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Found 507 with Last Name = 'brullo' and Initial = 'c'
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50436581(CHEMBL2397805)
Affinity DataKi:  5nMAssay Description:Binding affinity to recombinant wild type human Abl using abitide as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50176833(CHEMBL224545 | methyl 4-(4-methoxyphenethylamino)-...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176833(CHEMBL224545 | methyl 4-(4-methoxyphenethylamino)-...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranes in absence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176822(CHEMBL375154 | isopropyl 4-(4-methoxyphenethylamin...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50102904(CHEMBL3394091)
Affinity DataKi:  7nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176822(CHEMBL375154 | isopropyl 4-(4-methoxyphenethylamin...)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranes in absence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176833(CHEMBL224545 | methyl 4-(4-methoxyphenethylamino)-...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranes in presence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176822(CHEMBL375154 | isopropyl 4-(4-methoxyphenethylamin...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranes in presence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176835(CHEMBL223871 | ethyl 4-(4-methoxyphenethylamino)-1...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50102908(CHEMBL3393071)
Affinity DataKi:  10nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176815(CHEMBL225398 | ethyl 4-(4-fluorophenethylamino)-1-...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKi:  13nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKi:  13nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176838(1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamin...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50176815(CHEMBL225398 | ethyl 4-(4-fluorophenethylamino)-1-...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176842(CHEMBL224620 | ethyl 4-(2-fluorophenethylamino)-1-...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50176822(CHEMBL375154 | isopropyl 4-(4-methoxyphenethylamin...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50354489(CHEMBL1836680)
Affinity DataKi:  18nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176832(CHEMBL224909 | ethyl 4-(4-chlorophenethylamino)-1-...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50372736(CHEMBL270492)
Affinity DataKi:  20nMAssay Description:Binding affinity to human recombinant Abl by cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50436582(CHEMBL2397804)
Affinity DataKi:  21nMAssay Description:Binding affinity to recombinant wild type human Abl using abitide as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176855(1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamin...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176844(CHEMBL389405 | isopropyl 1-(2-chloro-2-phenylethyl...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50354480(CHEMBL1836678)
Affinity DataKi:  25nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50176835(CHEMBL223871 | ethyl 4-(4-methoxyphenethylamino)-1...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50354481(CHEMBL1836679)
Affinity DataKi:  25nMAssay Description:Inhibition human recombinant cSRC using KVEKIGEGTYGVVYK peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50176842(CHEMBL224620 | ethyl 4-(2-fluorophenethylamino)-1-...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50102872(CHEMBL3394083)
Affinity DataKi:  30nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176849(CHEMBL427255 | isopropyl 1-(2-chloro-2-phenylethyl...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176828(CHEMBL224097 | ethyl 4-(3-fluorophenethylamino)-1-...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176840(CHEMBL224083 | isopropyl 1-(2-chloro-2-phenylethyl...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50354485(CHEMBL412298)
Affinity DataKi:  40nMAssay Description:Binding affinity to human recombinant Abl by cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50354485(CHEMBL412298)
Affinity DataKi:  40nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50101585(CHEMBL3393986)
Affinity DataKi:  40nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50354485(CHEMBL412298)
Affinity DataKi:  40nMAssay Description:Binding affinity to recombinant wild type human Abl using abitide as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176825(CHEMBL389060 | isopropyl 4-(4-chlorophenethylamino...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50050937((S)-2-[(S)-2-((S)-2-Formylamino-4-methylsulfanyl-b...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]-fMLP from FPR in human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176839(CHEMBL223821 | isopropyl 4-(2-chlorophenethylamino...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176848(1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamin...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176834(CHEMBL224307 | cyclopropylmethyl 1-(2-chloro-2-phe...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50436570(CHEMBL2397818)
Affinity DataKi:  50nMAssay Description:Binding affinity to recombinant wild type human Abl using abitide as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176850(CHEMBL223450 | sec-butyl 1-(2-chloro-2-phenylethyl...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50436590(CHEMBL2397796)
Affinity DataKi:  55nMAssay Description:Binding affinity to recombinant wild type human Abl using abitide as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50436571(CHEMBL2397817)
Affinity DataKi:  60nMAssay Description:Binding affinity to recombinant wild type human Abl using abitide as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176843(CHEMBL374620 | sec-butyl 1-(2-chloro-2-phenylethyl...)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176852(1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamin...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50354484(CHEMBL1629808)
Affinity DataKi:  64nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50102878(CHEMBL3394082)
Affinity DataKi:  70nMAssay Description:Inhibition of human recombinant src kinase using KVEKIGEGTYGVVYK as substrate by filter binding assay in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50089575(CHEMBL3578214)
Affinity DataKi:  70nMAssay Description:Inhibition of human recombinant full-length Fyn using Src substrate peptide after 15 mins incubation by MicroBeta liquid scintillation counting analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176847(CHEMBL224313 | ethyl 4-(2-chlorophenethylamino)-1-...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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