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Found 36 with Last Name = 'bondon' and Initial = 'a'
TargetHistone deacetylase 1(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314133(CHEMBL1093713 | N-(3,5-Dimethylphenyl)-N'-hydroxyo...)
Affinity DataIC50:  17nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314134(CHEMBL1093041 | N-(3-Ethylphenyl)-N'-hydroxyoctane...)
Affinity DataIC50:  27nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314133(CHEMBL1093713 | N-(3,5-Dimethylphenyl)-N'-hydroxyo...)
Affinity DataIC50:  30nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314135(CHEMBL1093359 | N-(3,4-Dimethylphenyl)-N'-hydroxyo...)
Affinity DataIC50:  30nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314134(CHEMBL1093041 | N-(3-Ethylphenyl)-N'-hydroxyoctane...)
Affinity DataIC50:  35nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314135(CHEMBL1093359 | N-(3,4-Dimethylphenyl)-N'-hydroxyo...)
Affinity DataIC50:  56nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314136(CHEMBL1089339 | N-Hydroxy-N'-(3-methylphenyl)octan...)
Affinity DataIC50:  57nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314136(CHEMBL1089339 | N-Hydroxy-N'-(3-methylphenyl)octan...)
Affinity DataIC50:  58nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314137(CHEMBL1091487 | N-Hydroxy-N'-(4-methoxyphenyl)octa...)
Affinity DataIC50:  71nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314138(CHEMBL1092762 | N-Hydroxy-N'-(4-methylphenyl)octan...)
Affinity DataIC50:  76nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314138(CHEMBL1092762 | N-Hydroxy-N'-(4-methylphenyl)octan...)
Affinity DataIC50:  114nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  119nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314137(CHEMBL1091487 | N-Hydroxy-N'-(4-methoxyphenyl)octa...)
Affinity DataIC50:  137nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  147nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistone deacetylase 1(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314139(CHEMBL1093042 | N-(4-Ethylphenyl)-N'-hydroxyoctane...)
Affinity DataIC50:  149nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314139(CHEMBL1093042 | N-(4-Ethylphenyl)-N'-hydroxyoctane...)
Affinity DataIC50:  240nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314140(CHEMBL1076794 | N-Hydroxy-N'-(2-methylphenyl)octan...)
Affinity DataIC50:  576nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314141(CHEMBL1092032 | N-(2,4-Dimethylphenyl)-N'-hydroxyo...)
Affinity DataIC50:  638nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314141(CHEMBL1092032 | N-(2,4-Dimethylphenyl)-N'-hydroxyo...)
Affinity DataIC50:  1.10E+3nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314142(CHEMBL1093040 | N-(2-Ethylphenyl)-N'-hydroxyoctane...)
Affinity DataIC50:  1.10E+3nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314143(CHEMBL1093043 | N-(2,3-Dimethylphenyl)-N'-hydroxyo...)
Affinity DataIC50:  1.11E+3nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314144(CHEMBL1093357 | N-(2,5-Dimethylphenyl)-N'-hydroxyo...)
Affinity DataIC50:  1.14E+3nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314144(CHEMBL1093357 | N-(2,5-Dimethylphenyl)-N'-hydroxyo...)
Affinity DataIC50:  1.35E+3nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314140(CHEMBL1076794 | N-Hydroxy-N'-(2-methylphenyl)octan...)
Affinity DataIC50:  1.35E+3nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314143(CHEMBL1093043 | N-(2,3-Dimethylphenyl)-N'-hydroxyo...)
Affinity DataIC50:  1.75E+3nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314142(CHEMBL1093040 | N-(2-Ethylphenyl)-N'-hydroxyoctane...)
Affinity DataIC50:  2.26E+3nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314145(CHEMBL1093358 | N-(2,6-Dimethylphenyl)-N'-hydroxyo...)
Affinity DataIC50:  4.99E+3nMAssay Description:Ex vivo inhibition of human HDAC3 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Umr Cnrs 6026-Universit£

Curated by ChEMBL
LigandPNGBDBM50314145(CHEMBL1093358 | N-(2,6-Dimethylphenyl)-N'-hydroxyo...)
Affinity DataIC50:  1.16E+4nMAssay Description:Ex vivo inhibition of human HDAC1 in human Caco2 cells by flurometric cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte nuclear factor 4-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50304340(2-Nitro-naphtho[2,1-b]furan | 2-nitronaphtho[2,1-b...)
Affinity DataEC50:  2.09E+3nMAssay Description:Agonist activity at human full length HNF4alpha nuclear receptor expressed in human HepG2/C3A cells cotransfected with LexADBD assessed as increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte nuclear factor 4-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50304339(8-Methoxy-2-nitro-naphtho[2,1-b]furan | 8-methoxy-...)
Affinity DataEC50:  2.33E+3nMAssay Description:Agonist activity at human full length HNF4alpha nuclear receptor expressed in human HepG2/C3A cells cotransfected with LexADBD assessed as increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte nuclear factor 4-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50304338(1-Methyl-2-nitro-naphtho[2,1-b]furan | 1-methyl-2-...)
Affinity DataEC50:  1.28E+3nMAssay Description:Agonist activity at human full length HNF4alpha nuclear receptor expressed in human HepG2/C3A cells cotransfected with LexADBD assessed as increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte nuclear factor 4-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50304342(CHEMBL611816 | naphtho[2,1-b]furan-2-carboxamide)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human full length HNF4alpha nuclear receptor expressed in human HepG2/C3A cells cotransfected with LexADBD assessed as increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte nuclear factor 4-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50304336(2-Nitro-naphtho[2,1-b]furan-7-ol | 2-nitronaphtho[...)
Affinity DataEC50:  1.95E+3nMAssay Description:Agonist activity at human full length HNF4alpha nuclear receptor expressed in human HepG2/C3A cells cotransfected with LexADBD assessed as increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte nuclear factor 4-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM22594(7-methoxy-4-nitro-5-oxatricyclo[7.4.0.0^{2,6}]trid...)
Affinity DataEC50:  1.47E+3nMAssay Description:Agonist activity at human full length HNF4alpha nuclear receptor expressed in human HepG2/C3A cells cotransfected with LexADBD assessed as increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte nuclear factor 4-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50304341(7-Methoxy-2-nitro-naphtho[2,1-b]furan | 7-methoxy-...)
Affinity DataEC50:  2.57E+3nMAssay Description:Agonist activity at human full length HNF4alpha nuclear receptor expressed in human HepG2/C3A cells cotransfected with LexADBD assessed as increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte nuclear factor 4-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50304337(2-(2-Nitro-naphtho[2,1-b]furan-1-yl)-ethanol | 2-(...)
Affinity DataEC50:  1.22E+3nMAssay Description:Agonist activity at human full length HNF4alpha nuclear receptor expressed in human HepG2/C3A cells cotransfected with LexADBD assessed as increase i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed