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Found 210 with Last Name = 'brambilla' and Initial = 'e'
TargetPteridine reductase 1(Leishmania major)
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50551183(CHEMBL4747846)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibition of Leishmania major PTR1 using H2B as substrate preincubated for 10 mins followed by NADPH addition and measured up to 50 mins relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50551184(CHEMBL4797185)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibition of Leishmania major PTR1 using H2B as substrate preincubated for 10 mins followed by NADPH addition and measured up to 50 mins relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50551180(CHEMBL4760251)
Affinity DataKi:  1.48E+4nMAssay Description:Inhibition of Leishmania major PTR1 using H2B as substrate preincubated for 10 mins followed by NADPH addition and measured up to 50 mins relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50551177(CHEMBL4762279)
Affinity DataKi:  1.53E+4nMAssay Description:Inhibition of Leishmania major PTR1 using H2B as substrate preincubated for 10 mins followed by NADPH addition and measured up to 50 mins relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50551178(CHEMBL4785591)
Affinity DataKi:  1.92E+4nMAssay Description:Inhibition of Leishmania major PTR1 using H2B as substrate preincubated for 10 mins followed by NADPH addition and measured up to 50 mins relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50551181(CHEMBL54725)
Affinity DataKi:  3.72E+4nMAssay Description:Inhibition of Leishmania major PTR1 using H2B as substrate preincubated for 10 mins followed by NADPH addition and measured up to 50 mins relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50551174(CHEMBL158919)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of Leishmania major PTR1 using H2B as substrate preincubated for 10 mins followed by NADPH addition and measured up to 50 mins relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50551179(CHEMBL4778279)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of Leishmania major PTR1 using H2B as substrate preincubated for 10 mins followed by NADPH addition and measured up to 50 mins relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50551173(CHEMBL4753331)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of Leishmania major PTR1 using H2B as substrate preincubated for 10 mins followed by NADPH addition and measured up to 50 mins relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50551176(CHEMBL4748094)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of Leishmania major PTR1 using H2B as substrate preincubated for 10 mins followed by NADPH addition and measured up to 50 mins relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50551182(CHEMBL4754292)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of Leishmania major PTR1 using H2B as substrate preincubated for 10 mins followed by NADPH addition and measured up to 50 mins relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50062821(6-Benzyloxy-pyrimidine-2,4-diamine | CHEMBL121445)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of Leishmania major PTR1 using H2B as substrate preincubated for 10 mins followed by NADPH addition and measured up to 50 mins relative to...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50386758(CHEMBL2046893)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of Leishmania major PTR1 using H2B as substrate preincubated for 10 mins followed by NADPH addition and measured up to 50 mins relative to...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
University Of Modena And Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50551175(CHEMBL1993081)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of Leishmania major PTR1 using H2B as substrate preincubated for 10 mins followed by NADPH addition and measured up to 50 mins relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50289537(1-(3-Phenyl-propyl)-3-((Z)-styryl)-piperidine | CH...)
Affinity DataIC50:  0.600nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289553(1-Phenethyl-3-((Z)-styryl)-piperidine | CHEMBL3697...)
Affinity DataIC50:  0.800nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289552(1-(3-Methyl-but-2-enyl)-3-((Z)-styryl)-piperidine ...)
Affinity DataIC50:  1nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(RAT)
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070198((6aR,9R,10aR)-3-tert-Butyl-7-methyl-4,6,6a,7,8,9,1...)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor in rat pre frontal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289539(1-Cyclohexyl-3-((Z)-styryl)-piperidine | CHEMBL398...)
Affinity DataIC50:  2nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(RAT)
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070192((6aR,9R,10aR)-3-tert-Butyl-7-methyl-4,6,6a,7,8,9,1...)
Affinity DataIC50:  3nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor in rat pre frontal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070187(1-Acetyl-3-((6aR,9S,10aR)-3-tert-butyl-7-methyl-4,...)
Affinity DataIC50:  3nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor in rat pre frontal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289541(1-(3-Phenyl-propyl)-3-((E)-styryl)-piperidine | CH...)
Affinity DataIC50:  4nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289538(1-Allyl-3-((E)-styryl)-piperidine | CHEMBL39735)
Affinity DataIC50:  4nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289547(1-Phenethyl-3-((E)-styryl)-piperidine | CHEMBL2879...)
Affinity DataIC50:  6nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289549(1-Cyclohexyl-3-((E)-styryl)-piperidine | CHEMBL291...)
Affinity DataIC50:  6nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50070193(1-((6aR,9R,10aR)-2-tert-Butyl-7-methyl-4,6,6a,7,8,...)
Affinity DataIC50:  7nMAssay Description:Displacement of [3H]yohimbine from Alpha-2 adrenergic receptor in rat frontal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289551(1-(4-Phenyl-butyl)-3-((Z)-styryl)-piperidine | CHE...)
Affinity DataIC50:  7nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289545(1-(2-Cyclohexyl-ethyl)-3-((Z)-styryl)-piperidine |...)
Affinity DataIC50:  7nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289536(1-Benzyl-3-((E)-styryl)-piperidine | CHEMBL39855)
Affinity DataIC50:  10nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289554(1-Pent-4-enyl-3-((E)-styryl)-piperidine | CHEMBL38...)
Affinity DataIC50:  12nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070203(CHEMBL14048 | N-((6aR,9S,10aR)-7-Methyl-4,6,6a,7,8...)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289544(1-Phenyl-4-[3-((Z)-styryl)-piperidin-1-yl]-butan-1...)
Affinity DataIC50:  15nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070201(((6aR,9S,10aR)-2-tert-Butyl-7-methyl-4,6,6a,7,8,9,...)
Affinity DataIC50:  15nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289540(1-(3-Phenoxy-propyl)-3-((Z)-styryl)-piperidine | C...)
Affinity DataIC50:  15nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(RAT)
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070191(1-((6aR,9R,10aR)-3-tert-Butyl-7-methyl-4,6,6a,7,8,...)
Affinity DataIC50:  19nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor in rat pre frontal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289556(1,1-Dioxo-2-{4-[3-((E)-styryl)-piperidin-1-yl]-but...)
Affinity DataIC50:  23nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289557(Adamantane-1-carboxylic acid {4-[3-((Z)-styryl)-pi...)
Affinity DataIC50:  23nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070185(CHEMBL273526 | N-((6aR,9S,10aR)-2-tert-Butyl-7-met...)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289543(2-{3-[3-((Z)-Styryl)-piperidin-1-yl]-propylsulfany...)
Affinity DataIC50:  27nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070190(((6aR,9S,10aR)-3-tert-Butyl-7-methyl-4,6,6a,7,8,9,...)
Affinity DataIC50:  27nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070202(CHEMBL267799 | N-((6aR,9S,10aR)-3-tert-Butyl-7-met...)
Affinity DataIC50:  31nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070188(1-((6aR,9R,10aR)-3-tert-Butyl-7-methyl-4,6,6a,7,8,...)
Affinity DataIC50:  32nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor in rat pre frontal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289550(1-(3-Phenoxy-propyl)-3-((E)-styryl)-piperidine | C...)
Affinity DataIC50:  33nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289546(1-(3-Methyl-but-2-enyl)-3-((E)-styryl)-piperidine ...)
Affinity DataIC50:  38nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(RAT)
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070202(CHEMBL267799 | N-((6aR,9S,10aR)-3-tert-Butyl-7-met...)
Affinity DataIC50:  48nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor in rat pre frontal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070181(1-(3-Dimethylamino-propyl)-3-ethyl-1-((6aR,9R,10aR...)
Affinity DataIC50:  50nMAssay Description:Displacement of [3H]-spiroperidol from D2 receptor in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070190(((6aR,9S,10aR)-3-tert-Butyl-7-methyl-4,6,6a,7,8,9,...)
Affinity DataIC50:  54nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor in rat pre frontal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070184(((6aR,9S,10aR)-7-Methyl-4,6,6a,7,8,9,10,10a-octahy...)
Affinity DataIC50:  60nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289542(3-((Z)-Styryl)-piperidine | CHEMBL38345)
Affinity DataIC50:  64nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070203(CHEMBL14048 | N-((6aR,9S,10aR)-7-Methyl-4,6,6a,7,8...)
Affinity DataIC50:  75nMAssay Description:Displacement of [3H]-spiroperidol from D2 receptor in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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