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Found 78 with Last Name = 'boigegrain' and Initial = 'r'
TargetNeurotensin(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM85050(CAS_184162-64-9 | SR 142948A | SR142948 | SR142948...)
Affinity DataKi:  0.170nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeurotensin/neuromedin N(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM85050(CAS_184162-64-9 | SR 142948A | SR142948 | SR142948...)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeurotensin(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50248034(2-{[1-(7-Chloro-quinolin-4-yl)-5-(2,6-dimethoxy-ph...)
Affinity DataKi:  3.90nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280583(CHEMBL423832 | N*2*,N*2*-Diethyl-2-methyl-N*1*-(6-...)
Affinity DataKi:  112nMAssay Description:Compound was tested for its affinity for muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267344((S)-3-amino-1-(4-(benzyloxy)phenyl)-4-(1H-imidazol...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267344((S)-3-amino-1-(4-(benzyloxy)phenyl)-4-(1H-imidazol...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267345((S)-3-amino-1-(2,4-difluorophenyl)-4-(1H-imidazol-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267346((S)-3-amino-1-(3,4-dichlorophenyl)-4-(1H-imidazol-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267371((S)-3-amino-4-(1H-imidazol-4-yl)-1-(perfluoropheny...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267467((S)-3-amino-4-(1H-imidazol-4-yl)-1-(naphthalen-1-y...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267468((S)-3-amino-4-(1H-imidazol-4-yl)-1-(naphthalen-2-y...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267469((S)-3-amino-1-(benzo[d][1,3]dioxol-5-yl)-4-(1H-imi...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267343((S)-3-amino-4-(1H-imidazol-4-yl)-1-(4-phenoxypheny...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267975((S)-3-Amino-1-(4-bromo-phenyl)-4-(1H-imidazol-4-yl...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267972((S)-3-Amino-4-(1H-imidazol-4-yl)-1-phenyl-butan-2-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267973((S)-3-amino-1-(4-fluorophenyl)-4-(1H-imidazol-4-yl...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267342((S)-3-Amino-4-(1H-imidazol-4-yl)-1-(4-methoxy-phen...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267341((S)-3-amino-4-(1H-imidazol-4-yl)-1-p-tolylbutan-2-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267976((S)-3-Amino-1-biphenyl-4-yl-4-(1H-imidazol-4-yl)-b...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267975((S)-3-Amino-1-(4-bromo-phenyl)-4-(1H-imidazol-4-yl...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267974((S)-3-Amino-1-(4-chloro-phenyl)-4-(1H-imidazol-4-y...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50280609(2-[6-(1-Ethyl-pyrrolidin-2-ylamino)-4-methyl-pyrid...)
Affinity DataIC50:  8nMAssay Description:Displacement of [3H]-pirenzepine from cerebral Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280589((+)-(1-Ethyl-pyrrolidin-2-yl)-(6-phenyl-5-propyl-p...)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]-pirenzepine from cerebral Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267345((S)-3-amino-1-(2,4-difluorophenyl)-4-(1H-imidazol-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50280589((+)-(1-Ethyl-pyrrolidin-2-yl)-(6-phenyl-5-propyl-p...)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]-pirenzepine from cerebral Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM29578(isatin Michael acceptor (IMA) analogue, 13a)
Affinity DataIC50:  12nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267976((S)-3-Amino-1-biphenyl-4-yl-4-(1H-imidazol-4-yl)-b...)
Affinity DataIC50:  12.5nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267468((S)-3-amino-4-(1H-imidazol-4-yl)-1-(naphthalen-2-y...)
Affinity DataIC50:  14.5nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267973((S)-3-amino-1-(4-fluorophenyl)-4-(1H-imidazol-4-yl...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267341((S)-3-amino-4-(1H-imidazol-4-yl)-1-p-tolylbutan-2-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267343((S)-3-amino-4-(1H-imidazol-4-yl)-1-(4-phenoxypheny...)
Affinity DataIC50:  16nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267346((S)-3-amino-1-(3,4-dichlorophenyl)-4-(1H-imidazol-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50280612((1-Ethyl-pyrrolidin-2-yl)-(6-methyl-5-phenyl-pyrid...)
Affinity DataIC50:  20nMAssay Description:Displacement of [3H]-pirenzepine from cerebral Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280599(CHEMBL168670 | N*2*,N*2*-Diethyl-N*1*-(6-isobutyl-...)
Affinity DataIC50:  20nMAssay Description:Displacement of [3H]-pirenzepine from cerebral Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267469((S)-3-amino-1-(benzo[d][1,3]dioxol-5-yl)-4-(1H-imi...)
Affinity DataIC50:  25nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50280589((+)-(1-Ethyl-pyrrolidin-2-yl)-(6-phenyl-5-propyl-p...)
Affinity DataIC50:  30nMAssay Description:Displacement of [3H]-pirenzepine from cerebral Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280587(CHEMBL167016 | N*1*-(5,6-Diphenyl-pyridazin-3-yl)-...)
Affinity DataIC50:  40nMAssay Description:Displacement of [3H]-pirenzepine from cerebral Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267972((S)-3-Amino-4-(1H-imidazol-4-yl)-1-phenyl-butan-2-...)
Affinity DataIC50:  40nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50280617(CHEMBL169663 | N'-(6,7-Dihydro-5H-benzo[6,7]cycloh...)
Affinity DataIC50:  50nMAssay Description:Displacement of [3H]-pirenzepine from cerebral Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280605(CHEMBL353869 | N*2*,N*2*-Diethyl-2-methyl-N*1*-(5-...)
Affinity DataIC50:  50nMAssay Description:Displacement of [3H]-pirenzepine from cerebral Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50370977(CHEMBL556799)
Affinity DataIC50:  70nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50280583(CHEMBL423832 | N*2*,N*2*-Diethyl-2-methyl-N*1*-(6-...)
Affinity DataIC50:  110nMAssay Description:Displacement of [3H]-pirenzepine from cerebral Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280582(2-[6-(2-Diethylamino-2-methyl-propylamino)-4-propy...)
Affinity DataIC50:  130nMAssay Description:Displacement of [3H]-pirenzepine from cerebral Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280603(CHEMBL352419 | N,N-Dimethyl-N'-(2-methyl-biphenyl-...)
Affinity DataIC50:  140nMAssay Description:Displacement of [3H]-pirenzepine from cerebral Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267342((S)-3-Amino-4-(1H-imidazol-4-yl)-1-(4-methoxy-phen...)
Affinity DataIC50:  150nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50280616((5,6-Diphenyl-pyridazin-3-yl)-(2-morpholin-4-yl-et...)
Affinity DataIC50:  170nMAssay Description:Displacement of [3H]-pirenzepine from cerebral Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280588(CHEMBL165815 | N*2*,N*2*-Diethyl-2-methyl-N*1*-(6-...)
Affinity DataIC50:  180nMAssay Description:Displacement of [3H]-pirenzepine from cerebral Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistidinol dehydrogenase(Brucella suis)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50267467((S)-3-amino-4-(1H-imidazol-4-yl)-1-(naphthalen-1-y...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50280614(CHEMBL151705 | N,N-Dimethyl-N'-(4-methyl-6-phenyl-...)
Affinity DataIC50:  230nMAssay Description:Displacement of [3H]-pirenzepine from cerebral Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280594(CHEMBL168674 | N'-(6,7-Dihydro-5H-benzo[6,7]cycloh...)
Affinity DataIC50:  240nMAssay Description:Displacement of [3H]-pirenzepine from cerebral Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
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