TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University
Purdue University
Affinity DataKi: 96nM IC50: 360nMpH: 5.52Assay Description:A zhang-poorman assay confirms a competitive inhibition mechanism or inhibit HIV-1 PR as a dimerization or mixed type inhibitor.More data for this Ligand-Target Pair
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University
Purdue University
Affinity DataKi: 175nM IC50: 730nMpH: 5.52Assay Description:A zhang-poorman assay confirms a competitive inhibition mechanism or inhibit HIV-1 PR as a dimerization or mixed type inhibitor.More data for this Ligand-Target Pair
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University
Purdue University
Affinity DataKi: 220nM IC50: 350nMpH: 5.52Assay Description:The competitive assay requires two inhibitors to act by a purely competitive mechanism, whereas the binding site of on the inhibitors has been establ...More data for this Ligand-Target Pair
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University
Purdue University
Affinity DataKi: 600nM IC50: 2.90E+3nMpH: 5.52Assay Description:A zhang-poorman assay confirms a competitive inhibition mechanism or inhibit HIV-1 PR as a dimerization or mixed type inhibitor.More data for this Ligand-Target Pair
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University
Purdue University
Affinity DataKi: 650nM IC50: 2.50E+3nMpH: 5.52Assay Description:A zhang-poorman assay confirms a competitive inhibition mechanism or inhibit HIV-1 PR as a dimerization or mixed type inhibitor.More data for this Ligand-Target Pair
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University
Purdue University
Affinity DataKi: 720nM IC50: 2.70E+3nMpH: 5.52Assay Description:A zhang-poorman assay confirms a competitive inhibition mechanism or inhibit HIV-1 PR as a dimerization or mixed type inhibitor.More data for this Ligand-Target Pair
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University
Purdue University
Affinity DataKi: 1.13E+3nM IC50: 4.40E+3nMpH: 5.52Assay Description:The competitive assay requires two inhibitors to act by a purely competitive mechanism, whereas the binding site of on the inhibitors has been establ...More data for this Ligand-Target Pair
Affinity DataKi: 1.25E+3nMAssay Description:Inhibition of HIV1 protease dimerization by Zhang-Poorman kinetic assayMore data for this Ligand-Target Pair
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University
Purdue University
Affinity DataKi: 1.29E+3nM IC50: 4.90E+3nMpH: 5.52Assay Description:The competitive assay requires two inhibitors to act by a purely competitive mechanism, whereas the binding site of on the inhibitors has been establ...More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Inhibition of HIV1 protease dimerization by Zhang-Poorman kinetic assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+3nMAssay Description:Inhibition of HIV1 protease dimerization by Zhang-Poorman kinetic assayMore data for this Ligand-Target Pair
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University
Purdue University
Affinity DataKi: 3.00E+3nM IC50: 5.90E+3nMpH: 5.52Assay Description:The competitive assay requires two inhibitors to act by a purely competitive mechanism, whereas the binding site of on the inhibitors has been establ...More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of HIV1 protease dimerization by Zhang-Poorman kinetic assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.80E+3nMAssay Description:Inhibition of HIV1 protease dimerization by Zhang-Poorman kinetic assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.30E+3nMAssay Description:Inhibition of HIV1 protease dimerization by Zhang-Poorman kinetic assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.69E+4nMAssay Description:Inhibition of HIV1 protease by competitive inhibition assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.01E+4nMAssay Description:Inhibition of HIV1 protease dimerization by Zhang-Poorman kinetic assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.80E+4nMAssay Description:Inhibition of HIV1 protease dimerization by Zhang-Poorman kinetic assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.10E+5nMAssay Description:Inhibition of HIV1 protease dimerization by Zhang-Poorman kinetic assayMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 0.140nMAssay Description:Inhibitory activity against Gamma-secretase in HeLa cells expressing APP-reporterMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against Gamma-secretase from APP-transfected CHO cellsMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against Gamma-secretase in HeLa cells expressing APP-reporterMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against Gamma-secretase in HeLa cells expressing APP-reporterMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibitory activity against Gamma-secretase in HeLa cells expressing APP-reporterMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against Gamma-secretase in HeLa cells expressing APP-reporterMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibitory activity against Gamma-secretase in HeLa cells expressing APP-reporterMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against Gamma-secretase in HeLa cells expressing APP-reporterMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibitory activity against Gamma-secretase in HeLa cells expressing APP-reporterMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibitory activity against Gamma-secretase in HeLa cells expressing APP-reporterMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 780nMAssay Description:Inhibitory activity against Gamma-secretase in HeLa cells expressing APP-reporterMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 910nMAssay Description:Inhibitory activity against Gamma-secretase in HeLa cells expressing APP-reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of HIV1 protease by continuous fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of HIV1 protease by continuous fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of HIV1 protease by continuous fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of HIV1 protease by continuous fluorometric assayMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibitory activity against Gamma-secretase in HeLa cells expressing APP-reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of HIV1 protease by continuous fluorometric assayMore data for this Ligand-Target Pair
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University
Purdue University
Affinity DataIC50: 4.30E+3nMpH: 5.52Assay Description:A zhang-poorman assay confirms a competitive inhibition mechanism or inhibit HIV-1 PR as a dimerization or mixed type inhibitor.More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibitory concentration against ProteaseMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibitory activity against Gamma-secretase in HeLa cells expressing APP-reporterMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibitory concentration against ProteaseMore data for this Ligand-Target Pair
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University
Purdue University
Affinity DataIC50: 5.80E+3nMpH: 5.52Assay Description:The competitive assay requires two inhibitors to act by a purely competitive mechanism, whereas the binding site of on the inhibitors has been establ...More data for this Ligand-Target Pair
TargetCapsid scaffolding protein(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
Purdue University
Purdue University
Affinity DataIC50: 5.80E+3nMpH: 5.52Assay Description:A zhang-poorman assay confirms a competitive inhibition mechanism or inhibit HIV-1 PR as a dimerization or mixed type inhibitor.More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibitory concentration against ProteaseMore data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of HIV1 protease by continuous fluorometric assayMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory concentration against ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibitory concentration against ProteaseMore data for this Ligand-Target Pair
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of HIV1 protease by continuous fluorometric assayMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibitory concentration against ProteaseMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against Gamma-secretase in HeLa cells expressing APP-reporterMore data for this Ligand-Target Pair