (N-Methylscopolamine) as the radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.47E+3nMAssay Description:Binding affinity against muscarinic acetylcholine receptor from rat brain crude membrane, using [3H]-NMS (N-Methylscopolamine) as the radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition constant from beta adrenergic receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Inhibition constant from beta adrenergic receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.63E+3nMAssay Description:Binding affinity against muscarinic acetylcholine receptor from rat brain crude membrane, using [3H]-NMS (N-Methylscopolamine) as the radioligand.More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: 2.20E+3nMAssay Description:Binding affinity in rat forebrain against Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Inhibition constant from beta adrenergic receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Compound was evaluated for its affinity towards Muscarinic acetylcholine receptor M2, using [3H]- N-methyl-scopolamine, a radioligand displacement as...More data for this Ligand-Target Pair
Affinity DataKi: 2.58E+3nMAssay Description:Binding affinity against muscarinic acetylcholine receptor from rat brain crude membrane, using [3H]-NMS (N-Methylscopolamine) as the radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 2.68E+3nMAssay Description:Binding affinity against muscarinic acetylcholine receptor from rat brain crude membrane, using [3H]-NMS (N-Methylscopolamine) as the radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 3.10E+3nMAssay Description:Compound was evaluated for its affinity towards Muscarinic acetylcholine receptor M1, using [3H]- pirenzepine, a radioligand displacement assay in ra...More data for this Ligand-Target Pair
Affinity DataKi: 3.67E+3nMAssay Description:Binding affinity against muscarinic acetylcholine receptor from rat brain crude membrane, using [3H]-NMS (N-Methylscopolamine) as the radioligand.More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: 3.70E+3nMAssay Description:Binding affinity in rat hippocampi against Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
Affinity DataKi: 3.80E+3nMAssay Description:Ability to displace [3H]- pirenzepine from M1 receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.80E+3nMAssay Description:Compound was evaluated for its affinity towards Muscarinic acetylcholine receptor M1, using [3H]- pirenzepine, a radioligand displacement assay in ra...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: 4.00E+3nMAssay Description:Binding affinity in rat hippocampi against Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
Affinity DataKi: 4.10E+3nMAssay Description:Compound was evaluated for its affinity towards Muscarinic acetylcholine receptor M1, using [3H]- pirenzepine, a radioligand displacement assay in ra...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: >4.30E+3nMAssay Description:Binding affinity in rat hippocampi against Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
Affinity DataKi: 4.80E+3nMAssay Description:Ability to displace [3H]- pirenzepine from M1 receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.30E+3nMAssay Description:Compound was evaluated for its affinity towards Muscarinic acetylcholine receptor M2, using [3H]- N-methyl-scopolamine, a radioligand displacement as...More data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nMAssay Description:Inhibition constant obtained from beta adrenergic receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.12E+3nMAssay Description:Binding affinity against muscarinic acetylcholine receptor from rat brain crude membrane, using [3H]-NMS (N-Methylscopolamine) as the radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 7.50E+3nMAssay Description:Inhibition constant from beta adrenergic receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.50E+3nMAssay Description:Inhibition constant from beta adrenergic receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Ability to displace [3H]- pirenzepine from M1 receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 8.26E+3nMAssay Description:Binding affinity against muscarinic acetylcholine receptor from rat brain crude membrane, using [3H]-NMS (N-Methylscopolamine) as the radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 8.80E+3nMAssay Description:Ability to displace [3H]- pirenzepine from M1 receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 9.00E+3nMAssay Description:Ability to displace [3H]- pirenzepine from M1 receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: 9.40E+3nMAssay Description:binding affinity in rat hippocampi against alpha7 nicotinic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.50E+3nMAssay Description:Ability to displace [3H]- pirenzepine from M1 receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 9.80E+3nMAssay Description:Compound was evaluated for its affinity towards Muscarinic acetylcholine receptor M2, using [3H]- N-methyl-scopolamine, a radioligand displacement as...More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Ability to displace [3H]- pirenzepine from M1 receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: 1.10E+4nMAssay Description:Binding affinity in rat forebrain against Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+4nMAssay Description:Inhibition constant from beta adrenergic receptor binding assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: >1.30E+4nMAssay Description:Binding affinity in rat hippocampi against Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Astrazeneca R&D Boston
Curated by ChEMBL
Astrazeneca R&D Boston
Curated by ChEMBL
Affinity DataKi: >1.30E+4nMAssay Description:Binding affinity in rat hippocampi against Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair