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Found 380 with Last Name = 'boi' and Initial = 'c'
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50143282((-)-cytisine | (1R,5S)-1,2,3,4,5,6-Hexahydro-1,5-m...)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50057463(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  0.450nMAssay Description:The binding affinity of the compound was determined towards Alpha-1B adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073570(2-(4-Furan-2-yl-piperazin-1-yl)-6,7-dimethoxy-quin...)
Affinity DataKi:  0.460nMAssay Description:The binding affinity of the compound was determined towards Alpha-1B adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50143282((-)-cytisine | (1R,5S)-1,2,3,4,5,6-Hexahydro-1,5-m...)
Affinity DataKi:  0.480nMAssay Description:Displacement of (+/-)-[3H]epibatidine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073570(2-(4-Furan-2-yl-piperazin-1-yl)-6,7-dimethoxy-quin...)
Affinity DataKi:  0.720nMAssay Description:The binding affinity of the compound was determined towards Alpha-1A adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073570(2-(4-Furan-2-yl-piperazin-1-yl)-6,7-dimethoxy-quin...)
Affinity DataKi:  1.39nMAssay Description:The binding affinity of the compound was determined towards Alpha-1C adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073563(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  1.48nMAssay Description:The binding affinity of the compound was determined towards Alpha-1A adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073563(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  1.57nMAssay Description:The binding affinity of the compound was determined towards Alpha-1B adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073563(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  1.59nMAssay Description:The binding affinity of the compound was determined towards Alpha-1C adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Lausanne

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  2.06nMAssay Description:Binding affinity towards mu receptor in rat brain using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279279(1-Phenyl-3-(cytisin-12-yl)-1-propanone | CHEMBL502...)
Affinity DataKi:  2.60nMAssay Description:Displacement of (+/-)-[3H]epibatidine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50240956((1R,5S)-3-(3-Oxo-butyl)-1,2,3,4,5,6-hexahydro-1,5-...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073573(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  4.43nMAssay Description:The binding affinity of the compound was determined towards Alpha-1B adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279280(1-(4-Fluorophenyl)-3-(cytisin-12-yl)-1-propanone |...)
Affinity DataKi:  5.30nMAssay Description:Displacement of (+/-)-[3H]epibatidine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073556(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  5.43nMAssay Description:The binding affinity of the compound was determined towards Alpha-1B adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073573(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  5.68nMAssay Description:The binding affinity of the compound was determined towards Alpha-1A adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Lausanne

Curated by ChEMBL
LigandPNGBDBM50106278(3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-thiazol...)
Affinity DataKi:  6.41nMAssay Description:Binding affinity towards mu receptor in rat brain using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279279(1-Phenyl-3-(cytisin-12-yl)-1-propanone | CHEMBL502...)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279210(CHEMBL525735 | N-[2-(Pyridin-4-yl)ethyl]cytisine)
Affinity DataKi:  7.20nMAssay Description:Displacement of (+/-)-[3H]epibatidine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Recordati

Curated by ChEMBL
LigandPNGBDBM50057463(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  7.5nMAssay Description:The binding affinity of the compound was determined towards Alpha-1A adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Lausanne

Curated by ChEMBL
LigandPNGBDBM50106280(3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-oxazoli...)
Affinity DataKi:  7.86nMAssay Description:Binding affinity towards mu receptor in rat brain using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073556(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  8.17nMAssay Description:The binding affinity of the compound was determined towards Alpha-1C adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073565(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  8.56nMAssay Description:The binding affinity of the compound was determined towards Alpha-1B adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Lausanne

Curated by ChEMBL
LigandPNGBDBM50106284(3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-thiazol...)
Affinity DataKi:  8.57nMAssay Description:Binding affinity towards mu receptor in rat brain using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50240956((1R,5S)-3-(3-Oxo-butyl)-1,2,3,4,5,6-hexahydro-1,5-...)
Affinity DataKi:  8.70nMAssay Description:Displacement of (+/-)-[3H]epibatidine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073566(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  9.05nMAssay Description:The binding affinity of the compound was determined towards Alpha-1B adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50057463(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  10.3nMAssay Description:The binding affinity of the compound was determined towards Alpha-1C adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073556(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  11.0nMAssay Description:The binding affinity of the compound was determined towards Alpha-1A adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279280(1-(4-Fluorophenyl)-3-(cytisin-12-yl)-1-propanone |...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073559(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  14.7nMAssay Description:The binding affinity of the compound was determined towards Alpha-1B adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279277(1-Phenyl-2-(cytisin-12-yl)-1-ethanone | CHEMBL5020...)
Affinity DataKi:  17nMAssay Description:Displacement of (+/-)-[3H]epibatidine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073565(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  18.9nMAssay Description:The binding affinity of the compound was determined towards Alpha-1C adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073565(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  18.9nMAssay Description:The binding affinity of the compound was determined towards Alpha-1A adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073573(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  19.4nMAssay Description:The binding affinity of the compound was determined towards Alpha-1C adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073566(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  23.7nMAssay Description:The binding affinity of the compound was determined towards Alpha-1C adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279206((1R,5S)-3-Phenethyl-1,2,3,4,5,6-hexahydro-1,5-meth...)
Affinity DataKi:  28nMAssay Description:Displacement of (+/-)-[3H]epibatidine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279333(3-(Cytisin-12-yl)propionamide | CHEMBL483804)
Affinity DataKi:  35nMAssay Description:Displacement of (+/-)-[3H]epibatidine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Lausanne

Curated by ChEMBL
LigandPNGBDBM50106282(3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrolid...)
Affinity DataKi:  35.2nMAssay Description:Binding affinity towards mu receptor in rat brain using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073566(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  36.2nMAssay Description:The binding affinity of the compound was determined towards Alpha-1A adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Lausanne

Curated by ChEMBL
LigandPNGBDBM50106283(3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-2,2-dim...)
Affinity DataKi:  37.7nMAssay Description:Binding affinity towards mu receptor in rat brain using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279242((1R,5S)-3-(3-Phenyl-propyl)-1,2,3,4,5,6-hexahydro-...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279367((1R,5S)-3-Pentyl-1,2,3,4,5,6-hexahydro-1,5-methano...)
Affinity DataKi:  43.5nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Lausanne

Curated by ChEMBL
LigandPNGBDBM50106281(3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-2,2-dim...)
Affinity DataKi:  46.9nMAssay Description:Binding affinity towards mu receptor in rat brain using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Lausanne

Curated by ChEMBL
LigandPNGBDBM50106279(3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-2,2-dim...)
Affinity DataKi:  50.4nMAssay Description:Binding affinity towards mu receptor in rat brain using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Lausanne

Curated by ChEMBL
LigandPNGBDBM50106275(3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-oxazoli...)
Affinity DataKi:  58.9nMAssay Description:Binding affinity towards mu receptor in rat brain using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279242((1R,5S)-3-(3-Phenyl-propyl)-1,2,3,4,5,6-hexahydro-...)
Affinity DataKi:  63nMAssay Description:Displacement of (+/-)-[3H]epibatidine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279206((1R,5S)-3-Phenethyl-1,2,3,4,5,6-hexahydro-1,5-meth...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Lausanne

Curated by ChEMBL
LigandPNGBDBM50106277(3-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-2,2-dim...)
Affinity DataKi:  96.5nMAssay Description:Binding affinity towards mu receptor in rat brain using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50038163((6,7-Dichloro-2,3-dioxo-3,4-dihydro-2H-quinoxalin-...)
Affinity DataKi:  110nMAssay Description:Binding affinity for glycine site-NMDA receptor was determined by the ability to displace [3H]glycine in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Recordati

Curated by ChEMBL
LigandPNGBDBM50073559(1-[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-piper...)
Affinity DataKi:  156nMAssay Description:The binding affinity of the compound was determined towards Alpha-1A adrenergic receptor in the COS cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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