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Found 74 with Last Name = 'boakye' and Initial = 'k'
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200411((S)-2-(5-(3-((2-(4-ethylphenyl)-5-methylpyrimidin-...)
Affinity DataIC50:  30nMAssay Description:Activity at human PPARdelta expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200403((S)-2-(5-(3-((2-(4-isopropylphenyl)-5-methylpyrimi...)
Affinity DataIC50:  49nMAssay Description:Activity at human PPARdelta expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200402(2-((S)-5-(3-(5-(5-acetyl-4-methylthiazol-2-yl)pyri...)
Affinity DataIC50:  56nMAssay Description:Activity at human PPARdelta expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200411((S)-2-(5-(3-((2-(4-ethylphenyl)-5-methylpyrimidin-...)
Affinity DataIC50:  175nMAssay Description:Activity at human PPARalpha expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200403((S)-2-(5-(3-((2-(4-isopropylphenyl)-5-methylpyrimi...)
Affinity DataIC50:  237nMAssay Description:Activity at human PPARalpha expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200411((S)-2-(5-(3-((2-(4-ethylphenyl)-5-methylpyrimidin-...)
Affinity DataIC50:  370nMAssay Description:Activity at mouse PPARdelta expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200403((S)-2-(5-(3-((2-(4-isopropylphenyl)-5-methylpyrimi...)
Affinity DataIC50:  610nMAssay Description:Activity at mouse PPARdelta expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200411((S)-2-(5-(3-((2-(4-ethylphenyl)-5-methylpyrimidin-...)
Affinity DataIC50:  670nMAssay Description:Activity at mouse PPARalpha expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200402(2-((S)-5-(3-(5-(5-acetyl-4-methylthiazol-2-yl)pyri...)
Affinity DataIC50:  1.39E+3nMAssay Description:Activity at mouse PPARdelta expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200403((S)-2-(5-(3-((2-(4-isopropylphenyl)-5-methylpyrimi...)
Affinity DataIC50:  2.53E+3nMAssay Description:Activity at mouse PPARalpha expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200402(2-((S)-5-(3-(5-(5-acetyl-4-methylthiazol-2-yl)pyri...)
Affinity DataIC50: >6.00E+3nMAssay Description:Activity at human PPARalpha expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200399((S)-2-(5-(3-((2-(4-ethylphenyl)pyrimidin-4-yl)(met...)
Affinity DataEC50:  800nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200400(2-((S)-5-(3-(5-(4,5-dimethylthiazol-2-yl)pyridin-2...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200401(2-((S)-5-(3-(methyl(5-methyl-2-m-tolylpyrimidin-4-...)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200403((S)-2-(5-(3-((2-(4-isopropylphenyl)-5-methylpyrimi...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200402(2-((S)-5-(3-(5-(5-acetyl-4-methylthiazol-2-yl)pyri...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200404((S)-2-(5-(3-((2-(4-ethylphenyl)-5-fluoropyrimidin-...)
Affinity DataEC50:  425nMAssay Description:Agonist activity at human PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200405(2-((S)-5-(3-((2-(3-ethoxyphenyl)-5-methylpyrimidin...)
Affinity DataEC50:  3.54E+3nMAssay Description:Agonist activity at human PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200406((S)-2-(5-(3-((5-ethyl-2-(4-ethylphenyl)pyrimidin-4...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200408((S)-2-(5-(3-(methyl(5-methyl-2-phenylpyrimidin-4-y...)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200407((S)-2-(5-(3-(methyl(5-methyl-2-p-tolylpyrimidin-4-...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200409((S)-2-(5-(3-((2-(4-fluorophenyl)-5-methylpyrimidin...)
Affinity DataEC50:  860nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200400(2-((S)-5-(3-(5-(4,5-dimethylthiazol-2-yl)pyridin-2...)
Affinity DataEC50:  6.78E+3nMAssay Description:Agonist activity at human PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200410((S)-2-(5-(3-((2-(4-tert-butylphenyl)-5-methylpyrim...)
Affinity DataEC50:  641nMAssay Description:Agonist activity at human PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200406((S)-2-(5-(3-((5-ethyl-2-(4-ethylphenyl)pyrimidin-4...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200412(2-((S)-5-(3-(5-(4-ethoxythiazol-2-yl)pyridin-2-ylo...)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200413(2-((S)-5-(3-((2-(3-chlorophenyl)-5-methylpyrimidin...)
Affinity DataEC50:  2.37E+3nMAssay Description:Agonist activity at human PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200415((S)-2-(5-(3-((2-(4-acetylphenyl)-5-methylpyrimidin...)
Affinity DataEC50:  237nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200414((S)-2-(5-(3-((2-(4-methoxyphenyl)-5-methylpyrimidi...)
Affinity DataEC50:  7.01E+3nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200416((S)-2-(5-(3-((2-(4-ethoxyphenyl)-5-methylpyrimidin...)
Affinity DataEC50:  161nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200401(2-((S)-5-(3-(methyl(5-methyl-2-m-tolylpyrimidin-4-...)
Affinity DataEC50:  670nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200418((S)-2-(5-(3-((2-(4-ethylphenyl)-6-methylpyrimidin-...)
Affinity DataEC50:  600nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200408((S)-2-(5-(3-(methyl(5-methyl-2-phenylpyrimidin-4-y...)
Affinity DataEC50:  678nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200417(2-((S)-5-(3-(5-(4-ethylthiazol-2-yl)pyridin-2-ylox...)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200405(2-((S)-5-(3-((2-(3-ethoxyphenyl)-5-methylpyrimidin...)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200412(2-((S)-5-(3-(5-(4-ethoxythiazol-2-yl)pyridin-2-ylo...)
Affinity DataEC50:  411nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200401(2-((S)-5-(3-(methyl(5-methyl-2-m-tolylpyrimidin-4-...)
Affinity DataEC50:  4.39E+3nMAssay Description:Agonist activity at human PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200404((S)-2-(5-(3-((2-(4-ethylphenyl)-5-fluoropyrimidin-...)
Affinity DataEC50:  360nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200404((S)-2-(5-(3-((2-(4-ethylphenyl)-5-fluoropyrimidin-...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200403((S)-2-(5-(3-((2-(4-isopropylphenyl)-5-methylpyrimi...)
Affinity DataEC50:  34nMAssay Description:Agonist activity at human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200411((S)-2-(5-(3-((2-(4-ethylphenyl)-5-methylpyrimidin-...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200410((S)-2-(5-(3-((2-(4-tert-butylphenyl)-5-methylpyrim...)
Affinity DataEC50:  28nMAssay Description:Agonist activity at human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200402(2-((S)-5-(3-(5-(5-acetyl-4-methylthiazol-2-yl)pyri...)
Affinity DataEC50:  35nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200417(2-((S)-5-(3-(5-(4-ethylthiazol-2-yl)pyridin-2-ylox...)
Affinity DataEC50:  421nMAssay Description:Agonist activity at human PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200407((S)-2-(5-(3-(methyl(5-methyl-2-p-tolylpyrimidin-4-...)
Affinity DataEC50:  1.15E+3nMAssay Description:Agonist activity at human PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200400(2-((S)-5-(3-(5-(4,5-dimethylthiazol-2-yl)pyridin-2...)
Affinity DataEC50:  511nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200414((S)-2-(5-(3-((2-(4-methoxyphenyl)-5-methylpyrimidi...)
Affinity DataEC50:  1.39E+3nMAssay Description:Agonist activity at human PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200412(2-((S)-5-(3-(5-(4-ethoxythiazol-2-yl)pyridin-2-ylo...)
Affinity DataEC50:  807nMAssay Description:Agonist activity at human PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200418((S)-2-(5-(3-((2-(4-ethylphenyl)-6-methylpyrimidin-...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200415((S)-2-(5-(3-((2-(4-acetylphenyl)-5-methylpyrimidin...)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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