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Found 79 with Last Name = 'boggetto' and Initial = 'n'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156909(CHEMBL376817 | methyl (2S)-3-carbamoyl-2-[(2S)-2-[...)
Affinity DataKi:  80nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  100nMAssay Description:Inhibition of dimerization of HIV1 protease 150V mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156906(CHEMBL375050 | methyl (2S)-2-[(2S)-2-[(2S)-2-(4-{[...)
Affinity DataKi:  130nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191464(CHEMBL212749 | methyl (2S)-2-[(2S)-2-[(2S)-2-(4-{[...)
Affinity DataKi:  200nMAssay Description:Inhibition of wild type HIV1 protease dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  200nMAssay Description:Inhibition of dimerization of HIV1 protease ANAM-11 mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156901((S)-tert-butyl 5-((S)-1-amino-4-methyl-1-oxopentan...)
Affinity DataKi:  230nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  240nMAssay Description:Inhibition of dimerization of HIV1 protease V82A mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50051763(2-iodophenyl 6-(chloromethyl)-2-oxo-2H-chromene-3-...)
Affinity DataKi:  250nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156902((S)-methyl 2-((S)-2-((S)-2-(4-(2-(4-((2S,3S)-1-((2...)
Affinity DataKi:  250nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM23563(3-Carboxylate-coumarin deriv., 3 | CHEMBL13357 | p...)
Affinity DataKi:  340nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50051762(6-Chloromethyl-2-oxo-2H-chromene-3-carboxylic acid...)
Affinity DataKi:  380nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156903((S)-methyl 2-((2S,3R)-3-hydroxy-2-((2S,3S)-2-(4-(7...)
Affinity DataKi:  400nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50135844((2S,8S)-2-[({[({[(1S)-1-{[(1S,2R)-2-(benzyloxy)-1-...)
Affinity DataKi:  400nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  400nMAssay Description:Inhibition of wild type HIV1 protease dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156910((S)-tert-butyl 5-((S)-1-amino-4-methyl-1-oxopentan...)
Affinity DataKi:  410nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156908((S)-tert-butyl 5-((S)-1-amino-4-methyl-1-oxopentan...)
Affinity DataKi:  420nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  500nMAssay Description:Inhibition of dimerization of HIV1 protease D30N mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  500nMAssay Description:Inhibition of dimerization of HIV1 protease G48V/L90M mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156904((S)-tert-butyl 5-((S)-1-amino-4-methyl-1-oxopentan...)
Affinity DataKi:  530nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50074687(2-[2-(2-{4-[7-(3-{1-[1-(1-Methoxycarbonyl-2-methyl...)
Affinity DataKi:  560nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50051761(2-chlorophenyl 6-(chloromethyl)-2-oxo-2H-chromene-...)
Affinity DataKi:  790nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156911((S)-5-((S)-1-amino-4-methyl-1-oxopentan-2-ylamino)...)
Affinity DataKi:  900nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156905((S)-methyl 2-((2S,3R)-3-hydroxy-2-(4-(7-(4-((S)-1-...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156914((S)-methyl 2-((S)-2-((S)-2-(4-(7-(4-((2S,3S)-1-((2...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156913((S)-methyl 2-((2S,3R)-3-hydroxy-2-(4-(7-(4-((S)-1-...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156912(CHEMBL376602 | methyl (2S)-2-[(2S,3R)-2-[(2S,3R)-3...)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156907((S)-methyl 2-((S)-2-((S)-2-(4-(7-(4-((S)-5-amino-1...)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156902((S)-methyl 2-((S)-2-((S)-2-(4-(2-(4-((2S,3S)-1-((2...)
Affinity DataKi:  4.30E+3nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  4.80E+3nMAssay Description:Inhibition of dimerization of HIV1 protease MDR-HM mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50135845(Bicyclic Guanidinium Subunit | CHEMBL266754)
Affinity DataKi:  5.25E+3nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50135842(Bicyclic Guanidinium Subunit | CHEMBL386994)
Affinity DataKi:  6.00E+3nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156914((S)-methyl 2-((S)-2-((S)-2-(4-(7-(4-((2S,3S)-1-((2...)
Affinity DataKi:  6.20E+3nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50135847(Bicyclic Guanidinium Subunit | CHEMBL404936)
Affinity DataKi:  7.00E+3nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191465(CHEMBL386205 | methyl (2S)-2-[(2R)-2-[(2S)-2-[4-({...)
Affinity DataKi:  8.40E+3nMAssay Description:Inhibition of wild type HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191466(CHEMBL426149 | methyl (2S)-2-[(2R)-2-[(2S)-2-(4-{[...)
Affinity DataKi:  9.70E+3nMAssay Description:Inhibition of wild type HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156905((S)-methyl 2-((2S,3R)-3-hydroxy-2-(4-(7-(4-((S)-1-...)
Affinity DataKi:  1.03E+4nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Cnrs-Cercoa

Curated by ChEMBL
LigandPNGBDBM50368614(CHEMBL540392)
Affinity DataKi:  1.20E+4nMAssay Description:Apparent binding constant against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50051760(6-Chloromethyl-2-oxo-2H-chromene-3-carboxylic acid...)
Affinity DataKi:  1.60E+4nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Cnrs-Cercoa

Curated by ChEMBL
LigandPNGBDBM50047473(CHEMBL38512 | N-[3-(11-Bromomethyl-3,6,9-trioxo-2,...)
Affinity DataKi:  2.00E+4nMAssay Description:Apparent binding constant against porcine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50051764(6-Chloromethyl-2-oxo-2H-chromene-3-carboxylic acid...)
Affinity DataKi:  3.30E+4nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Cnrs-Cercoa

Curated by ChEMBL
LigandPNGBDBM50368615(CHEMBL553244)
Affinity DataKi:  4.10E+4nMAssay Description:Apparent binding constant against Human urokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Cnrs-Cercoa

Curated by ChEMBL
LigandPNGBDBM50047473(CHEMBL38512 | N-[3-(11-Bromomethyl-3,6,9-trioxo-2,...)
Affinity DataKi:  5.50E+4nMAssay Description:Apparent binding constant against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50051765(6-Chloromethyl-2-oxo-2H-chromene-3-carboxylic acid...)
Affinity DataKi:  5.90E+4nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Cnrs-Cercoa

Curated by ChEMBL
LigandPNGBDBM50047476(4-(4-Amino-butyl)-11-bromomethyl-2,5,8-triaza-bicy...)
Affinity DataKi:  8.00E+4nMAssay Description:Apparent binding constant against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Cnrs-Cercoa

Curated by ChEMBL
LigandPNGBDBM50368613(CHEMBL557221)
Affinity DataKi:  8.70E+4nMAssay Description:Apparent binding constant against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Cnrs-Cercoa

Curated by ChEMBL
LigandPNGBDBM50368614(CHEMBL540392)
Affinity DataKi:  9.00E+4nMAssay Description:Apparent binding constant against Human urokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Cnrs-Cercoa

Curated by ChEMBL
LigandPNGBDBM50047473(CHEMBL38512 | N-[3-(11-Bromomethyl-3,6,9-trioxo-2,...)
Affinity DataKi:  9.20E+4nMAssay Description:Apparent binding constant against Human urokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Cnrs-Cercoa

Curated by ChEMBL
LigandPNGBDBM50368613(CHEMBL557221)
Affinity DataKi:  5.00E+5nMAssay Description:Apparent binding constant against Human urokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156910((S)-tert-butyl 5-((S)-1-amino-4-methyl-1-oxopentan...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156908((S)-tert-butyl 5-((S)-1-amino-4-methyl-1-oxopentan...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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