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Found 136 with Last Name = 'brömme' and Initial = 'd'
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409589(CHEMBL2028920)
Affinity DataKi:  0.100nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409598(CHEMBL2028910)
Affinity DataKi:  0.120nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409597(CHEMBL2028912)
Affinity DataKi:  0.280nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409590(CHEMBL2028909)
Affinity DataKi:  0.560nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409583(CHEMBL2028921)
Affinity DataKi:  0.580nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409586(CHEMBL2028907)
Affinity DataKi:  0.770nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409592(CHEMBL2028908)
Affinity DataKi:  0.780nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409587(CHEMBL2028911)
Affinity DataKi:  0.950nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409588(CHEMBL2028919)
Affinity DataKi:  1.35nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032805(CHEMBL107495 | N-[2-(3-Morpholin-4-yl-ureido)-1-na...)
Affinity DataKi:  1.80nMAssay Description:Compound is evaluated for inhibitory potency against cathepsin SMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032803(2-((E)-2-Benzenesulfonyl-vinylamino)-N-[3-methyl-1...)
Affinity DataKi:  5.90nMAssay Description:Compound is evaluated for inhibitory potency against cathepsin SMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50118425(CHEMBL263061 | Z-leu-Val-Agly-Val-OBzl)
Affinity DataKi:  6.70nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032802(2-((E)-2-Benzenesulfonyl-vinylamino)-N-[1-benzyl-2...)
Affinity DataKi:  11nMAssay Description:Compound is evaluated for inhibitory potency against cathepsin SMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409584(CHEMBL2028906)
Affinity DataKi:  17nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032805(CHEMBL107495 | N-[2-(3-Morpholin-4-yl-ureido)-1-na...)
Affinity DataKi:  18nMAssay Description:Compound is evaluated for inhibitory potency against cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409599(CHEMBL2028925)
Affinity DataKi:  20nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409594(CHEMBL2028924)
Affinity DataKi:  21nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50118412(Boc-Agly-Val-Agly-OEt | CHEMBL135413)
Affinity DataKi:  24nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409596(CHEMBL2028923)
Affinity DataKi:  28nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409591(CHEMBL2028922)
Affinity DataKi:  30nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409582(CHEMBL2028926)
Affinity DataKi:  32nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50118425(CHEMBL263061 | Z-leu-Val-Agly-Val-OBzl)
Affinity DataKi:  34nMAssay Description:Inhibition of Human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50118425(CHEMBL263061 | Z-leu-Val-Agly-Val-OBzl)
Affinity DataKi:  40nMAssay Description:Inhibition of Human Cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032805(CHEMBL107495 | N-[2-(3-Morpholin-4-yl-ureido)-1-na...)
Affinity DataKi:  48nMAssay Description:Compound is evaluated for inhibitory potency against CruzaineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409585(CHEMBL2028918)
Affinity DataKi:  59nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50118412(Boc-Agly-Val-Agly-OEt | CHEMBL135413)
Affinity DataKi:  61nMAssay Description:Inhibition of Human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409595(CHEMBL2028917)
Affinity DataKi:  61nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409593(CHEMBL2028913)
Affinity DataKi:  100nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50032805(CHEMBL107495 | N-[2-(3-Morpholin-4-yl-ureido)-1-na...)
Affinity DataKi:  150nMAssay Description:Compound is evaluated for inhibitory potency against cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50385972(CHEMBL2042470)
Affinity DataKi:  200nMAssay Description:Competitive inhibition of human recombinant cathepsin L expressed in Pichia pastoris using Z-Phe-Arg-MCA as substrate by Lineweaver-Burk plot analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin L2(Homo sapiens (Human))
Universidade Federal De S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50336482(CHEMBL1668599 | citibrasine)
Affinity DataKi:  200nMAssay Description:Inhibition of human recombinant cathepsin V expressed in Pichia pastoris by Lineweaver-Burk double-reciprocal plotsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032803(2-((E)-2-Benzenesulfonyl-vinylamino)-N-[3-methyl-1...)
Affinity DataKi:  220nMAssay Description:Compound is evaluated for inhibitory potency against CruzaineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50032803(2-((E)-2-Benzenesulfonyl-vinylamino)-N-[3-methyl-1...)
Affinity DataKi:  230nMAssay Description:Compound is evaluated for inhibitory potency against cathepsin O2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50032804(2-((E)-2-Benzenesulfonyl-vinylamino)-N-[1-(4-hydro...)
Affinity DataKi:  340nMAssay Description:Compound is evaluated for inhibition kinetic constant Ki for the cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032802(2-((E)-2-Benzenesulfonyl-vinylamino)-N-[1-benzyl-2...)
Affinity DataKi:  360nMAssay Description:Compound is evaluated for inhibitory potency against CruzaineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin L2(Homo sapiens (Human))
Universidade Federal De S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50385972(CHEMBL2042470)
Affinity DataKi:  400nMAssay Description:Competitive inhibition of human recombinant cathepsin V expressed in Pichia pastoris using Z-Phe-Arg-MCA as substrate by Lineweaver-Burk plot analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin L2(Homo sapiens (Human))
Universidade Federal De S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50336477(1,3,5-trihydroxy-4-methoxy-10-methyl-2,8-bis(3-met...)
Affinity DataKi:  500nMAssay Description:Inhibition of human recombinant cathepsin V expressed in Pichia pastoris by Lineweaver-Burk double-reciprocal plotsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032803(2-((E)-2-Benzenesulfonyl-vinylamino)-N-[3-methyl-1...)
Affinity DataKi:  720nMAssay Description:Compound is evaluated for inhibitory potency against cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin L2(Homo sapiens (Human))
Universidade Federal De S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50385984(CHEMBL2042454)
Affinity DataKi:  800nMAssay Description:Uncompetitive inhibition of human recombinant cathepsin V expressed in Pichia pastoris using Z-Phe-Arg-MCA as substrate by Lineweaver-Burk plot analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin L2(Homo sapiens (Human))
Universidade Federal De S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50385977(CHEMBL2042446)
Affinity DataKi:  800nMAssay Description:Noncompetitive inhibition of human recombinant cathepsin V expressed in Pichia pastoris using Z-Phe-Arg-MCA as substrate by Lineweaver-Burk plot anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50385966(CHEMBL2042465)
Affinity DataKi:  900nMAssay Description:Competitive inhibition of human recombinant cathepsin L expressed in Pichia pastoris using Z-Phe-Arg-MCA as substrate by Lineweaver-Burk plot analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032802(2-((E)-2-Benzenesulfonyl-vinylamino)-N-[1-benzyl-2...)
Affinity DataKi:  1.00E+3nMAssay Description:Compound is evaluated for inhibitory potency against cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin L2(Homo sapiens (Human))
Universidade Federal De S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50336481(CHEMBL451705 | citrusinine I | citrusinine-I)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human recombinant cathepsin V expressed in Pichia pastoris by Lineweaver-Burk double-reciprocal plotsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin L2(Homo sapiens (Human))
Universidade Federal De S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50336478(1,3,5-trihydroxy-4-methoxy-2-(3-methylbut-2-enyl)-...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human recombinant cathepsin V expressed in Pichia pastoris by Lineweaver-Burk double-reciprocal plotsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin L2(Homo sapiens (Human))
Universidade Federal De S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50385962(CHEMBL2042461)
Affinity DataKi:  1.10E+3nMAssay Description:Uncompetitive inhibition of human recombinant cathepsin V expressed in Pichia pastoris using Z-Phe-Arg-MCA as substrate by Lineweaver-Burk plot analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin L2(Homo sapiens (Human))
Universidade Federal De S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50336476(1,3,5-trihydroxy-2,8-bis(3-methylbut-2-enyl)-10-me...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of human recombinant cathepsin V expressed in Pichia pastoris by Lineweaver-Burk double-reciprocal plotsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin L2(Homo sapiens (Human))
Universidade Federal De S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50385966(CHEMBL2042465)
Affinity DataKi:  1.30E+3nMAssay Description:Competitive inhibition of human recombinant cathepsin V expressed in Pichia pastoris using Z-Phe-Arg-MCA as substrate by Lineweaver-Burk plot analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50385977(CHEMBL2042446)
Affinity DataKi:  1.50E+3nMAssay Description:Noncompetitive inhibition of human recombinant cathepsin L expressed in Pichia pastoris using Z-Phe-Arg-MCA as substrate by Lineweaver-Burk plot anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin L2(Homo sapiens (Human))
Universidade Federal De S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50336486(3,4-dihydro-3,5,8-trihydroxy-6-methoxy-2,2,7-trime...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of human recombinant cathepsin V expressed in Pichia pastoris by Lineweaver-Burk double-reciprocal plotsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50385962(CHEMBL2042461)
Affinity DataKi:  1.90E+3nMAssay Description:Uncompetitive inhibition of human recombinant cathepsin L expressed in Pichia pastoris using Z-Phe-Arg-MCA as substrate by Lineweaver-Burk plot analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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