Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-2(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-2(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Mcgill University
Curated by PDSP Ki Database
Mcgill University
Curated by PDSP Ki Database
TargetGABA A receptor alpha-4/beta-3/gamma-2(Homo sapiens (Human))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Negative allosteric modulation activity at human GABAA alpha4beta3gamma2 stably expressed in HEK cells by patch clamp methodMore data for this Ligand-Target Pair
TargetGABA A receptor alpha-1/beta-1/gamma-2(Homo sapiens (Human))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Negative allosteric modulation activity at human GABAA alpha1beta1gamma2 stably expressed in HEK cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 5.50E+3nMAssay Description:Negative allosteric modulation activity at human GABAA alpha3beta3gamma2 stably expressed in HEK cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 1.57E+4nMAssay Description:Negative allosteric modulation activity at human GABAA alpha2beta3gamma2 stably expressed in HEK cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 1.94E+4nMAssay Description:Negative allosteric modulation activity at human GABAA alpha5beta3gamma2 stably expressed in HEK cells by patch clamp methodMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Negative allosteric modulation activity at human GABAA alpha1beta3gamma2 stably expressed in HEK cells by whole cell patch clamp methodMore data for this Ligand-Target Pair