Compile Data Set for Download or QSAR
maximum 50k data
Found 32 with Last Name = 'boyd' and Initial = 'mr'
TargetProtein kinase C zeta type(Rattus norvegicus)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478518(CHEMBL514017)
Affinity DataIC50:  17nMAssay Description:Displacement of [3H]PDBu from rat brain membrane PKCMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50090045((2,3-Dihydroxy-4-methoxy-phenyl)-(3,4,5-trimethoxy...)
Affinity DataIC50:  820nMAssay Description:Inhibition of tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of tubulin polymerizationMore data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50090044((Z)-2',3'-dihydroxy-3,4,4',5-tetramethoxystilbene ...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  1.20E+3nMAssay Description:The compound was tested for the concentration to inhibit 50% of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50006677(1,2,3-Trimethoxy-5-[(Z)-2-(4-methoxy-phenyl)-vinyl...)
Affinity DataIC50:  1.30E+3nMAssay Description:The compound was tested for the concentration to inhibit 50% of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataIC50:  1.90E+3nMAssay Description:Tested for 50 % inhibition of tubulin polymerization by turbidimetric assayMore data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50064891(5,7,3'-trihydroxy-3,6-4'-trimethoxyflavone | 5,7-D...)
Affinity DataIC50:  3.00E+3nMAssay Description:Tested for 50 % inhibition of tubulin polymerization by turbidimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478521(CHEMBL465805)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50471653(CHEMBL297299)
Affinity DataIC50:  3.50E+3nMAssay Description:The compound was tested for the concentration to inhibit 50% of tubulin polymerization.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50292441(1beta-hydroxyaleuritolic acid 3-p-hydroxybenzoate ...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478525(CHEMBL465804)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478526(CHEMBL448121)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478416(CHEBI:65536 | CHEMBL444821)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478527(Aleuritolic Acid 3-P-Hydroxybenzoate | CHEMBL45689...)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478523(Aleuritolic Acid 3-P-Hydroxycinnamate | CHEMBL5033...)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478415(Buchapine | CHEBI:65535)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478524(CHEMBL450856)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478522(CHEMBL454238)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50471654(CHEMBL44574)
Affinity DataIC50:  2.10E+4nMAssay Description:The compound was tested for the concentration to inhibit 50% of tubulin polymerization.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478522(CHEMBL454238)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by NCI assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50090046(CHEMBL329267 | Phosphoric acid mono-[3-methoxy-2-p...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50064259(CHEMBL289351 | Combretastatin A4 phosphate | Di-So...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478528(CHEMBL451536)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478526(CHEMBL448121)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by NCI assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478523(Aleuritolic Acid 3-P-Hydroxycinnamate | CHEMBL5033...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by NCI assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50064259(CHEMBL289351 | Combretastatin A4 phosphate | Di-So...)
Affinity DataIC50: >8.00E+4nMAssay Description:The compound was tested for the concentration to inhibit 50% of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478521(CHEMBL465805)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by NCI assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50292441(1beta-hydroxyaleuritolic acid 3-p-hydroxybenzoate ...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by NCI assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478528(CHEMBL451536)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by NCI assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478524(CHEMBL450856)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by NCI assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478527(Aleuritolic Acid 3-P-Hydroxybenzoate | CHEMBL45689...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by NCI assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed