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Found 62 with Last Name = 'bojanic' and Initial = 'd'
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286792((R)-2-[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4...)
Affinity DataIC50:  2.5nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286804((R)-2-[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4...)
Affinity DataIC50:  5.30nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286795((R)-2-[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4...)
Affinity DataIC50:  8nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286800((R)-2-[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4...)
Affinity DataIC50:  8nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286802(3-[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  62nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286791(4-[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  140nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050632(8-ETHYL-6-METHOXY-3-METHYL-8H-1,3A,7,8,9-PENTAAZA-...)
Affinity DataIC50:  156nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050632(8-ETHYL-6-METHOXY-3-METHYL-8H-1,3A,7,8,9-PENTAAZA-...)
Affinity DataIC50:  190nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050636(8-Cyclopropyl-4-methyl-8H-1,3a,7,8,9-pentaaza-dibe...)
Affinity DataIC50:  217nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286805(CHEMBL170121 | [(R)-2-{(S)-2-[(Azepane-1-carbonyl)...)
Affinity DataIC50:  220nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050633(8-Ethyl-4-methyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,...)
Affinity DataIC50:  245nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050628(8-Ethyl-6-methoxy-8H-1,3a,7,8,9-pentaaza-dibenzo[e...)
Affinity DataIC50:  258nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286793((R)-2-[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4...)
Affinity DataIC50:  295nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286801(3-(3-{[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4...)
Affinity DataIC50:  420nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050640(8-Ethyl-3-methyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,...)
Affinity DataIC50:  425nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050628(8-Ethyl-6-methoxy-8H-1,3a,7,8,9-pentaaza-dibenzo[e...)
Affinity DataIC50:  598nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286798(2-[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  730nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50280306(8-Ethyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,h]azulene...)
Affinity DataIC50:  775nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286794(2-{[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-me...)
Affinity DataIC50:  1.10E+3nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050634((8-Ethyl-3-methyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e...)
Affinity DataIC50:  1.10E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50280315(3,8-Diethyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,h]azu...)
Affinity DataIC50:  1.10E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050640(8-Ethyl-3-methyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,...)
Affinity DataIC50:  1.22E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286803((S)-2-[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4...)
Affinity DataIC50:  1.32E+3nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM1517(2-ethyl-7-methyl-2,4,9,15-tetraazatricyclo[9.4.0.0...)
Affinity DataIC50:  1.50E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050633(8-Ethyl-4-methyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,...)
Affinity DataIC50:  1.62E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50280311(8-Ethyl-3-methyl-6-pyrrolidin-1-yl-8H-1,3a,7,8,9-p...)
Affinity DataIC50:  1.77E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50280308(8-Ethyl-6-pyrrolidin-1-yl-8H-1,3a,7,8,9-pentaaza-d...)
Affinity DataIC50:  2.00E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050636(8-Cyclopropyl-4-methyl-8H-1,3a,7,8,9-pentaaza-dibe...)
Affinity DataIC50:  2.05E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataIC50:  2.11E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050637((8-Ethyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,h]azulen...)
Affinity DataIC50:  2.19E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050634((8-Ethyl-3-methyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e...)
Affinity DataIC50:  2.40E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50280311(8-Ethyl-3-methyl-6-pyrrolidin-1-yl-8H-1,3a,7,8,9-p...)
Affinity DataIC50:  2.70E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050638(8-Ethyl-2-methyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,...)
Affinity DataIC50:  2.75E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50280313(8-Ethyl-3-methyl-7H,8H-1,3a,7,8,9-pentaaza-dibenzo...)
Affinity DataIC50:  3.20E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286799(6-[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >3.50E+3nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286796(5-[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >3.50E+3nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286797((R)-2-[(R)-2-{(S)-2-[(Azepane-1-carbonyl)-amino]-4...)
Affinity DataIC50: >3.50E+3nMAssay Description:Binding affinity against ETA receptor from dog spleen membranes using [125I]-ET1 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50280308(8-Ethyl-6-pyrrolidin-1-yl-8H-1,3a,7,8,9-pentaaza-d...)
Affinity DataIC50:  3.90E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050637((8-Ethyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,h]azulen...)
Affinity DataIC50:  3.90E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50280315(3,8-Diethyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,h]azu...)
Affinity DataIC50:  5.63E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataIC50:  6.44E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50280312(8-Ethyl-4-methyl-8H-1,2,3,3a,7,8,9-heptaaza-dibenz...)
Affinity DataIC50:  6.72E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50280309(8-Ethyl-7H,8H-1,3a,7,8,9-pentaaza-dibenzo[e,h]azul...)
Affinity DataIC50:  6.98E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050630(8-Cyclopropyl-3-methyl-8H-1,2,3a,7,8,9-hexaaza-dib...)
Affinity DataIC50:  7.82E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM1517(2-ethyl-7-methyl-2,4,9,15-tetraazatricyclo[9.4.0.0...)
Affinity DataIC50:  1.03E+4nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050638(8-Ethyl-2-methyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,...)
Affinity DataIC50:  1.12E+4nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50280306(8-Ethyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,h]azulene...)
Affinity DataIC50:  1.12E+4nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050630(8-Cyclopropyl-3-methyl-8H-1,2,3a,7,8,9-hexaaza-dib...)
Affinity DataIC50:  1.15E+4nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50280313(8-Ethyl-3-methyl-7H,8H-1,3a,7,8,9-pentaaza-dibenzo...)
Affinity DataIC50:  1.22E+4nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50280314(3,8-Diethyl-8H-1,2,3a,7,8,9-hexaaza-dibenzo[e,h]az...)
Affinity DataIC50:  2.02E+4nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
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