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Found 32 with Last Name = 'blum' and Initial = 'g'
TargetCathepsin B(Rattus norvegicus)
Stanford University

LigandPNGBDBM36331(Ac-YFR-AMOK 10b)
Affinity DataIC50:  7.30nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Rattus norvegicus)
Stanford University

LigandPNGBDBM36328(Z-FR-AMOK 9b)
Affinity DataIC50:  15nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Rattus norvegicus)
Stanford University

LigandPNGBDBM36327(Z-FG-AOMK 9a)
Affinity DataIC50:  120nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50296357(4,4'-(benzo[d][1,3]dioxol-5-ylazanediyl)bis(methyl...)
Affinity DataIC50:  170nMAssay Description:Inhibition of human IGF1R-mediated Poly Glu4Tyr phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50326005(4,4'-(1H-indazol-6-ylazanediyl)bis(methylene)diben...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human IGF1R-mediated Poly Glu4Tyr phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Rattus norvegicus)
Stanford University

LigandPNGBDBM36330(AC-YFG-AMOK 10a)
Affinity DataIC50:  220nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50326005(4,4'-(1H-indazol-6-ylazanediyl)bis(methylene)diben...)
Affinity DataIC50:  380nMAssay Description:Inhibition of human insulin receptor-mediated Poly Glu4Tyr phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50296357(4,4'-(benzo[d][1,3]dioxol-5-ylazanediyl)bis(methyl...)
Affinity DataIC50:  610nMAssay Description:Inhibition of human insulin receptor-mediated Poly Glu4Tyr phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50296357(4,4'-(benzo[d][1,3]dioxol-5-ylazanediyl)bis(methyl...)
Affinity DataIC50:  830nMAssay Description:Inhibition of human GST-fused Src-mediated Poly Glu4Tyr phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Rattus norvegicus)
Stanford University

LigandPNGBDBM36329(Z-LG-AOMK 9c)
Affinity DataIC50:  920nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Rattus norvegicus)
Stanford University

LigandPNGBDBM36325(Cathepsin Inhibitor III)
Affinity DataIC50:  1.20E+3nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50326008(4-((7,7a-dihydrobenzo[d][1,3]dioxol-5-ylamino)meth...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human IGF1R-mediated Poly Glu4Tyr phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin Z(Rattus norvegicus)
Stanford University

LigandPNGBDBM36325(Cathepsin Inhibitor III)
Affinity DataIC50:  1.50E+3nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50326004(4-((1H-indazol-6-ylamino)methyl)benzene-1,2-diol |...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human IGF1R-mediated Poly Glu4Tyr phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50326007(4,4'-(naphthalen-2-ylazanediyl)bis(methylene)diben...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human insulin receptor-mediated Poly Glu4Tyr phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50326003(4-((benzo[d][1,3]dioxol-5-ylamino)methyl)benzene-1...)
Affinity DataIC50:  1.69E+3nMAssay Description:Inhibition of human IGF1R-mediated Poly Glu4Tyr phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50326003(4-((benzo[d][1,3]dioxol-5-ylamino)methyl)benzene-1...)
Affinity DataIC50:  1.86E+3nMAssay Description:Inhibition of human GST-fused Src-mediated Poly Glu4Tyr phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50326003(4-((benzo[d][1,3]dioxol-5-ylamino)methyl)benzene-1...)
Affinity DataIC50:  2.08E+3nMAssay Description:Inhibition of human insulin receptor-mediated Poly Glu4Tyr phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50326004(4-((1H-indazol-6-ylamino)methyl)benzene-1,2-diol |...)
Affinity DataIC50:  2.25E+3nMAssay Description:Inhibition of human insulin receptor-mediated Poly Glu4Tyr phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50326007(4,4'-(naphthalen-2-ylazanediyl)bis(methylene)diben...)
Affinity DataIC50:  2.45E+3nMAssay Description:Inhibition of human IGF1R-mediated Poly Glu4Tyr phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50296357(4,4'-(benzo[d][1,3]dioxol-5-ylazanediyl)bis(methyl...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of IGF1R-mediated colony formation in human LNCaP cells after 12 days by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50326006(4-((naphthalen-2-ylamino)methyl)benzene-1,2-diol |...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of human IGF1R-mediated Poly Glu4Tyr phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin Z(Rattus norvegicus)
Stanford University

LigandPNGBDBM36331(Ac-YFR-AMOK 10b)
Affinity DataIC50:  4.70E+3nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50326006(4-((naphthalen-2-ylamino)methyl)benzene-1,2-diol |...)
Affinity DataIC50:  5.15E+3nMAssay Description:Inhibition of human insulin receptor-mediated Poly Glu4Tyr phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50296357(4,4'-(benzo[d][1,3]dioxol-5-ylazanediyl)bis(methyl...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of IGF1R-mediated colony formation in human MCF7 cells after 12 days by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50296357(4,4'-(benzo[d][1,3]dioxol-5-ylazanediyl)bis(methyl...)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of IGF1R-mediated colony formation in human PC3 cells after 12 days by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPro-cathepsin H(Rattus norvegicus)
Stanford University

LigandPNGBDBM36325(Cathepsin Inhibitor III)
Affinity DataIC50:  6.60E+3nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPro-cathepsin H(Rattus norvegicus)
Stanford University

LigandPNGBDBM36329(Z-LG-AOMK 9c)
Affinity DataIC50:  7.90E+3nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPro-cathepsin H(Rattus norvegicus)
Stanford University

LigandPNGBDBM36330(AC-YFG-AMOK 10a)
Affinity DataIC50:  7.90E+3nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50326008(4-((7,7a-dihydrobenzo[d][1,3]dioxol-5-ylamino)meth...)
Affinity DataIC50:  9.90E+3nMAssay Description:Inhibition of human insulin receptor-mediated Poly Glu4Tyr phosphorylation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPro-cathepsin H(Rattus norvegicus)
Stanford University

LigandPNGBDBM36331(Ac-YFR-AMOK 10b)
Affinity DataIC50:  1.20E+4nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin Z(Rattus norvegicus)
Stanford University

LigandPNGBDBM36330(AC-YFG-AMOK 10a)
Affinity DataIC50:  3.90E+4nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed