TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of dimerization of HIV1 protease 150V mutantMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Inhibition of wild type HIV1 protease dimerizationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Inhibition of dimerization of HIV1 protease ANAM-11 mutantMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 240nMAssay Description:Inhibition of dimerization of HIV1 protease V82A mutantMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
Affinity DataKi: 380nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Inhibition of wild type HIV1 protease dimerizationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 410nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 420nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Inhibition of dimerization of HIV1 protease D30N mutantMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Inhibition of dimerization of HIV1 protease G48V/L90M mutantMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 530nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 560nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 790nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 900nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 1.90E+3nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 2.30E+3nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 4.30E+3nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 4.80E+3nMAssay Description:Inhibition of dimerization of HIV1 protease MDR-HM mutantMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 5.25E+3nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 6.00E+3nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 6.20E+3nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 7.00E+3nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 8.40E+3nMAssay Description:Inhibition of wild type HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 9.70E+3nMAssay Description:Inhibition of wild type HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 1.03E+4nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+4nMAssay Description:Apparent binding constant against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+4nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+4nMAssay Description:Apparent binding constant against porcine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+4nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
Affinity DataKi: 4.10E+4nMAssay Description:Apparent binding constant against Human urokinaseMore data for this Ligand-Target Pair
Affinity DataKi: 5.50E+4nMAssay Description:Apparent binding constant against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 5.90E+4nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+4nMAssay Description:Apparent binding constant against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 8.70E+4nMAssay Description:Apparent binding constant against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 9.00E+4nMAssay Description:Apparent binding constant against Human urokinaseMore data for this Ligand-Target Pair
Affinity DataKi: 9.20E+4nMAssay Description:Apparent binding constant against Human urokinaseMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+5nMAssay Description:Apparent binding constant against Human urokinaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair