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Found 232 with Last Name = 'borst' and Initial = 'aj'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50172158((S)-N-(1-(4-(4-chloro-2-(2-fluorophenylsulfonyl)ph...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309538(5-Ethyl-2-methyl-1-phenyl-1H-imidazole-4-carboxyli...)
Affinity DataKi:  1.03nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309540(2-Ethyl-5-methyl-1-phenyl-1H-imidazole-4-carboxyli...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309534(2,5-Dimethyl-1-phenyl-1H-imidazole-4-carboxylic ac...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354607(CHEMBL1834337)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354585(CHEMBL1834226)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354585(CHEMBL1834226)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317250(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methy...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303835(3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309537(2,5-dimethyl-1-phenyl-N-(2-(trifluoromethyl)benzyl...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354608(CHEMBL1834342)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354609(CHEMBL1834348)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354610(CHEMBL1834338)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354611(CHEMBL1834347)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354612(CHEMBL1834350)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354614(CHEMBL1834341)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354613(CHEMBL1834333)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354585(CHEMBL1834226)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354615(CHEMBL1834230)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354616(CHEMBL1834238)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309543(5-Bromo-2-methyl-1-phenyl-1H-imidazole-4-carboxyli...)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354617(CHEMBL1834340)
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317246(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methy...)
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354618(CHEMBL1834235)
Affinity DataKi:  9.30nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303837(CHEMBL570623 | [3-(4-Chlorophenyl)-4-phenyl-4,5-di...)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309536(2,5-Dimethyl-1-phenyl-1H-imidazole-4-carboxylic ac...)
Affinity DataKi:  9.70nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309539(5-Butyl-2-methyl-1-phenyl-1H-imidazole-4-carboxyli...)
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317253(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-iodo-N...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309544(2-Methyl-5-methylsulfanyl-1-phenyl-1H-imidazole-4-...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317251(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methy...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317254(CHEMBL1088507 | N-(azepan-1-yl)-1-(4-chlorophenyl)...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317248(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methy...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309541(2-Ethyl-1-phenyl-1H-imidazole-4-carboxylic acid ad...)
Affinity DataKi:  12.7nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317252(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methy...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309535(2,5-Dimethyl-1-phenyl-1H-imidazole-4-carboxylic ac...)
Affinity DataKi:  13.8nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163112(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-ethy...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163112(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-ethy...)
Affinity DataKi:  14nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303844(1-(4-Chlorophenyl)-2-(2-chlorophenyl)-5-ethyl-N-(p...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354619(CHEMBL1834227)
Affinity DataKi:  14.6nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354587(CHEMBL1834241)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354588(CHEMBL1834339)
Affinity DataKi:  17.2nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354589(CHEMBL1834228)
Affinity DataKi:  17.8nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354590(CHEMBL1834242)
Affinity DataKi:  17.9nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354591(CHEMBL1834240)
Affinity DataKi:  18.5nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303836(3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163139(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-meth...)
Affinity DataKi:  19nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309533(CHEMBL599070 | N-(((cis)-6,6-dimethylbicyclo[3.1.1...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317245(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methy...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50309546(1-Cyclohexyl-2,5-dimethyl-1H-imidazole-4-carboxyli...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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