Affinity DataKi: 9.80nMAssay Description:Inhibition of human CYP2D6 by Lineweaver-Burk plotMore data for this Ligand-Target Pair
Affinity DataKi: 28.1nMAssay Description:Inhibition of human CYP2D6 by Lineweaver-Burk plotMore data for this Ligand-Target Pair
Affinity DataKi: 54.7nMAssay Description:Inhibition of human CYP2D6 by Lineweaver-Burk plotMore data for this Ligand-Target Pair
Affinity DataKi: 450nMAssay Description:Inhibition of human CYP2D6 by Lineweaver-Burk plotMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of human butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human CYP2D6 expressed in baculovirus-infected insect cell systemMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of human acetylcholinesterase using acetylcholine iodide as substrate preincubated for 30 mins followed by substrate addition measured aft...More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Binding affinity of the compound was determined against Nicotinic acetylcholine receptor using [3H]-(-)-nicotine radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 56.1nMAssay Description:Inhibition of human CYP2D6 expressed in baculovirus-infected insect cell systemMore data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 83nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 96nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 106nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 109nMAssay Description:Inhibition of human CYP2D6 expressed in baculovirus-infected insect cell systemMore data for this Ligand-Target Pair
Affinity DataIC50: 115nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 199nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 208nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 231nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 238nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 374nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 474nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 531nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 565nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 723nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 852nMAssay Description:Inhibition of human acetylcholinesterase using acetylcholine iodide as substrate preincubated for 30 mins followed by substrate addition measured aft...More data for this Ligand-Target Pair
Affinity DataIC50: 875nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of human CYP2D6 expressed in baculovirus-infected insect cell systemMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Albert-Ludwigs-University Of Freiburg
Curated by ChEMBL
Albert-Ludwigs-University Of Freiburg
Curated by ChEMBL
Affinity DataIC50: 1.47E+3nMAssay Description:Inhibition of p38alpha after 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of human acetylcholinesterase using acetylcholine iodide as substrate preincubated for 30 mins followed by substrate addition measured aft...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Albert-Ludwigs-University Of Freiburg
Curated by ChEMBL
Albert-Ludwigs-University Of Freiburg
Curated by ChEMBL
Affinity DataIC50: 2.21E+3nMAssay Description:Inhibition of p38alpha after 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Heinrich-Heine-UniversitäT
Curated by ChEMBL
Heinrich-Heine-UniversitäT
Curated by ChEMBL
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of human recombinant EGFR kinase expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of human recombinant CDK4/cyclin D1 kinase expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of human acetylcholinesterase using acetylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair
Affinity DataIC50: 1.48E+4nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 4.5 mins followed by substrate addition me...More data for this Ligand-Target Pair