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Found 48 with Last Name = 'bopp' and Initial = 's'
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50128678(CHEMBL310855 | N-(1-Carbamoyl-2-phenyl-ethyl)-2-(2...)
Affinity DataKi:  8.40nMAssay Description:Inhibitory activity against human Calpain 1 isolated from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50128679(CHEMBL77784 | N-(1-Carbamoyl-pentyl)-2-[2-(4-dimet...)
Affinity DataKi:  13.3nMAssay Description:Inhibitory activity against human Calpain 1 isolated from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50128680(CHEMBL80903 | N-(1-Benzyl-2-oxo-ethyl)-2-(2-naphth...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against human Calpain 1 isolated from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50073850((S)-2-((S)-2-Benzyloxycarbonylamino-3-methyl-butyr...)
Affinity DataKi:  15.5nMAssay Description:Inhibitory activity against human Calpain 1 isolated from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50073850((S)-2-((S)-2-Benzyloxycarbonylamino-3-methyl-butyr...)
Affinity DataKi:  18nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50128681(CHEMBL80933 | N-(1-Carbamoyl-2-phenyl-ethyl)-2-[2-...)
Affinity DataKi:  18.3nMAssay Description:Inhibitory activity against human Calpain 1 isolated from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50128679(CHEMBL77784 | N-(1-Carbamoyl-pentyl)-2-[2-(4-dimet...)
Affinity DataKi:  27nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50128682(CHEMBL80605 | N-(1-Carbamoyl-2-phenyl-ethyl)-2-[2-...)
Affinity DataKi:  27nMAssay Description:Inhibitory activity against human Calpain 1 isolated from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50128682(CHEMBL80605 | N-(1-Carbamoyl-2-phenyl-ethyl)-2-[2-...)
Affinity DataKi:  62nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50128681(CHEMBL80933 | N-(1-Carbamoyl-2-phenyl-ethyl)-2-[2-...)
Affinity DataKi:  83nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50128678(CHEMBL310855 | N-(1-Carbamoyl-2-phenyl-ethyl)-2-(2...)
Affinity DataKi:  99nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50112839(CHEMBL26631 | N-(1-Benzyl-2-oxo-ethyl)-2-styryl-be...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against human Calpain 1 isolated from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50112838(CHEMBL281874 | N-(1-Benzyl-2-oxo-ethyl)-benzamide)
Affinity DataKi:  1.08E+3nMAssay Description:Inhibitory activity against human Calpain 1 isolated from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50022775((m-Hydroxyphenyl)trimethylammonium dimethylcarbama...)
Affinity DataIC50:  40nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50022775((m-Hydroxyphenyl)trimethylammonium dimethylcarbama...)
Affinity DataIC50:  41nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50022775((m-Hydroxyphenyl)trimethylammonium dimethylcarbama...)
Affinity DataIC50:  53nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298426(1-(2,5-dichloro benzene)-sulfonyl-cis-2,6-dimethyl...)
Affinity DataIC50:  75nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298421(CHEMBL576005 | cis-2,6-dimethyl-1-methyl sulfonyl ...)
Affinity DataIC50:  75nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298426(1-(2,5-dichloro benzene)-sulfonyl-cis-2,6-dimethyl...)
Affinity DataIC50:  81nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298421(CHEMBL576005 | cis-2,6-dimethyl-1-methyl sulfonyl ...)
Affinity DataIC50:  85nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298421(CHEMBL576005 | cis-2,6-dimethyl-1-methyl sulfonyl ...)
Affinity DataIC50:  90nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298426(1-(2,5-dichloro benzene)-sulfonyl-cis-2,6-dimethyl...)
Affinity DataIC50:  90nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298427(1-(2-nitro benzene)-sulfonyl-cis-2,6-dimethylpiper...)
Affinity DataIC50:  180nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298427(1-(2-nitro benzene)-sulfonyl-cis-2,6-dimethylpiper...)
Affinity DataIC50:  185nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298428(1-(3-nitro benzene)-sulfonyl-cis-2,6-dimethylpiper...)
Affinity DataIC50:  186nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298428(1-(3-nitro benzene)-sulfonyl-cis-2,6-dimethylpiper...)
Affinity DataIC50:  192nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298427(1-(2-nitro benzene)-sulfonyl-cis-2,6-dimethylpiper...)
Affinity DataIC50:  195nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298428(1-(3-nitro benzene)-sulfonyl-cis-2,6-dimethylpiper...)
Affinity DataIC50:  200nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298425((2R,6S)-1-(4-chlorophenylsulfonyl)-2,6-dimethylpip...)
Affinity DataIC50:  312nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298425((2R,6S)-1-(4-chlorophenylsulfonyl)-2,6-dimethylpip...)
Affinity DataIC50:  318nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298425((2R,6S)-1-(4-chlorophenylsulfonyl)-2,6-dimethylpip...)
Affinity DataIC50:  325nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298423(1-(4-methyl benzene)-sulfonyl-cis-2,6-dimethylpipe...)
Affinity DataIC50:  362nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298422(1-benzene sulfonyl-cis-2,6-dimethyl piperidine | C...)
Affinity DataIC50:  362nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298423(1-(4-methyl benzene)-sulfonyl-cis-2,6-dimethylpipe...)
Affinity DataIC50:  365nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298423(1-(4-methyl benzene)-sulfonyl-cis-2,6-dimethylpipe...)
Affinity DataIC50:  368nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298422(1-benzene sulfonyl-cis-2,6-dimethyl piperidine | C...)
Affinity DataIC50:  388nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298422(1-benzene sulfonyl-cis-2,6-dimethyl piperidine | C...)
Affinity DataIC50:  392nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298424(1-(4-tert-butyl benzene)-sulfonyl-cis-2,6-dimethyl...)
Affinity DataIC50:  450nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298424(1-(4-tert-butyl benzene)-sulfonyl-cis-2,6-dimethyl...)
Affinity DataIC50:  458nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298424(1-(4-tert-butyl benzene)-sulfonyl-cis-2,6-dimethyl...)
Affinity DataIC50:  463nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50073850((S)-2-((S)-2-Benzyloxycarbonylamino-3-methyl-butyr...)
Affinity DataIC50:  700nMAssay Description:Inhibition of degradation of tyrosine kinase pp60src by Calpain 1 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50128682(CHEMBL80605 | N-(1-Carbamoyl-2-phenyl-ethyl)-2-[2-...)
Affinity DataIC50:  700nMAssay Description:Inhibition of degradation of tyrosine kinase pp60src by Calpain 1 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50128679(CHEMBL77784 | N-(1-Carbamoyl-pentyl)-2-[2-(4-dimet...)
Affinity DataIC50:  800nMAssay Description:Inhibition of degradation of tyrosine kinase pp60src by Calpain 1 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50128681(CHEMBL80933 | N-(1-Carbamoyl-2-phenyl-ethyl)-2-[2-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of degradation of tyrosine kinase pp60src by Calpain 1 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298429(1-(4-nitro benzene)-sulfonyl-cis-2,6-dimethylpiper...)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298429(1-(4-nitro benzene)-sulfonyl-cis-2,6-dimethylpiper...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50298429(1-(4-nitro benzene)-sulfonyl-cis-2,6-dimethylpiper...)
Affinity DataIC50:  1.21E+3nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Abbott

Curated by ChEMBL
LigandPNGBDBM50128678(CHEMBL310855 | N-(1-Carbamoyl-2-phenyl-ethyl)-2-(2...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of degradation of tyrosine kinase pp60src by Calpain 1 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed