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Found 58 with Last Name = 'breen' and Initial = 'a'
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073419(2-Biphenyl-4-yl-1,1-dioxo-1H-1lambda*6*-thiochrome...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073422(2-(4-Nitro-phenyl)-1,1-dioxo-1H-1lambda*6*-thiochr...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073414(5-Methyl-2-(4-nitro-phenyl)-1,1-dioxo-1H-1lambda*6...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073418(1,1-Dioxo-2-pyridin-4-yl-1H-1lambda*6*-thiochromen...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073411(2-(4-Methanesulfonyl-phenyl)-1,1-dioxo-1H-1lambda*...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073415(8-Methyl-2-(4-nitro-phenyl)-1,1-dioxo-1H-1lambda*6...)
Affinity DataIC50:  110nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50029987(12-Hydroxy-6,6,10,11-tetramethyl-4-phenyl-11,12-di...)
Affinity DataIC50:  130nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50029982(12-Hydroxy-6,6,10,11-tetramethyl-4-phenyl-11,12-di...)
Affinity DataIC50:  160nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase mutant (Tyr-181 to Cys)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50029982(12-Hydroxy-6,6,10,11-tetramethyl-4-phenyl-11,12-di...)
Affinity DataIC50:  160nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase mutant (Tyr-181 to Cys)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073408(8-Isopropyl-2-(4-nitro-phenyl)-1,1-dioxo-1H-1lambd...)
Affinity DataIC50:  180nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073413(2-(4-Nitro-phenyl)-1,1,4-trioxo-1,4-dihydro-1lambd...)
Affinity DataIC50:  180nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073421(1,1-Dioxo-2-pyridin-3-yl-1H-1lambda*6*-thiochromen...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50029982(12-Hydroxy-6,6,10,11-tetramethyl-4-phenyl-11,12-di...)
Affinity DataIC50:  410nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase mutant (Tyr-181 to Leu)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073420(1,1-Dioxo-2-thiophen-2-yl-1H-1lambda*6*-thiochrome...)
Affinity DataIC50:  460nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073424(1,1-Dioxo-2-(1-oxy-pyridin-4-yl)-1H-1lambda*6*-thi...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073423(1,1-Dioxo-2-(1-oxy-pyridin-3-yl)-1H-1lambda*6*-thi...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50279762((5S)-9-chloro-5-methyl-6-(3-methylbut-2-enyl)-4,5,...)
Affinity DataIC50:  700nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50029996(Acetic acid 2,3,10,10-tetramethyl-6-oxo-8-phenyl-3...)
Affinity DataIC50:  720nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073407(2-Heptyl-1,1-dioxo-1H-1lambda*6*-thiochromen-4-one...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073412(1,1-Dioxo-2-phenyl-1H-1lambda*6*-thiochromen-4-one...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290547((R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-[6-meth...)
Affinity DataIC50:  5.20E+3nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290549((R)-[2-(4-Chloro-phenyl)-6-methoxy-quinolin-4-yl]-...)
Affinity DataIC50:  5.50E+3nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290549((R)-[2-(4-Chloro-phenyl)-6-methoxy-quinolin-4-yl]-...)
Affinity DataIC50:  5.90E+3nMAssay Description:Compound was tested in vitro for its binding affinity towards recombinant human Calcitonin gene-related peptide type receptor (membranes of HEK-293 c...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50029985(6,6,10,11-Tetramethyl-4-phenyl-6H,10H-dipyrano[2,3...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290551((R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-[6-meth...)
Affinity DataIC50:  9.90E+3nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50029988(6,6,10,11-Tetramethyl-4-phenyl-10,11-dihydro-6H-di...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073416(1-Oxo-2-phenyl-1H-1lambda*4*-thiochromen-4-one | 4...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50029992(12-Hydroxy-6,6,10,11-tetramethyl-4-phenyl-11,12-di...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290558((R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-[6-meth...)
Affinity DataIC50:  1.20E+4nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290553((R)-[2-(3-Chloro-4-fluoro-phenyl)-6-methoxy-quinol...)
Affinity DataIC50:  1.70E+4nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
TBA

Curated by ChEMBL
LigandPNGBDBM50281340(5-{[(2-Chloro-ethyl)-ethyl-amino]-methyl}-3,3-diph...)
Affinity DataIC50:  3.00E+4nMAssay Description:Tested for ability to block the CD4-gp120 interaction measured by binding of [125I]-sCD4 to gp120More data for this Ligand-Target Pair
In DepthDetails Article
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
TBA

Curated by ChEMBL
LigandPNGBDBM50281340(5-{[(2-Chloro-ethyl)-ethyl-amino]-methyl}-3,3-diph...)
Affinity DataIC50:  3.00E+4nMAssay Description:Tested in an HIV viral syncytium assay for inhibition of binding of recombinant CD4-gp120More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50029981(12-Hydroxy-6,6,10,11-tetramethyl-4-phenyl-11,12-di...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290548((R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-(6-meth...)
Affinity DataIC50:  3.30E+4nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073409(2-Phenyl-thiochromen-4-one | CHEMBL58311)
Affinity DataIC50: >3.40E+4nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073410(2-tert-Butyl-1,1-dioxo-1H-1lambda*6*-thiochromen-4...)
Affinity DataIC50: >3.40E+4nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073417(1,1-Dioxo-2-thiophen-3-yl-1H-1lambda*6*-thiochrome...)
Affinity DataIC50: >3.40E+4nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073406(2-Pyridin-3-yl-thiochromen-4-one | CHEMBL123060)
Affinity DataIC50: >3.40E+4nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCapsid scaffolding protein(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50073405(2-(4-Methanesulfonyl-phenyl)-thiochromen-4-one | C...)
Affinity DataIC50: >3.40E+4nMAssay Description:Inhibitory activity of the compound against human cytomegalovirus (HCMV) protease was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290556((R)-[2-(2,4-Dichloro-phenyl)-6-methoxy-quinolin-4-...)
Affinity DataIC50:  3.70E+4nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290552((R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-[6-meth...)
Affinity DataIC50:  4.10E+4nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50029986(12-(4-Bromo-benzoyl)-6,6,10,11-tetramethyl-4-pheny...)
Affinity DataIC50:  4.60E+4nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50029994(4-hydroxy-2,3,10,10-tetramethyl-8-phenyl-(2R,3S,4S...)
Affinity DataIC50:  7.00E+4nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290550((R)-(2-Benzo[1,3]dioxol-5-yl-6-methoxy-quinolin-4-...)
Affinity DataIC50:  7.40E+4nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290546((R)-(5-Ethyl-1-aza-bicyclo[2.2.2]oct-2-yl)-(6-meth...)
Affinity DataIC50:  9.60E+4nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50029995(6,6,10,11-Tetramethyl-4-phenyl-10,11-dihydro-6H-di...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
TBA

Curated by ChEMBL
LigandPNGBDBM50281339((S)-2-{(S)-2-[(4S,9S)-9-((R)-1-Amino-2-hydroxy-eth...)
Affinity DataIC50: >1.00E+5nMAssay Description:Tested for inhibition of binding of soluble recombinant CD4-gp120 using ELISA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50029993(3-(5-Hydroxy-2,3,8,8-tetramethyl-4-oxo-3,4-dihydro...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50029983(3-[7-Hydroxy-5-methoxy-2,2-dimethyl-6-(2-methyl-bu...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290554((R)-[2-(3-Amino-phenyl)-6-methoxy-quinolin-4-yl]-(...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [125I]-hCGRP human Calcitonin gene-related peptide type receptor expressed in SK-N-MC neuroblastoma cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
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