TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 9.70nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 83nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 94nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 157nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 201nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 252nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 277nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMT: 2°CAssay Description:Phopholipase D1(PLD)enzymatic inhibition assay using PLD1.d311More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.5nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.40nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.5nMT: 2°CAssay Description:PLD in vitro enzymatic assay using phospholipase D1(PLD1).More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMT: 2°CAssay Description:Phopholipase D1(PLD)enzymatic inhibition assay using PLD1.d311More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of GFP-labelled human PLD2 HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMT: 2°CAssay Description:PLD in vitro enzymatic assay using phospholipase D2(PLD2).More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMT: 2°CAssay Description:Phopholipase D1(PLD)enzymatic inhibition assay using PLD1.d311More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of GFP-labelled human PLD2 HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of GFP-labelled human PLD2 HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibition of human PLD1 in Calu1 cellsMore data for this Ligand-Target Pair