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Found 10 with Last Name = 'bowyer' and Initial = 'sl'
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50237727(CHEMBL4060938)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249034(CHEMBL4077729)
Affinity DataIC50:  2.42E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249036(CHEMBL4066742)
Affinity DataIC50:  3.38E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249039(CHEMBL4101998)
Affinity DataIC50:  4.24E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249038(CHEMBL1409841)
Affinity DataIC50:  4.54E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249041(CHEMBL4081253)
Affinity DataIC50:  4.96E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249040(CHEMBL4080320)
Affinity DataIC50:  5.95E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249037(CHEMBL4104553)
Affinity DataIC50:  6.41E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249035(CHEMBL4094266)
Affinity DataIC50:  6.75E+3nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50249033(CHEMBL4078657)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed