TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase mutant (Tyr-181 to Cys)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase mutant (Tyr-181 to Cys)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase mutant (Tyr-181 to Leu)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Tested in an HIV viral syncytium assay for inhibition of binding of recombinant CD4-gp120More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Tested for ability to block the CD4-gp120 interaction measured by binding of [125I]-sCD4 to gp120More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Tested for inhibition of binding of soluble recombinant CD4-gp120 using ELISA assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for rate constant of binding to inhibit soluble recombinant CD4-gp120 ; value ranges form 4-20 uMMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Tested for inhibition of binding of soluble recombinant CD4-gp120 using ELISA assayMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKd: 4.00E+3nMAssay Description:Tested for inhibition of binding of soluble recombinant CD4-gp120 using ELISA assayMore data for this Ligand-Target Pair