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Found 28 with Last Name = 'breliere' and Initial = 'jc'
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
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Curated by PDSP Ki Database
LigandPNGBDBM81780(CAS_6438382 | NSC_6438382 | SR 46349B)
Affinity DataKi:  5.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM21395(3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H...)
Affinity DataKi:  14.5nMMore data for this Ligand-Target Pair
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Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001775((ritanserin)6-(2-{4-[Bis-(4-fluoro-phenyl)-methyle...)
Affinity DataKi:  58.1nMMore data for this Ligand-Target Pair
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Target5-hydroxytryptamine receptor 2C(PIG)
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Curated by PDSP Ki Database
LigandPNGBDBM81780(CAS_6438382 | NSC_6438382 | SR 46349B)
Affinity DataKi:  120nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(RAT)
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Curated by PDSP Ki Database
LigandPNGBDBM81780(CAS_6438382 | NSC_6438382 | SR 46349B)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
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Curated by PDSP Ki Database
LigandPNGBDBM81780(CAS_6438382 | NSC_6438382 | SR 46349B)
Affinity DataKi:  3.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H1 receptor(RAT)
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Curated by PDSP Ki Database
LigandPNGBDBM81780(CAS_6438382 | NSC_6438382 | SR 46349B)
Affinity DataKi:  5.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(1A) dopamine receptor(RAT)
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Curated by PDSP Ki Database
LigandPNGBDBM81780(CAS_6438382 | NSC_6438382 | SR 46349B)
Affinity DataKi:  9.00E+3nMMore data for this Ligand-Target Pair
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Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81780(CAS_6438382 | NSC_6438382 | SR 46349B)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium channel protein type 10 subunit alpha(Rattus norvegicus (Rat))
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81780(CAS_6438382 | NSC_6438382 | SR 46349B)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81780(CAS_6438382 | NSC_6438382 | SR 46349B)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine 1D receptor(Bos taurus (Bovine))
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81780(CAS_6438382 | NSC_6438382 | SR 46349B)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50282270(4'-(2-Butyl-4-cyclopentyl-4-methyl-5-oxo-4,5-dihyd...)
Affinity DataIC50:  3.30nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282264(2-Butyl-5-cyclohexyl-5-methyl-3-[2'-(1H-tetrazol-5...)
Affinity DataIC50:  5.20nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282264(2-Butyl-5-cyclohexyl-5-methyl-3-[2'-(1H-tetrazol-5...)
Affinity DataIC50:  5.20nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282267(4'-(2-Butyl-4-isopropyl-4-methyl-5-oxo-4,5-dihydro...)
Affinity DataIC50:  7.30nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282263(2-Butyl-5-cyclopentyl-5-methyl-3-[2'-(2H-tetrazol-...)
Affinity DataIC50:  7.60nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282262(4'-(2-Butyl-4-cyclohexyl-4-methyl-5-oxo-4,5-dihydr...)
Affinity DataIC50:  12nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282268(4'-(2-Butyl-4-cyclopropyl-4-methyl-5-oxo-4,5-dihyd...)
Affinity DataIC50:  18nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282265(4'-(2-Butyl-4-methyl-5-oxo-4-phenyl-4,5-dihydro-im...)
Affinity DataIC50:  19nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50042244(4'-(2-Butyl-4,4-dimethyl-5-oxo-4,5-dihydro-imidazo...)
Affinity DataIC50:  35nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282269(4'-(2-Butyl-4-cyclohexyl-4-ethyl-5-oxo-4,5-dihydro...)
Affinity DataIC50:  52nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50042240(4'-(2-Butyl-4,4-diethyl-5-oxo-4,5-dihydro-imidazol...)
Affinity DataIC50:  56nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50042239(4'-(2-Butyl-4,4-dicyclopropyl-5-oxo-4,5-dihydro-im...)
Affinity DataIC50:  80nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282266(4'-(2-Butyl-4-cyclohexylmethyl-4-methyl-5-oxo-4,5-...)
Affinity DataIC50:  150nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282271(4'-[2-Butyl-4-(2,4-dimethyl-pentyl)-4-methyl-5-oxo...)
Affinity DataIC50:  230nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50042222(4'-(2,4,4-Tributyl-5-oxo-4,5-dihydro-imidazol-1-yl...)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50042241(4'-(2-Butyl-4,4-diisobutyl-5-oxo-4,5-dihydro-imida...)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article