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Found 44 with Last Name = 'bourne' and Initial = 'g'
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50007916(3-{1-[1-aminobutyl oxycarbonylamino-2-(1H-3-indoly...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataIC50:  31nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50005459(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Affinity DataIC50:  50nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281743(CHEMBL169710 | [1-[2-(4-Hydroxy-phenyl)-ethylcarba...)
Affinity DataIC50:  57nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50089109(CHEMBL278780 | [2-{4-[3-(2-Chloro-phenyl)-ureido]-...)
Affinity DataIC50:  75nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281741(CHEMBL355275 | [1-(1H-Indol-3-ylmethyl)-1,2-bis-ph...)
Affinity DataIC50:  140nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281740(CHEMBL355052 | {1-(1H-Indol-3-ylmethyl)-1-phenethy...)
Affinity DataIC50:  190nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281738(CHEMBL170129 | [1-(1H-Indol-3-ylmethyl)-1-phenethy...)
Affinity DataIC50:  230nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281739(CHEMBL171375 | {1-(1H-Indol-3-ylmethyl)-2-phenethy...)
Affinity DataIC50:  330nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281743(CHEMBL169710 | [1-[2-(4-Hydroxy-phenyl)-ethylcarba...)
Affinity DataIC50:  540nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281740(CHEMBL355052 | {1-(1H-Indol-3-ylmethyl)-1-phenethy...)
Affinity DataIC50:  550nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50324491(CHEMBL1215159 | N-Benzhydryl-5-(3-hydroxyphenyl)th...)
Affinity DataIC50:  700nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281745(3-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol-3-y...)
Affinity DataIC50:  700nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM21625(2-phenyl-5-(1H-pyrazol-3-yl)-1,3-thiazole | 2-phen...)
Affinity DataIC50:  700nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
LigandPNGBDBM50281738(CHEMBL170129 | [1-(1H-Indol-3-ylmethyl)-1-phenethy...)
Affinity DataIC50:  810nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50324482(CHEMBL1215370 | N-(1-Amino-3-(1H-indol-3-yl)-1-oxo...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281739(CHEMBL171375 | {1-(1H-Indol-3-ylmethyl)-2-phenethy...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50324480(CHEMBL1215516 | N-(1-Amino-1-oxo-3-phenylpropan-2-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50324485(CHEMBL1215297 | N-(1-Amino-3-(4-hydroxyphenyl)-1-o...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50281742(CHEMBL434113 | [2-[2-(4-Hydroxy-phenyl)-ethylcarba...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM21624(4-{[4-(4-fluoro-3-methylphenyl)-1,3-thiazol-2-yl]a...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281746(CHEMBL352817 | [1-(1H-Indol-3-ylmethyl)-1-phenethy...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50324490(5-(3-Aminophenyl)-N-benzhydrylthiophene-2-carboxam...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50007916(3-{1-[1-aminobutyl oxycarbonylamino-2-(1H-3-indoly...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50324484(CHEMBL1215298 | N-(1-Amino-3-(1H-indol-3-yl)-1-oxo...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50281741(CHEMBL355275 | [1-(1H-Indol-3-ylmethyl)-1,2-bis-ph...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281744(CHEMBL171562 | [2-Benzylcarbamoyl-1-(1H-indol-3-yl...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50005459(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281742(CHEMBL434113 | [2-[2-(4-Hydroxy-phenyl)-ethylcarba...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50324486(CHEMBL1215296 | N-(1-Amino-1-oxo-3-phenylpropan-2-...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50300128(1-(3-(1H-tetrazol-5-yl)propyl)-4-(benzhydryloxy)pi...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50324483(CHEMBL1215369 | N-(1-amino-1-oxo-3-phenylpropan-2-...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50324487(CHEMBL1215295 | N-(1-Amino-4-methyl-1-oxopentan-2-...)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50324488(CHEMBL1215294 | N-(2-Amino-2-oxoethyl)-5-(3-hydrox...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50281744(CHEMBL171562 | [2-Benzylcarbamoyl-1-(1H-indol-3-yl...)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50324489(CHEMBL1215162 | N-benzhydryl-2-(3-hydroxyphenyl)th...)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50300127(CHEMBL567059 | NSC-4502 | phenyl(thiophen-2-yl)met...)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50281746(CHEMBL352817 | [1-(1H-Indol-3-ylmethyl)-1-phenethy...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50089109(CHEMBL278780 | [2-{4-[3-(2-Chloro-phenyl)-ureido]-...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50324479(5-amino-4-(3'-hydroxy-[1,1'-biphenyl]-4-ylcarboxam...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50324481(CHEMBL1215446 | N-(1-amino-1-oxo-3-phenylpropan-2-...)
Affinity DataIC50:  2.48E+4nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed