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TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23921(3-amidinophenylalanine deriv., 63 | 3-amino-N-(3-{...)
Affinity DataKi:  1.5nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23916(3-amidinophenylalanine deriv., 12 | 3-amino-N-(3-{...)
Affinity DataKi:  1.80nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Human)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50245500(CHEMBL447547 | N-[(2S)-1-(2-{[(1R)-1-{[(1R)-5-carb...)
Affinity DataKi:  3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23918(3-amidinophenylalanine deriv., 60 | 4-amino-N-(3-{...)
Affinity DataKi:  3.90nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23915(3-amidinophenylalanine deriv., 58 | 3-carbamimidam...)
Affinity DataKi:  4.20nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23920(3-amidinophenylalanine deriv., 62 | 3-amino-N-(3-{...)
Affinity DataKi:  5nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072840(CHEMBL346607 | N-[1-(4-Diaminomethyl-benzyl)-2-oxo...)
Affinity DataKi:  6nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50060033(3-[3-(4-Methyl-piperidin-1-yl)-2-(naphthalene-2-su...)
Affinity DataKi:  6.20nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23917(3-amidinophenylalanine deriv., 59 | 3-amino-N-(3-{...)
Affinity DataKi:  6.60nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Human)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50041224((R)-3-(7-Carbamimidoyl-naphthalen-2-yl)-2-{4-[(S)-...)
Affinity DataKi:  7nMAssay Description:Binding affinity of the compound towards Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072851(1-[3-(3-Carbamimidoyl-phenyl)-2-(naphthalene-2-sul...)
Affinity DataKi:  8.40nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23913(3-amidinophenylalanine deriv., 56 | 3-carbamimidam...)
Affinity DataKi:  8.70nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23911(3-[(2S)-3-[4-(2-carbamimidamidoethyl)piperidin-1-y...)
Affinity DataKi:  13nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23896(3-amidinophenylalanine deriv., 40 | N-(2-carbamimi...)
Affinity DataKi:  13nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072843(2,7-Bis-(4-diaminomethyl-benzylidene)-cycloheptano...)
Affinity DataKi:  13nMAssay Description:Inhibitory activity against bovine coagulation factor X expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23887(3-amidinophenylalanine deriv., 31 | 4-({4-[(2S)-3-...)
Affinity DataKi:  14nM ΔG°:  -44.8kJ/molepH: 8.0 T: 25°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072846(3-[3-(4-Methyl-piperidin-1-yl)-2-(naphthalene-1-su...)
Affinity DataKi:  16nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072854(1-[3-(3-Carbamimidoyl-phenyl)-2-(naphthalene-2-sul...)
Affinity DataKi:  17nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23895(3-amidinophenylalanine deriv., 39 | N-(2-aminoethy...)
Affinity DataKi:  21nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23900(3-amidinophenylalanine deriv., 44 | 4-({1-[(2S)-3-...)
Affinity DataKi:  26nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072847(3-[2-(9,10-Dioxo-9,10-dihydro-anthracene-2-sulfony...)
Affinity DataKi:  26nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072856(3-[3-(4-Methyl-piperidin-1-yl)-3-oxo-2-(toluene-4-...)
Affinity DataKi:  26nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50060047(3-[2-(Naphthalene-2-sulfonylamino)-3-oxo-3-(4-phen...)
Affinity DataKi:  27nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23914(3-amidinophenylalanine deriv., 57 | 3-amino-N-(4-{...)
Affinity DataKi:  28nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Human)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072843(2,7-Bis-(4-diaminomethyl-benzylidene)-cycloheptano...)
Affinity DataKi:  35nMAssay Description:Inhibitory activity against human tissue-type plasminogen activator expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072854(1-[3-(3-Carbamimidoyl-phenyl)-2-(naphthalene-2-sul...)
Affinity DataKi:  36nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072853(4-[3-(3-Diaminomethyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  37nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23910(3-[(2S)-3-[4-(2-carbamimidamidoethyl)piperidin-1-y...)
Affinity DataKi:  38nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50041224((R)-3-(7-Carbamimidoyl-naphthalen-2-yl)-2-{4-[(S)-...)
Affinity DataKi:  41nMAssay Description:Binding affinity of the compound towards Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23907(3-[(2S)-3-[4-(3-carbamimidamidopropyl)piperidin-1-...)
Affinity DataKi:  42nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23877(3-[(2S)-2-(anthracene-2-sulfonamido)-3-[4-(3-carba...)
Affinity DataKi:  44nM ΔG°:  -42.0kJ/molepH: 8.0 T: 25°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23909(3-amidinophenylalanine deriv., 52 | 4-{1-[(2S)-3-(...)
Affinity DataKi:  45nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23902(3-[(2S)-3-[4-(2-carbamimidamidoethyl)piperidin-1-y...)
Affinity DataKi:  46nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23890(3-amidinophenylalanine deriv., 34 | 4-({4-[(2S)-3-...)
Affinity DataKi:  50nM ΔG°:  -41.7kJ/molepH: 8.0 T: 25°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM23904(3-[(2S)-3-[4-(2-carbamimidamidoethyl)piperidin-1-y...)
Affinity DataKi:  51nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23912(3-[(2S)-3-[4-(2-carbamimidamidoethyl)piperidin-1-y...)
Affinity DataKi:  53nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23876(3-[(2S)-3-[4-(3-carbamimidamidopropanoyl)piperazin...)
Affinity DataKi:  53nM ΔG°:  -41.5kJ/molepH: 8.0 T: 25°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM23892(3-[(2S)-2-[(9,10-dioxo-9,10-dihydroanthracene-2-)s...)
Affinity DataKi:  54nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23867(3-[(2S)-3-[4-(3-carbamimidamidopropanoyl)piperazin...)
Affinity DataKi:  57nM ΔG°:  -41.3kJ/molepH: 8.0 T: 25°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072859(3-[3-(4-Methyl-piperidin-1-yl)-3-oxo-2-(2,4,6-trim...)
Affinity DataKi:  59nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23870(3-[(2S)-3-[4-(4-carbamimidamidobutanoyl)piperazin-...)
Affinity DataKi:  61nM ΔG°:  -41.2kJ/molepH: 8.0 T: 25°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23888(3-amidinophenylalanine deriv., 32 | 4-({4-[(2S)-3-...)
Affinity DataKi:  61nM ΔG°:  -41.2kJ/molepH: 8.0 T: 25°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23874(3-[(2S)-3-[4-(3-carbamimidamidopropanoyl)-1,4-diaz...)
Affinity DataKi:  65nM ΔG°:  -41.0kJ/molepH: 8.0 T: 25°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50060049(3-[2-(Naphthalene-2-sulfonylamino)-3-oxo-3-piperid...)
Affinity DataKi:  65nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23903(3-[(2S)-3-[4-(2-carbamimidamidoethyl)piperidin-1-y...)
Affinity DataKi:  72nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072847(3-[2-(9,10-Dioxo-9,10-dihydro-anthracene-2-sulfony...)
Affinity DataKi:  74nMAssay Description:Inhibitory activity against bovine trypsin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23919(2-amino-N-(3-{[(2S)-1-[4-(2-aminoethyl)piperidin-1...)
Affinity DataKi:  75nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bovine)
Institut FüR Biochemie

Curated by ChEMBL
LigandPNGBDBM50072857(3-[3-(4-Methyl-piperidin-1-yl)-3-oxo-2-(2,4,6-trii...)
Affinity DataKi:  75nMAssay Description:Inhibitory activity against bovine thrombin expressed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23898(3-amidinophenylalanine deriv., 42 | 4-({1-[(2S)-3-...)
Affinity DataKi:  84nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Curacyte Chemistry

LigandPNGBDBM23904(3-[(2S)-3-[4-(2-carbamimidamidoethyl)piperidin-1-y...)
Affinity DataKi:  88nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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