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Found 27 with Last Name = 'boonyarat' and Initial = 'c'
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50256010(3-{2,4-dimethyl-5-[2-oxo-5-(N'-phenylhydrazinocarb...)
Affinity DataIC50:  40nMAssay Description:Inhibition of PDGFRbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  50nMAssay Description:Inhibition of BuChE in human serum using butyrylthiocholine iodide as substrate measured every 30s for 5 mins by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM4811((Z)-3-[2,4-dimethyl-5-(2-oxo-1,2-dihydro-indol-3-y...)
Affinity DataIC50:  50nMAssay Description:Inhibition of PDGFRbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50256010(3-{2,4-dimethyl-5-[2-oxo-5-(N'-phenylhydrazinocarb...)
Affinity DataIC50:  70nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50256010(3-{2,4-dimethyl-5-[2-oxo-5-(N'-phenylhydrazinocarb...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human FGFR1 expressed in insect cells by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50217602((Z)-3-(5-((6-(3,5-dimethoxyphenyl)-2-oxoindolin-3-...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human FGFR1 kinase expressed in insect cell by HTRF detection methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50217602((Z)-3-(5-((6-(3,5-dimethoxyphenyl)-2-oxoindolin-3-...)
Affinity DataIC50:  520nMAssay Description:Inhibition of human FGFR1 expressed in insect cells by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM4811((Z)-3-[2,4-dimethyl-5-(2-oxo-1,2-dihydro-indol-3-y...)
Affinity DataIC50:  680nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50217602((Z)-3-(5-((6-(3,5-dimethoxyphenyl)-2-oxoindolin-3-...)
Affinity DataIC50:  780nMAssay Description:Inhibition of PDGFRbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50217602((Z)-3-(5-((6-(3,5-dimethoxyphenyl)-2-oxoindolin-3-...)
Affinity DataIC50:  930nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM4901(3-(5-{[(3Z)-6-(3-methoxyphenyl)-2-oxo-2,3-dihydro-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human FGFR1 kinase expressed in insect cell by HTRF detection methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50330180((S)-3-((4-(6-methoxynaphthalen-2-yl)-1H-1,2,3-tria...)
Affinity DataIC50:  1.49E+3nMAssay Description:Inhibition of human recombinant BACE1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM4811((Z)-3-[2,4-dimethyl-5-(2-oxo-1,2-dihydro-indol-3-y...)
Affinity DataIC50:  1.81E+3nMAssay Description:Inhibition of human FGFR1 expressed in insect cells by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50256010(3-{2,4-dimethyl-5-[2-oxo-5-(N'-phenylhydrazinocarb...)
Affinity DataIC50:  3.48E+3nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of BuChE in human serum using butyrylthiocholine iodide as substrate measured every 30s for 5 mins by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM4901(3-(5-{[(3Z)-6-(3-methoxyphenyl)-2-oxo-2,3-dihydro-...)
Affinity DataIC50:  1.79E+4nMAssay Description:Inhibition of rhFGF2-induced cellular proliferation of HUVECMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50217602((Z)-3-(5-((6-(3,5-dimethoxyphenyl)-2-oxoindolin-3-...)
Affinity DataIC50:  1.82E+4nMAssay Description:Inhibition of rhFGF2-induced cellular proliferation of HUVECMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50496396(CHEMBL3127382)
Affinity DataIC50:  1.94E+4nMAssay Description:Inhibition of BuChE in human serum using butyrylthiocholine iodide as substrate measured every 30s for 5 mins by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM4900(3-(2,4-dimethyl-5-{[(3Z)-2-oxo-6-phenyl-2,3-dihydr...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of rhFGF2-induced cellular proliferation of HUVECMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM4811((Z)-3-[2,4-dimethyl-5-(2-oxo-1,2-dihydro-indol-3-y...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of rhFGF2-induced cellular proliferation of HUVECMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50496393(CHEMBL3127381)
Affinity DataIC50:  5.21E+4nMAssay Description:Inhibition of BuChE in human serum using butyrylthiocholine iodide as substrate measured every 30s for 5 mins by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50496394(CHEMBL3127383)
Affinity DataIC50:  6.43E+4nMAssay Description:Inhibition of BuChE in human serum using butyrylthiocholine iodide as substrate measured every 30s for 5 mins by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50217602((Z)-3-(5-((6-(3,5-dimethoxyphenyl)-2-oxoindolin-3-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50496392(CHEBI:69927 | Heptaphylline)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of BuChE in human serum using butyrylthiocholine iodide as substrate measured every 30s for 5 mins by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM4811((Z)-3-[2,4-dimethyl-5-(2-oxo-1,2-dihydro-indol-3-y...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50496395(7-Methoxyheptaphylline | CHEBI:69928 | CHEMBL46427...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of BuChE in human serum using butyrylthiocholine iodide as substrate measured every 30s for 5 mins by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50330180((S)-3-((4-(6-methoxynaphthalen-2-yl)-1H-1,2,3-tria...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant Cathepsin D by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed